Sfoglia per Autore
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare
A fast route for the synthesis of tetrazolyl oximes by a novel multicomponent reaction between Z-chlorooximes, isocyanides and trimethylsilyl azide
2017-01-01 Mariateresa, Giustiniano; Sveva, Pelliccia; Ana Belen, Muñoz garcia; Michele, Pavone; Bruno, Pagano; Galli, Ubaldina; Ettore, Novellino; Tron, Gian Cesare
A Successful Replacement of Phenols with Isocyanides in the Bargellini Reaction: Synthesis of 3-Carboxamido-Isobutyric Acids
2016-01-01 Giustiniano, Mariateresa; Pelliccia, Sveva; Galli, Ubaldina; Amato, Jussara; Travagin, Fabio; Novellino, Ettore; Tron, Gian Cesare
Nicotinamide phosphoribosyltransferase (NAMPT/PBEF/visfatin): a new cytokine in tumour progression
2015-01-01 Grolla, Ambra; Torretta, Simone; Travelli, Cristina; Amoruso, Angela; Orsomando, G.; Galli, Ubaldina; Canonico, Pier Luigi; Genazzani, Armando
Nicotinamide phosphoribosyltransferase (NAMPT) inhibitors: novel modulators of antitumor immunity
2015-01-01 Travelli, Cristina; Morlacchi, S.; Grolla, Ambra; Galli, Ubaldina; Tron, Gian Cesare; Sangaletti, S.; Colombo, M. P.; Canonico, Pier Luigi; Genazzani, Armando; Sica, Antonio
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement
2015-01-01 Theeramunkong, S.; Galli, Ubaldina; Grolla, Ambra; Caldarelli, Antonio; Travelli, Cristina; Massarotti, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; Genazzani, Armando; Tron, Gian Cesare
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors
2015-01-01 Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare
Nicotinamide phosphoribosyltransferase (NAMPT/PBEF/visfatin): a new cytokine in tumour progression
2015-01-01 Grolla, Ambra; Torretta, Simone; Travelli, Cristina; Gnemmi, Ilaria; Amoruso, Angela; Orsomando, G.; Galli, Ubaldina; Canonico, Pier Luigi; Genazzani, Armando
Combretabenzodiazepines: a novel class of antitubulin agents
2015-01-01 Galli, Ubaldina; Travelli, Cristina; Genazzani, Armando; Tron, Gian Cesare
Nicotinamide phosphoribosyltransferase (NAMPT) inhibitors are novel modulators of myeloid-derived suppressor cells
2015-01-01 Travelli, Cristina; Galli, Ubaldina; Tron, Gian Cesare; Sangaletti, S.; Canonico, Pier Luigi; Sica, Antonio; Genazzani, Armando
Reaction Between (Z)-Arylchlorooximes and alpha-Isocyanoacetamides: a Procedure For The Synthesis of Aryl-alpha-Ketoamide amides
2014-01-01 Giustiniano, Mariateresa; Mercalli, Valentina; Cassese, Hilde; Di Maro, Salvatore; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare
Inhibitors of Nicotinamide Phosphoribosyltransferase, compositions, products and uses thereof.
2014-01-01 Genazzani Armando, A.; Tron, Gian Cesare; Galli, Ubaldina; Travelli, Cristina; Cuzzocrea, Salvatore; Grosa, Giorgio; Sorba, Giovanni; Canonico Pier, Luigi
“Sirtuins, new potential targets for HIV-therapy”
2013-01-01 I., Gnemmi; B., Riva; M., Di Rosa; G., Nunnari; Galli, Ubaldina; A. A., Genazzani; Condorelli, Fabrizio; P. L., Canonico
Nicotinamide Phosphorybosyltransferase (NAMPT) Inhibitors are Novel Modulator of Cancer-Related Inflammation
2013-01-01 C., Travelli; S., Morlacchi; Galli, Ubaldina; Sica, Antonio; P. L., Canonico; A. A., Genazzani
Nicotinamide phosphoribosyltransferase (NAMPT) is over-expressed in melanoma lesions.
2013-01-01 Maldi, E; Travelli, Cristina; Caldarelli, Antonio; Agazzone, N; Cintura, S; Galli, Ubaldina; Scatolini, M; Ostano, P; Miglino, B; Chiorino, G; Boldorini, Renzo Luciano; Genazzani, Armando
“Visfatin: new role as cytokine in tumour microenviroment”
2013-01-01 A. A, Grolla; S., Torretta; A., Amoruso; Galli, Ubaldina; G., Orsomando; C., Travelli; P. L., Canonico; A. A., Genazzani
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors.
2013-01-01 Galli, Ubaldina; Travelli, Cristina; Massarotti, Alberto; Fakhfouri, G; Rahimian, R; Tron, Gian Cesare; Genazzani, Armando
“Synthesis and in vitro evaluation of tetrasubstituted pyridines as potential PI3Ks inhibitors”
2013-01-01 Galli, Ubaldina; E., Ciraolo; E., Hirsch; Sorba, Giovanni; Tron, Gian Cesare
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases
2012-01-01 Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 1-gen-2017 | Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare | |
A fast route for the synthesis of tetrazolyl oximes by a novel multicomponent reaction between Z-chlorooximes, isocyanides and trimethylsilyl azide | 1-gen-2017 | Mariateresa, Giustiniano; Sveva, Pelliccia; Ana Belen, Muñoz garcia; Michele, Pavone; Bruno, Pagano; Galli, Ubaldina; Ettore, Novellino; Tron, Gian Cesare | |
A Successful Replacement of Phenols with Isocyanides in the Bargellini Reaction: Synthesis of 3-Carboxamido-Isobutyric Acids | 1-gen-2016 | Giustiniano, Mariateresa; Pelliccia, Sveva; Galli, Ubaldina; Amato, Jussara; Travagin, Fabio; Novellino, Ettore; Tron, Gian Cesare | |
Nicotinamide phosphoribosyltransferase (NAMPT/PBEF/visfatin): a new cytokine in tumour progression | 1-gen-2015 | Grolla, Ambra; Torretta, Simone; Travelli, Cristina; Amoruso, Angela; Orsomando, G.; Galli, Ubaldina; Canonico, Pier Luigi; Genazzani, Armando | |
Nicotinamide phosphoribosyltransferase (NAMPT) inhibitors: novel modulators of antitumor immunity | 1-gen-2015 | Travelli, Cristina; Morlacchi, S.; Grolla, Ambra; Galli, Ubaldina; Tron, Gian Cesare; Sangaletti, S.; Colombo, M. P.; Canonico, Pier Luigi; Genazzani, Armando; Sica, Antonio | |
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement | 1-gen-2015 | Theeramunkong, S.; Galli, Ubaldina; Grolla, Ambra; Caldarelli, Antonio; Travelli, Cristina; Massarotti, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; Genazzani, Armando; Tron, Gian Cesare | |
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 1-gen-2015 | Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare | |
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors | 1-gen-2015 | Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare | |
Nicotinamide phosphoribosyltransferase (NAMPT/PBEF/visfatin): a new cytokine in tumour progression | 1-gen-2015 | Grolla, Ambra; Torretta, Simone; Travelli, Cristina; Gnemmi, Ilaria; Amoruso, Angela; Orsomando, G.; Galli, Ubaldina; Canonico, Pier Luigi; Genazzani, Armando | |
Combretabenzodiazepines: a novel class of antitubulin agents | 1-gen-2015 | Galli, Ubaldina; Travelli, Cristina; Genazzani, Armando; Tron, Gian Cesare | |
Nicotinamide phosphoribosyltransferase (NAMPT) inhibitors are novel modulators of myeloid-derived suppressor cells | 1-gen-2015 | Travelli, Cristina; Galli, Ubaldina; Tron, Gian Cesare; Sangaletti, S.; Canonico, Pier Luigi; Sica, Antonio; Genazzani, Armando | |
Reaction Between (Z)-Arylchlorooximes and alpha-Isocyanoacetamides: a Procedure For The Synthesis of Aryl-alpha-Ketoamide amides | 1-gen-2014 | Giustiniano, Mariateresa; Mercalli, Valentina; Cassese, Hilde; Di Maro, Salvatore; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare | |
Inhibitors of Nicotinamide Phosphoribosyltransferase, compositions, products and uses thereof. | 1-gen-2014 | Genazzani Armando, A.; Tron, Gian Cesare; Galli, Ubaldina; Travelli, Cristina; Cuzzocrea, Salvatore; Grosa, Giorgio; Sorba, Giovanni; Canonico Pier, Luigi | |
“Sirtuins, new potential targets for HIV-therapy” | 1-gen-2013 | I., Gnemmi; B., Riva; M., Di Rosa; G., Nunnari; Galli, Ubaldina; A. A., Genazzani; Condorelli, Fabrizio; P. L., Canonico | |
Nicotinamide Phosphorybosyltransferase (NAMPT) Inhibitors are Novel Modulator of Cancer-Related Inflammation | 1-gen-2013 | C., Travelli; S., Morlacchi; Galli, Ubaldina; Sica, Antonio; P. L., Canonico; A. A., Genazzani | |
Nicotinamide phosphoribosyltransferase (NAMPT) is over-expressed in melanoma lesions. | 1-gen-2013 | Maldi, E; Travelli, Cristina; Caldarelli, Antonio; Agazzone, N; Cintura, S; Galli, Ubaldina; Scatolini, M; Ostano, P; Miglino, B; Chiorino, G; Boldorini, Renzo Luciano; Genazzani, Armando | |
“Visfatin: new role as cytokine in tumour microenviroment” | 1-gen-2013 | A. A, Grolla; S., Torretta; A., Amoruso; Galli, Ubaldina; G., Orsomando; C., Travelli; P. L., Canonico; A. A., Genazzani | |
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. | 1-gen-2013 | Galli, Ubaldina; Travelli, Cristina; Massarotti, Alberto; Fakhfouri, G; Rahimian, R; Tron, Gian Cesare; Genazzani, Armando | |
“Synthesis and in vitro evaluation of tetrasubstituted pyridines as potential PI3Ks inhibitors” | 1-gen-2013 | Galli, Ubaldina; E., Ciraolo; E., Hirsch; Sorba, Giovanni; Tron, Gian Cesare | |
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases | 1-gen-2012 | Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey |
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