IRIS
MASSAROTTI, Alberto
 Distribuzione geografica
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Continente #
EU - Europa 3.042
NA - Nord America 2.613
AS - Asia 1.755
SA - Sud America 282
AF - Africa 36
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 1
Totale 7.733
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Nazione #
US - Stati Uniti d'America 2.538
IT - Italia 678
SG - Singapore 661
IE - Irlanda 660
DE - Germania 452
SE - Svezia 335
CN - Cina 323
HK - Hong Kong 272
UA - Ucraina 248
BR - Brasile 213
RU - Federazione Russa 169
FI - Finlandia 148
IN - India 137
VN - Vietnam 126
TR - Turchia 111
EE - Estonia 101
GB - Regno Unito 69
FR - Francia 57
CA - Canada 51
AR - Argentina 32
CZ - Repubblica Ceca 27
PL - Polonia 24
BD - Bangladesh 22
IR - Iran 21
JP - Giappone 19
BE - Belgio 17
ID - Indonesia 16
EC - Ecuador 15
MX - Messico 14
NL - Olanda 13
ZA - Sudafrica 12
BJ - Benin 11
ES - Italia 11
AT - Austria 10
LT - Lituania 10
KR - Corea 8
IQ - Iraq 6
VE - Venezuela 6
AZ - Azerbaigian 5
MA - Marocco 5
CL - Cile 4
CO - Colombia 4
EU - Europa 4
IL - Israele 4
PK - Pakistan 4
UZ - Uzbekistan 4
DO - Repubblica Dominicana 3
GR - Grecia 3
PE - Perù 3
PY - Paraguay 3
SA - Arabia Saudita 3
AE - Emirati Arabi Uniti 2
DK - Danimarca 2
GE - Georgia 2
PH - Filippine 2
PR - Porto Rico 2
TH - Thailandia 2
TN - Tunisia 2
AL - Albania 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
BO - Bolivia 1
CI - Costa d'Avorio 1
DZ - Algeria 1
ET - Etiopia 1
GT - Guatemala 1
HN - Honduras 1
HU - Ungheria 1
JM - Giamaica 1
JO - Giordania 1
KE - Kenya 1
KZ - Kazakistan 1
LV - Lettonia 1
MD - Moldavia 1
MR - Mauritania 1
MY - Malesia 1
NO - Norvegia 1
OM - Oman 1
PA - Panama 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
SV - El Salvador 1
TG - Togo 1
UY - Uruguay 1
Totale 7.733
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Città #
Dublin 658
Jacksonville 457
Hong Kong 272
Dearborn 237
Singapore 190
Beijing 164
Piemonte 154
Ashburn 149
Ann Arbor 138
Wilmington 113
Chandler 108
Novara 93
Ankara 86
Lawrence 83
Princeton 83
Los Angeles 77
Moscow 77
Munich 68
San Mateo 58
Ho Chi Minh City 55
New York 46
Vercelli 42
Bremen 33
Dallas 31
Helsinki 31
Milan 30
São Paulo 30
Buffalo 29
Andover 26
Brno 26
Redondo Beach 24
Turku 23
Turin 22
Hanoi 21
Frankfurt am Main 20
Santa Clara 20
Toronto 20
Warsaw 20
Torino 19
Tokyo 18
Chicago 17
Monmouth Junction 17
Houston 16
Montreal 16
Brussels 15
Denver 14
Hefei 14
Kocaeli 13
Phoenix 12
Poplar 12
Seattle 12
Stockholm 12
Cotonou 11
London 11
Norwalk 11
Orem 11
Savignano Sul Panaro 11
Tianjin 11
Atlanta 10
Chennai 10
Johannesburg 10
Kunming 10
Boston 9
Brooklyn 9
Grafing 9
Nanjing 9
Formigine 8
Leawood 8
Woodbridge 8
Fairfield 7
Nuremberg 7
San Francisco 7
Seoul 7
Strasbourg 7
Udine 7
Zanjan 7
Ardabil 6
Dhaka 6
Haiphong 6
Imola 6
Mexico City 6
Nanchang 6
Noicattaro 6
Reston 6
Rome 6
Zola Predosa 6
Amsterdam 5
Baku 5
Biên Hòa 5
Bologna 5
Cambridge 5
Cerano 5
Grignasco 5
Jakarta 5
Quito 5
Rio de Janeiro 5
Augusta 4
Berlin 4
Bexley 4
Boardman 4
Totale 4.362
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Nome #
Small molecule inhibitors of West Nile virus 213
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors 194
Identification of a novel DGKa inhibitor for XLP-1 therapy by virtual screening 162
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement 158
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents 139
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe 131
Psychotropic Drugs Show Anticancer Activity by Disrupting Mitochondrial and Lysosomal Function 129
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity 127
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents 126
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? 124
Crystal structure of human nicotinic acid phosphoribosyltransferase 121
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 117
Capitolo 23. Istamina e agenti antistaminici 116
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. 114
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 113
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors 112
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs 111
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase 111
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors 110
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement 109
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles 108
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors 106
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)" 105
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY 102
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones 101
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors 100
null 100
Estrogenic analogues synthesized by click chemistry 99
Combretastatin analogues: from conformationally restricted compounds to virtual screening 98
Parallel synthesis of “click” chalcones as antitubulin agents 97
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues 96
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases 95
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis 94
Essential Medicinal Chemistry of Essential Medicines 93
De novo computer-aided design of novel antiviral agents 92
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation 90
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination 87
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis 87
Medicinal Chemistry of Isocyanides 87
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus 86
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? 85
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS 85
Broad tuning of the human bitter taste receptor hTAS2R46 to various sesquiterpene lactones, clerodane and labdane diterpenoids, strychnine, and denatonium 84
The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate 84
Solution-phase parallel synthesis and biological evaluation of combretatriazoles 83
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols 83
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy 83
Natural Product Fragments Preference for Protein Residues 83
ChemInform Abstract: Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Study (MFA 3D-QSAR) Unveil Novel Features of Bile Acid Recognition at TGR5 83
Descriptive structure-separation relationship studies in chiral ligand-exchange chromatography 82
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles 81
Computational chemistry approaches for discovering new antitubulin compounds 80
Sintesi e caratterizzazione di nuovi inibitori di DGKα 80
Synthesis and cytotoxic evaluation of combretafurans, potential scaffolds for dual-action antitumoral agents 78
The hitchhiker's guide to the chemical-biological galaxy 77
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles 75
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis 74
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 74
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles 73
Identification of an inhibitor of Chikungunya virus by virtual screening 72
Synthesis and biological evaluation of combretatriazoles 72
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable 72
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications 66
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring 66
A nonnatural peptide targeting the A-kinase anchoring function of PI3Kγ for therapeutic cAMP modulation in pulmonary cells 64
Structure-property relationship studies in chiral ligand-exchange chromatography 64
The metal face of protein tyrosine phosphatase 1B 63
PI(3,4)P2-mediated cytokinetic abscission prevents early senescence and cataract formation 63
The taste receptor hTAS2R46 as a general sensor for bitter sesquiterpene lactones 62
Rational Discovery of (+) (S) Abscisic Acid as a Potential Antifungal Agent: a Repurposing Approach 62
Identification of Novel Antitubulin Agents by using a virtual screening approach based on a 7-point pharmacophore model of the tubulin colchi-site 62
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 61
Synthesis and biological evaluation of combretatriazoles 61
Terpenoidi dall’assenzio marino (Artemisia arborescens) e loro interazione con il re-cettore dell’amaro 61
Photocatalytic Isocyanide-based Multicomponent Domino Cascade Towards the Stereoselective Formation of Iminofurans 61
2‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition 61
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity 60
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives 58
The tubulin colchicine domain: a molecular modelling perspective 57
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 57
Therapeutic peptides for the treatment of cystic fibrosis: Challenges and perspectives 57
Molecular Field Analysis and 3D-Quantitative Structure-Activity Relationship Studies (MFA 3D-QSAR) of Bile Acids and Fexaramine Derivatives as Agonists of Farnesoid X Receptor (FXR) 56
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction 54
Investigation of the Click-Chemical Space for Drug Design Using ZINClick 53
Structural biology in antiviral drug discovery 52
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 51
Molecular field analysis and quantitative structure-activity studies (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 receptor 47
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 45
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT2 36
Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity 32
Acute Myeloid Leukemia: A Key Role of DGKα and DGKζ in Cell Viability 29
In silico approach reveals N-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits 20
Modulators of Diacylglycerol Kinase Activity: A Review of Advances and Challenges 19
Totale 7.963
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Categoria #
all - tutte 38.214
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 38.214
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021417 0 0 0 0 0 45 100 21 112 49 81 9
2021/2022612 56 17 53 67 26 11 53 20 35 44 84 146
2022/20231.379 95 76 83 26 77 111 61 82 685 9 40 34
2023/2024433 38 25 70 36 71 12 77 20 4 0 23 57
2024/20251.470 37 29 77 25 69 154 122 114 239 184 138 282
2025/20261.638 197 107 289 562 428 55 0 0 0 0 0 0
Totale 7.963