Sfoglia per Autore
Crystal structure of human nicotinic acid phosphoribosyltransferase
2015-01-01 Marletta, ADA SERENA; Massarotti, Alberto; Orsomando, Giuseppe; Magni, Giulio; Rizzi, Menico; Garavaglia, Silvia
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors
2015-01-01 Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement
2015-01-01 Theeramunkong, S.; Galli, Ubaldina; Grolla, Ambra; Caldarelli, Antonio; Travelli, Cristina; Massarotti, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; Genazzani, Armando; Tron, Gian Cesare
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement
2015-01-01 Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare
Capitolo 23. Istamina e agenti antistaminici
2014-01-01 Sorba, Giovanni; Massarotti, Alberto
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?
2014-01-01 Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity
2014-01-01 E., Bellomo; Massarotti, Alberto; C., Hogstrand; W., Maret
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles
2014-01-01 Massarotti, Alberto; A., Brunco; Sorba, Giovanni; Tron, Gian Cesare
Sintesi e caratterizzazione di nuovi inibitori di DGKα
2014-01-01 Malacarne, V.; Ruffo, E.; Massarotti, Alberto; Baldanzi, Gianluca; Tron, Gian Cesare; Graziani, A.
Small molecule inhibitors of West Nile virus
2014-01-01 Elseginy, Sa; Massarotti, Alberto; Nawwar, Ga; Amin, Km; Brancale, A.
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols
2014-01-01 Mercalli, Valentina; M., Giustiniano; DEL GROSSO, Erika; Varese, Monica; H., Cassese; Massarotti, Alberto; E., Novellino; Tron, Gian Cesare
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable
2013-01-01 Massarotti, Alberto; Tron, Gian Cesare
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors.
2013-01-01 Galli, Ubaldina; Travelli, Cristina; Massarotti, Alberto; Fakhfouri, G; Rahimian, R; Tron, Gian Cesare; Genazzani, Armando
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus
2013-01-01 Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A.
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents
2013-01-01 Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey
Parallel synthesis of “click” chalcones as antitubulin agents
2013-01-01 Utsintong, M; Massarotti, Alberto; Caldarelli, Antonio; Theeramunkong, S.
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases
2012-01-01 Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups?
2012-01-01 Massarotti, Alberto; Genazzani, A. A.; Tron, Gian Cesare
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives
2012-01-01 Ricci, A; Anthopoulos, A; Massarotti, Alberto; Grimstead, I; Brancale, A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Crystal structure of human nicotinic acid phosphoribosyltransferase | 1-gen-2015 | Marletta, ADA SERENA; Massarotti, Alberto; Orsomando, Giuseppe; Magni, Giulio; Rizzi, Menico; Garavaglia, Silvia | |
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors | 1-gen-2015 | Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare | |
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 1-gen-2015 | Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare | |
Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement | 1-gen-2015 | Theeramunkong, S.; Galli, Ubaldina; Grolla, Ambra; Caldarelli, Antonio; Travelli, Cristina; Massarotti, Alberto; Troiani, M. P.; Alisi, M. A.; Orsomando, G.; Genazzani, Armando; Tron, Gian Cesare | |
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement | 1-gen-2015 | Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare | |
Capitolo 23. Istamina e agenti antistaminici | 1-gen-2014 | Sorba, Giovanni; Massarotti, Alberto | |
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? | 1-gen-2014 | Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare | |
Zinc Ions Modulate Protein Tyrosine Phosphatase 1B activity | 1-gen-2014 | E., Bellomo; Massarotti, Alberto; C., Hogstrand; W., Maret | |
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles | 1-gen-2014 | Massarotti, Alberto; A., Brunco; Sorba, Giovanni; Tron, Gian Cesare | |
Sintesi e caratterizzazione di nuovi inibitori di DGKα | 1-gen-2014 | Malacarne, V.; Ruffo, E.; Massarotti, Alberto; Baldanzi, Gianluca; Tron, Gian Cesare; Graziani, A. | |
Small molecule inhibitors of West Nile virus | 1-gen-2014 | Elseginy, Sa; Massarotti, Alberto; Nawwar, Ga; Amin, Km; Brancale, A. | |
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols | 1-gen-2014 | Mercalli, Valentina; M., Giustiniano; DEL GROSSO, Erika; Varese, Monica; H., Cassese; Massarotti, Alberto; E., Novellino; Tron, Gian Cesare | |
ZINClick: a database of 16 million of new and patentable 1,4 disubstituted triazoles easily synthetizable | 1-gen-2013 | Massarotti, Alberto; Tron, Gian Cesare | |
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. | 1-gen-2013 | Galli, Ubaldina; Travelli, Cristina; Massarotti, Alberto; Fakhfouri, G; Rahimian, R; Tron, Gian Cesare; Genazzani, Armando | |
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus | 1-gen-2013 | Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A. | |
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents | 1-gen-2013 | Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey | |
Parallel synthesis of “click” chalcones as antitubulin agents | 1-gen-2013 | Utsintong, M; Massarotti, Alberto; Caldarelli, Antonio; Theeramunkong, S. | |
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases | 1-gen-2012 | Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey | |
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? | 1-gen-2012 | Massarotti, Alberto; Genazzani, A. A.; Tron, Gian Cesare | |
Haptic-Driven applications to Molecular Modelling: State of the Art and Perspectives | 1-gen-2012 | Ricci, A; Anthopoulos, A; Massarotti, Alberto; Grimstead, I; Brancale, A. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile