IRIS
MASSAROTTI, Alberto
 Distribuzione geografica
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Continente #
EU - Europa 2.364
NA - Nord America 1.919
AS - Asia 600
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 4
AF - Africa 1
Totale 4.892
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Nazione #
US - Stati Uniti d'America 1.896
IE - Irlanda 660
IT - Italia 546
DE - Germania 352
SE - Svezia 323
UA - Ucraina 234
CN - Cina 149
SG - Singapore 119
FI - Finlandia 117
IN - India 115
TR - Turchia 102
HK - Hong Kong 78
GB - Regno Unito 34
CZ - Repubblica Ceca 27
FR - Francia 26
CA - Canada 21
IR - Iran 21
BE - Belgio 15
RU - Federazione Russa 9
NL - Olanda 6
EU - Europa 4
GR - Grecia 3
LT - Lituania 3
VN - Vietnam 3
AZ - Azerbaigian 2
DK - Danimarca 2
PH - Filippine 2
TH - Thailandia 2
AT - Austria 1
BR - Brasile 1
CL - Cile 1
EC - Ecuador 1
EE - Estonia 1
GE - Georgia 1
HN - Honduras 1
HU - Ungheria 1
IL - Israele 1
IQ - Iraq 1
JP - Giappone 1
KR - Corea 1
MA - Marocco 1
MD - Moldavia 1
MY - Malesia 1
NO - Norvegia 1
PA - Panama 1
PE - Perù 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
UZ - Uzbekistan 1
Totale 4.892
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Città #
Dublin 658
Jacksonville 457
Dearborn 237
Piemonte 154
Ann Arbor 138
Wilmington 113
Chandler 108
Singapore 89
Lawrence 83
Princeton 83
Ankara 80
Hong Kong 78
Beijing 62
San Mateo 58
Ashburn 41
Bremen 33
Vercelli 31
Andover 26
Brno 26
Helsinki 23
Milan 23
Torino 19
Munich 18
Monmouth Junction 17
Toronto 16
Brussels 15
Hefei 14
Turin 14
Kocaeli 13
Novara 13
Norwalk 11
Savignano Sul Panaro 11
Kunming 10
Santa Clara 10
Dallas 9
Grafing 9
Houston 9
Nanjing 9
Formigine 8
Leawood 8
Woodbridge 8
Fairfield 7
Strasbourg 7
Udine 7
Zanjan 7
Ardabil 6
Imola 6
Nanchang 6
Noicattaro 6
Seattle 6
Zola Predosa 6
Bologna 5
Cambridge 5
Cerano 5
Grignasco 5
Berlin 4
Boardman 4
Chengdu 4
Kecioeren 4
Legnano 4
London 4
Marigliano 4
Modena 4
Shenyang 4
Wuhan 4
Albano Laziale 3
Athens 3
Des Moines 3
Espoo 3
Forio 3
Fuzhou 3
Guangzhou 3
Hebei 3
Huzhou 3
Jinan 3
Montesarchio 3
Pavia 3
Rome 3
Sacramento 3
San Giuliano Milanese 3
Wachtberg 3
Zhengzhou 3
Baku 2
Cameriano 2
Ceppaloni 2
Curcuris 2
Dong Ket 2
Florence 2
Frankfurt am Main 2
Gorla Maggiore 2
Gunzenhausen 2
Hangzhou 2
Lyngby 2
Occimiano 2
Odalengo Grande 2
Redmond 2
Sesto Fiorentino 2
Vergiate 2
Wenzhou 2
Aachen 1
Totale 3.052
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Nome #
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors 146
Identification of a novel DGKa inhibitor for XLP-1 therapy by virtual screening 122
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement 115
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents 100
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity 98
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles 89
Capitolo 23. Istamina e agenti antistaminici 87
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe 86
Psychotropic Drugs Show Anticancer Activity by Disrupting Mitochondrial and Lysosomal Function 85
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 84
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents 83
Crystal structure of human nicotinic acid phosphoribosyltransferase 82
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors 82
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. 81
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY 80
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors 79
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)" 79
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs 79
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors 78
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase 78
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? 75
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 75
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues 74
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 73
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases 72
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors 72
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS 71
The Essential Medicinal Chemistry of Essential Medicines 70
Estrogenic analogues synthesized by click chemistry 68
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation 66
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis 65
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols 64
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement 62
Descriptive structure-separation relationship studies in chiral ligand-exchange chromatography 60
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus 59
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis 59
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis 58
Solution-phase parallel synthesis and biological evaluation of combretatriazoles 56
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones 56
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? 56
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy 56
Synthesis and cytotoxic evaluation of combretafurans, potential scaffolds for dual-action antitumoral agents 55
Sintesi e caratterizzazione di nuovi inibitori di DGKα 55
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring 54
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles 53
Parallel synthesis of “click” chalcones as antitubulin agents 53
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles 52
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination 51
Combretastatin analogues: from conformationally restricted compounds to virtual screening 51
Computational chemistry approaches for discovering new antitubulin compounds 51
ChemInform Abstract: Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Study (MFA 3D-QSAR) Unveil Novel Features of Bile Acid Recognition at TGR5 50
The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate 50
De novo computer-aided design of novel antiviral agents 49
Identification of Novel Antitubulin Agents by using a virtual screening approach based on a 7-point pharmacophore model of the tubulin colchi-site 49
Identification of an inhibitor of Chikungunya virus by virtual screening 48
Broad tuning of the human bitter taste receptor hTAS2R46 to various sesquiterpene lactones, clerodane and labdane diterpenoids, strychnine, and denatonium 48
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity 47
The hitchhiker's guide to the chemical-biological galaxy 47
Terpenoidi dall’assenzio marino (Artemisia arborescens) e loro interazione con il re-cettore dell’amaro 46
Synthesis and biological evaluation of combretatriazoles 45
Natural Product Fragments Preference for Protein Residues 45
Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Studies (MFA 3D-QSAR) of Bile Acids and Fexaramine Derivatives as Agonists of Farnesoid X Receptor (FXR) 44
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable 44
Medicinal Chemistry of Isocyanides 44
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 44
The tubulin colchicine domain: a molecular modelling perspective 43
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications 43
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives 43
Small molecule inhibitors of West Nile virus 42
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 42
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction 42
Photocatalytic Isocyanide-based Multicomponent Domino Cascade Towards the Stereoselective Formation of Iminofurans 42
Structural biology in antiviral drug discovery 40
Rational Discovery of (+) (S) Abscisic Acid as a Potential Antifungal Agent: a Repurposing Approach 40
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles 39
Synthesis and biological evaluation of combretatriazoles 39
The taste receptor hTAS2R46 as a general sensor for bitter sesquiterpene lactones 38
The metal face of protein tyrosine phosphatase 1B 38
Structure-property relationship studies in chiral ligand-exchange chromatography 35
Investigation of the Click-Chemical Space for Drug Design Using ZINClick 34
Molecular field analysis and quantitative structure-activity studies (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 receptor 32
PI(3,4)P2-mediated cytokinetic abscission prevents early senescence and cataract formation 30
Therapeutic peptides for the treatment of cystic fibrosis: Challenges and perspectives 28
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 17
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 9
In silico approach reveals N-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits 7
2‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition 6
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT2 5
A nonnatural peptide targeting the A-kinase anchoring function of PI3Kγ for therapeutic cAMP modulation in pulmonary cells 4
Totale 5.093
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Categoria #
all - tutte 25.674
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 25.674
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020736 0 0 0 0 0 139 206 41 90 148 97 15
2020/2021700 87 2 82 13 99 45 100 21 112 49 81 9
2021/2022612 56 17 53 67 26 11 53 20 35 44 84 146
2022/20231.379 95 76 83 26 77 111 61 82 685 9 40 34
2023/2024433 38 25 70 36 71 12 77 20 4 0 23 57
2024/2025238 37 29 77 25 69 1 0 0 0 0 0 0
Totale 5.093