IRIS
MASSAROTTI, Alberto
 Distribuzione geografica
Salva come PNG Salva come JPEG
Continente #
EU - Europa 2.747
NA - Nord America 1.953
AS - Asia 922
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 4
AF - Africa 1
Totale 5.631
Salva come PNG Salva come JPEG
Nazione #
US - Stati Uniti d'America 1.929
IE - Irlanda 660
IT - Italia 628
DE - Germania 372
SE - Svezia 323
SG - Singapore 256
HK - Hong Kong 252
UA - Ucraina 239
RU - Federazione Russa 165
CN - Cina 149
FI - Finlandia 123
IN - India 115
TR - Turchia 102
EE - Estonia 101
GB - Regno Unito 35
FR - Francia 29
CZ - Repubblica Ceca 27
CA - Canada 22
IR - Iran 21
BE - Belgio 15
ID - Indonesia 10
AT - Austria 8
NL - Olanda 8
EU - Europa 4
LT - Lituania 4
GR - Grecia 3
VN - Vietnam 3
AZ - Azerbaigian 2
DK - Danimarca 2
GE - Georgia 2
PH - Filippine 2
TH - Thailandia 2
BR - Brasile 1
CL - Cile 1
EC - Ecuador 1
HN - Honduras 1
HU - Ungheria 1
IL - Israele 1
IQ - Iraq 1
JP - Giappone 1
KR - Corea 1
MA - Marocco 1
MD - Moldavia 1
MY - Malesia 1
NO - Norvegia 1
PA - Panama 1
PE - Perù 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
UZ - Uzbekistan 1
Totale 5.631
Salva come PNG Salva come JPEG
Città #
Dublin 658
Jacksonville 457
Hong Kong 252
Dearborn 237
Piemonte 154
Ann Arbor 138
Singapore 119
Wilmington 113
Chandler 108
Lawrence 83
Princeton 83
Ankara 80
Novara 78
Moscow 77
Beijing 62
San Mateo 58
Ashburn 42
Bremen 33
Vercelli 32
Helsinki 29
Andover 26
Brno 26
Milan 26
Torino 19
Munich 18
Monmouth Junction 17
Toronto 17
Brussels 15
Hefei 14
Turin 14
Kocaeli 13
Norwalk 11
Savignano Sul Panaro 11
Kunming 10
Santa Clara 10
Dallas 9
Grafing 9
Houston 9
Nanjing 9
Formigine 8
Leawood 8
Woodbridge 8
Fairfield 7
Strasbourg 7
Udine 7
Zanjan 7
Ardabil 6
Imola 6
Nanchang 6
Noicattaro 6
Nuremberg 6
Seattle 6
Zola Predosa 6
Bologna 5
Cambridge 5
Cerano 5
Grignasco 5
Berlin 4
Boardman 4
Chengdu 4
Jakarta 4
Kecioeren 4
Legnano 4
London 4
Marigliano 4
Modena 4
Rome 4
Shenyang 4
Wuhan 4
Albano Laziale 3
Athens 3
Carmagnola 3
Des Moines 3
Espoo 3
Falkenstein 3
Forio 3
Fuzhou 3
Guangzhou 3
Hebei 3
Huzhou 3
Jinan 3
Montesarchio 3
Pavia 3
Sacramento 3
San Giuliano Milanese 3
Vienna 3
Wachtberg 3
Zhengzhou 3
Baku 2
Cameriano 2
Casnate Con Bernate 2
Ceppaloni 2
Curcuris 2
Dong Ket 2
Florence 2
Frankfurt am Main 2
Gorla Maggiore 2
Gunzenhausen 2
Hangzhou 2
Los Angeles 2
Totale 3.419
Salva come PNG Salva come JPEG
Nome #
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors 169
Identification of a novel DGKa inhibitor for XLP-1 therapy by virtual screening 130
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement 120
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents 106
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity 104
null 100
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles 96
Psychotropic Drugs Show Anticancer Activity by Disrupting Mitochondrial and Lysosomal Function 95
Capitolo 23. Istamina e agenti antistaminici 94
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe 92
Crystal structure of human nicotinic acid phosphoribosyltransferase 89
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors 88
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents 87
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)" 87
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs 87
Essential Medicinal Chemistry of Essential Medicines 87
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors 86
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. 85
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors 85
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 85
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? 83
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY 83
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase 82
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors 81
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases 79
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 79
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues 78
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS 78
Estrogenic analogues synthesized by click chemistry 76
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis 76
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation 72
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement 70
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols 68
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy 66
Synthesis and cytotoxic evaluation of combretafurans, potential scaffolds for dual-action antitumoral agents 65
Descriptive structure-separation relationship studies in chiral ligand-exchange chromatography 65
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis 65
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus 64
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis 64
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? 64
Parallel synthesis of “click” chalcones as antitubulin agents 64
Solution-phase parallel synthesis and biological evaluation of combretatriazoles 63
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles 63
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles 62
The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate 62
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring 61
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles 61
Sintesi e caratterizzazione di nuovi inibitori di DGKα 61
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones 60
Computational chemistry approaches for discovering new antitubulin compounds 59
Identification of Novel Antitubulin Agents by using a virtual screening approach based on a 7-point pharmacophore model of the tubulin colchi-site 58
The hitchhiker's guide to the chemical-biological galaxy 58
Medicinal Chemistry of Isocyanides 57
De novo computer-aided design of novel antiviral agents 56
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination 56
ChemInform Abstract: Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Study (MFA 3D-QSAR) Unveil Novel Features of Bile Acid Recognition at TGR5 56
Combretastatin analogues: from conformationally restricted compounds to virtual screening 55
Broad tuning of the human bitter taste receptor hTAS2R46 to various sesquiterpene lactones, clerodane and labdane diterpenoids, strychnine, and denatonium 55
PI(3,4)P2-mediated cytokinetic abscission prevents early senescence and cataract formation 54
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives 53
Natural Product Fragments Preference for Protein Residues 53
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications 52
Synthesis and biological evaluation of combretatriazoles 52
Terpenoidi dall’assenzio marino (Artemisia arborescens) e loro interazione con il re-cettore dell’amaro 52
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable 52
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity 52
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 52
Identification of an inhibitor of Chikungunya virus by virtual screening 51
Synthesis and biological evaluation of combretatriazoles 51
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 50
Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Studies (MFA 3D-QSAR) of Bile Acids and Fexaramine Derivatives as Agonists of Farnesoid X Receptor (FXR) 50
Photocatalytic Isocyanide-based Multicomponent Domino Cascade Towards the Stereoselective Formation of Iminofurans 50
The tubulin colchicine domain: a molecular modelling perspective 49
Small molecule inhibitors of West Nile virus 49
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction 48
Rational Discovery of (+) (S) Abscisic Acid as a Potential Antifungal Agent: a Repurposing Approach 48
The metal face of protein tyrosine phosphatase 1B 46
Structural biology in antiviral drug discovery 45
Therapeutic peptides for the treatment of cystic fibrosis: Challenges and perspectives 44
The taste receptor hTAS2R46 as a general sensor for bitter sesquiterpene lactones 43
Structure-property relationship studies in chiral ligand-exchange chromatography 41
Investigation of the Click-Chemical Space for Drug Design Using ZINClick 40
Molecular field analysis and quantitative structure-activity studies (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 receptor 37
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 33
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 31
A nonnatural peptide targeting the A-kinase anchoring function of PI3Kγ for therapeutic cAMP modulation in pulmonary cells 22
2‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition 20
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT2 15
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 14
In silico approach reveals N-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits 12
Totale 5.858
Salva come PNG Salva come JPEG
Categoria #
all - tutte 29.743
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 29.743
Salva come PNG Salva come JPEG


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020260 0 0 0 0 0 0 0 0 0 148 97 15
2020/2021700 87 2 82 13 99 45 100 21 112 49 81 9
2021/2022612 56 17 53 67 26 11 53 20 35 44 84 146
2022/20231.379 95 76 83 26 77 111 61 82 685 9 40 34
2023/2024433 38 25 70 36 71 12 77 20 4 0 23 57
2024/20251.003 37 29 77 25 69 154 122 114 239 137 0 0
Totale 5.858