SORBA, Giovanni
SORBA, Giovanni
Dipartimento di Scienze del Farmaco
[3-(1H-Imidazol-4-yl)propyl]guanidines containing furoxan moieties: a New Class of H3-Antagonists endowed with NO-Donor properties
2003-01-01 Bertinaria, M.; DI STILO, A.; Tosco, P.; Sorba, Giovanni; Poli, E.; Pozzoli, C.; Coruzzi, G.; Fruttero, R.; Gasco, A.
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents
2013-01-01 Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
2018-01-01 Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia
A new furoxan NO-donor rabeprazole derivative and related compounds
2003-01-01 Sorba, Giovanni; Galli, Ubaldina; Cena, C.; Fruttero, R.; Gasco, A.; Morini, G.; Adami, M.; Coruzzi, G.; Brenciaglia, M. I.; Dubini, F.
A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry
2010-01-01 Colombano, Giampiero; Travelli, Cristina; Galli, Ubaldina; Caldarelli, Antonio; Chini, Mg; Canonico, Pier Luigi; Sorba, Giovanni; Bifulco, G; Tron, Gian Cesare; Genazzani, Armando
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination
2010-01-01 Giustiniano, M; Pirali, Tracey; Massarotti, Alberto; Biletta, B; Novellino, E; Campiglia, P; Sorba, Giovanni; Tron, Gian Cesare
Anti-Helicobacter pylori agents endowed with H2-antagonist properties
2001-01-01 Sorba, Giovanni; Bertinaria, M.; DI STILO, A.; Gasco, A.; Brenciaglia, M. I.; Dubini, F.
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?
2014-01-01 Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare
Capitolo 23. Istamina e agenti antistaminici
2014-01-01 Sorba, Giovanni; Massarotti, Alberto
Click chemistry reactions in medicinal chemistry: applications of the 1,3-dipolar cycloaddition between azides and alkynes
2008-01-01 Tron, Gian Cesare; Pirali, Tracey; Billington, Richard Andrew; Canonico, Pier Luigi; Sorba, Giovanni; Genazzani, Armando
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus
2013-01-01 Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A.
De novo computer-aided design of novel antiviral agents
2012-01-01 Massarotti, Alberto; Coluccia, A; Sorba, Giovanni; Silvestri, R; Brancale, A.
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare
Design, synthesis, and biological evaluation of new (2E,6E)-10-(dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol ethers as inhibitors of human and Trypanosoma cruzi oxidosqualene cyclase
2007-01-01 Galli, Ubaldina; Oliaro Bosso, S; Taramino, S; Venegoni, S; Pastore, E; Tron, Gian Cesare; Balliano, G; Viola, F; Sorba, Giovanni
Essential role of the p110β subunit of phosphoinositide 3-OH kinase in male fertility
2010-01-01 Ciraolo, Elisa; Morello, Fulvio; Hobbs, ; Robin, M; Wolf, Frieder; Marone, Romina; Iezzi, Manuela; Lu, Xiaoyun; Mengozzi, Giulio; Altruda, Fiorella; Sorba, Giovanni; Giovanni, Guan; Kaomei, Pandolfi; Pier, Paolo; Wymann, ; Matthias, P; Hirsch, Emilio
Estrogenic analogues synthesized by click chemistry
2007-01-01 Pirali, Tracey; Gatti, S; DI BRISCO, R; Tacchi, Sara; Zaninetti, Roberta; Brunelli, Elisa; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Moro, Laura; Genazzani, Armando; Tron, Gian Cesare; Billington, Richard Andrew
Furoxan Analogues of the Histamine H3 receptor antagonist imoproxifan and related furazan derivatives
2005-01-01 Tosco, P.; Bertinaria, M.; DI STILO, A.; Cena, C.; Sorba, Giovanni; Fruttero, R.; Gasco, A.
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors
2011-01-01 Guasconi, M; Lu, X; Massarotti, Alberto; Caldarelli, Antonio; Ciraolo, E; Tron, Gian Cesare; Hirsch, E; Sorba, Giovanni; Pirali, Tracey
Icilio Guareschi and his amazing “1897 reaction”
2021-01-01 Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G.
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| [3-(1H-Imidazol-4-yl)propyl]guanidines containing furoxan moieties: a New Class of H3-Antagonists endowed with NO-Donor properties | 1-gen-2003 | Bertinaria, M.; DI STILO, A.; Tosco, P.; Sorba, Giovanni; Poli, E.; Pozzoli, C.; Coruzzi, G.; Fruttero, R.; Gasco, A. | |
| A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents | 1-gen-2013 | Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey | |
| A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies | 1-gen-2018 | Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia | |
| A new furoxan NO-donor rabeprazole derivative and related compounds | 1-gen-2003 | Sorba, Giovanni; Galli, Ubaldina; Cena, C.; Fruttero, R.; Gasco, A.; Morini, G.; Adami, M.; Coruzzi, G.; Brenciaglia, M. I.; Dubini, F. | |
| A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry | 1-gen-2010 | Colombano, Giampiero; Travelli, Cristina; Galli, Ubaldina; Caldarelli, Antonio; Chini, Mg; Canonico, Pier Luigi; Sorba, Giovanni; Bifulco, G; Tron, Gian Cesare; Genazzani, Armando | |
| A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination | 1-gen-2010 | Giustiniano, M; Pirali, Tracey; Massarotti, Alberto; Biletta, B; Novellino, E; Campiglia, P; Sorba, Giovanni; Tron, Gian Cesare | |
| Anti-Helicobacter pylori agents endowed with H2-antagonist properties | 1-gen-2001 | Sorba, Giovanni; Bertinaria, M.; DI STILO, A.; Gasco, A.; Brenciaglia, M. I.; Dubini, F. | |
| Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? | 1-gen-2014 | Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare | |
| Capitolo 23. Istamina e agenti antistaminici | 1-gen-2014 | Sorba, Giovanni; Massarotti, Alberto | |
| Click chemistry reactions in medicinal chemistry: applications of the 1,3-dipolar cycloaddition between azides and alkynes | 1-gen-2008 | Tron, Gian Cesare; Pirali, Tracey; Billington, Richard Andrew; Canonico, Pier Luigi; Sorba, Giovanni; Genazzani, Armando | |
| Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus | 1-gen-2013 | Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A. | |
| De novo computer-aided design of novel antiviral agents | 1-gen-2012 | Massarotti, Alberto; Coluccia, A; Sorba, Giovanni; Silvestri, R; Brancale, A. | |
| Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 1-gen-2015 | Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare | |
| Design, synthesis, and biological evaluation of new (2E,6E)-10-(dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol ethers as inhibitors of human and Trypanosoma cruzi oxidosqualene cyclase | 1-gen-2007 | Galli, Ubaldina; Oliaro Bosso, S; Taramino, S; Venegoni, S; Pastore, E; Tron, Gian Cesare; Balliano, G; Viola, F; Sorba, Giovanni | |
| Essential role of the p110β subunit of phosphoinositide 3-OH kinase in male fertility | 1-gen-2010 | Ciraolo, Elisa; Morello, Fulvio; Hobbs, ; Robin, M; Wolf, Frieder; Marone, Romina; Iezzi, Manuela; Lu, Xiaoyun; Mengozzi, Giulio; Altruda, Fiorella; Sorba, Giovanni; Giovanni, Guan; Kaomei, Pandolfi; Pier, Paolo; Wymann, ; Matthias, P; Hirsch, Emilio | |
| Estrogenic analogues synthesized by click chemistry | 1-gen-2007 | Pirali, Tracey; Gatti, S; DI BRISCO, R; Tacchi, Sara; Zaninetti, Roberta; Brunelli, Elisa; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Moro, Laura; Genazzani, Armando; Tron, Gian Cesare; Billington, Richard Andrew | |
| Furoxan Analogues of the Histamine H3 receptor antagonist imoproxifan and related furazan derivatives | 1-gen-2005 | Tosco, P.; Bertinaria, M.; DI STILO, A.; Cena, C.; Sorba, Giovanni; Fruttero, R.; Gasco, A. | |
| Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors | 1-gen-2011 | Guasconi, M; Lu, X; Massarotti, Alberto; Caldarelli, Antonio; Ciraolo, E; Tron, Gian Cesare; Hirsch, E; Sorba, Giovanni; Pirali, Tracey | |
| Icilio Guareschi and his amazing “1897 reaction” | 1-gen-2021 | Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G. | |
| Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 1-gen-2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare |