IRIS
MASSAROTTI, Alberto
 Distribuzione geografica
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Continente #
EU - Europa 2.313
NA - Nord America 1.866
AS - Asia 534
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 3
AF - Africa 1
Totale 4.721
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Nazione #
US - Stati Uniti d'America 1.845
IE - Irlanda 660
IT - Italia 517
DE - Germania 348
SE - Svezia 323
UA - Ucraina 234
CN - Cina 148
IN - India 115
FI - Finlandia 112
TR - Turchia 97
HK - Hong Kong 74
SG - Singapore 68
GB - Regno Unito 28
CZ - Repubblica Ceca 27
FR - Francia 26
IR - Iran 21
CA - Canada 20
BE - Belgio 12
RU - Federazione Russa 9
NL - Olanda 5
EU - Europa 4
GR - Grecia 3
VN - Vietnam 3
DK - Danimarca 2
LT - Lituania 2
PH - Filippine 2
TH - Thailandia 2
AT - Austria 1
BR - Brasile 1
CL - Cile 1
EE - Estonia 1
HN - Honduras 1
IQ - Iraq 1
JP - Giappone 1
KR - Corea 1
MA - Marocco 1
MD - Moldavia 1
MY - Malesia 1
PE - Perù 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
Totale 4.721
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Città #
Dublin 658
Jacksonville 457
Dearborn 237
Piemonte 154
Ann Arbor 138
Wilmington 113
Chandler 108
Lawrence 83
Princeton 83
Ankara 79
Hong Kong 74
Beijing 62
San Mateo 58
Ashburn 41
Singapore 41
Bremen 33
Andover 26
Brno 26
Milan 23
Helsinki 21
Torino 19
Monmouth Junction 17
Munich 17
Toronto 15
Hefei 14
Turin 14
Kocaeli 13
Novara 13
Brussels 12
Norwalk 11
Savignano Sul Panaro 11
Kunming 10
Vercelli 10
Dallas 9
Grafing 9
Houston 9
Nanjing 9
Formigine 8
Leawood 8
Woodbridge 8
Fairfield 7
Strasbourg 7
Udine 7
Zanjan 7
Ardabil 6
Imola 6
Nanchang 6
Noicattaro 6
Seattle 6
Zola Predosa 6
Bologna 5
Cambridge 5
Cerano 5
Grignasco 5
Berlin 4
Boardman 4
Chengdu 4
Kecioeren 4
Legnano 4
Marigliano 4
Modena 4
Shenyang 4
Wuhan 4
Albano Laziale 3
Athens 3
Des Moines 3
Forio 3
Fuzhou 3
Guangzhou 3
Hebei 3
Huzhou 3
Jinan 3
Montesarchio 3
Pavia 3
Rome 3
Sacramento 3
San Giuliano Milanese 3
Wachtberg 3
Zhengzhou 3
Cameriano 2
Ceppaloni 2
Curcuris 2
Dong Ket 2
Florence 2
Gorla Maggiore 2
Gunzenhausen 2
Hangzhou 2
London 2
Lyngby 2
Occimiano 2
Odalengo Grande 2
Redmond 2
Sesto Fiorentino 2
Vergiate 2
Wenzhou 2
Aachen 1
Absecon 1
Augusta 1
Aveiro 1
Baghdad 1
Totale 2.956
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Nome #
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors 141
Identification of a novel DGKa inhibitor for XLP-1 therapy by virtual screening 121
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement 114
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity 97
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents 96
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles 87
Capitolo 23. Istamina e agenti antistaminici 85
Psychotropic Drugs Show Anticancer Activity by Disrupting Mitochondrial and Lysosomal Function 84
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe 83
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 83
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents 81
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. 80
Crystal structure of human nicotinic acid phosphoribosyltransferase 80
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors 80
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs 78
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY 78
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors 77
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)" 77
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors 77
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase 77
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 74
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues 72
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? 72
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases 71
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 71
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors 70
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS 69
The Essential Medicinal Chemistry of Essential Medicines 68
Estrogenic analogues synthesized by click chemistry 66
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation 64
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis 63
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols 62
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement 60
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis 58
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus 57
Descriptive structure-separation relationship studies in chiral ligand-exchange chromatography 57
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis 56
Solution-phase parallel synthesis and biological evaluation of combretatriazoles 54
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy 54
Sintesi e caratterizzazione di nuovi inibitori di DGKα 54
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones 53
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? 53
Synthesis and cytotoxic evaluation of combretafurans, potential scaffolds for dual-action antitumoral agents 52
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles 52
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring 52
Parallel synthesis of “click” chalcones as antitubulin agents 51
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles 50
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination 49
ChemInform Abstract: Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Study (MFA 3D-QSAR) Unveil Novel Features of Bile Acid Recognition at TGR5 49
The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate 49
De novo computer-aided design of novel antiviral agents 48
Combretastatin analogues: from conformationally restricted compounds to virtual screening 48
Computational chemistry approaches for discovering new antitubulin compounds 48
Broad tuning of the human bitter taste receptor hTAS2R46 to various sesquiterpene lactones, clerodane and labdane diterpenoids, strychnine, and denatonium 48
Identification of Novel Antitubulin Agents by using a virtual screening approach based on a 7-point pharmacophore model of the tubulin colchi-site 48
Identification of an inhibitor of Chikungunya virus by virtual screening 47
The hitchhiker's guide to the chemical-biological galaxy 47
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity 46
Terpenoidi dall’assenzio marino (Artemisia arborescens) e loro interazione con il re-cettore dell’amaro 45
Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Studies (MFA 3D-QSAR) of Bile Acids and Fexaramine Derivatives as Agonists of Farnesoid X Receptor (FXR) 44
Synthesis and biological evaluation of combretatriazoles 43
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable 43
Natural Product Fragments Preference for Protein Residues 43
Medicinal Chemistry of Isocyanides 43
The tubulin colchicine domain: a molecular modelling perspective 42
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives 42
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction 41
Photocatalytic Isocyanide-based Multicomponent Domino Cascade Towards the Stereoselective Formation of Iminofurans 41
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications 40
Small molecule inhibitors of West Nile virus 40
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 40
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 40
Structural biology in antiviral drug discovery 39
Rational Discovery of (+) (S) Abscisic Acid as a Potential Antifungal Agent: a Repurposing Approach 39
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles 38
The taste receptor hTAS2R46 as a general sensor for bitter sesquiterpene lactones 38
Synthesis and biological evaluation of combretatriazoles 38
The metal face of protein tyrosine phosphatase 1B 37
Structure-property relationship studies in chiral ligand-exchange chromatography 35
Investigation of the Click-Chemical Space for Drug Design Using ZINClick 32
Molecular field analysis and quantitative structure-activity studies (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 receptor 31
Therapeutic peptides for the treatment of cystic fibrosis: Challenges and perspectives 26
PI(3,4)P2-mediated cytokinetic abscission prevents early senescence and cataract formation 26
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 8
In silico approach reveals N-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits 4
2‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition 3
Totale 4.919
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Categoria #
all - tutte 22.704
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 22.704
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020981 0 5 76 9 155 139 206 41 90 148 97 15
2020/2021700 87 2 82 13 99 45 100 21 112 49 81 9
2021/2022612 56 17 53 67 26 11 53 20 35 44 84 146
2022/20231.379 95 76 83 26 77 111 61 82 685 9 40 34
2023/2024433 38 25 70 36 71 12 77 20 4 0 23 57
2024/202564 37 27 0 0 0 0 0 0 0 0 0 0
Totale 4.919