Sfoglia per Autore
Natural Product Fragments Preference for Protein Residues
2018-01-01 Levre', Doriana; Massarotti, Alberto
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe
2018-01-01 Rossi, Franca; Morrone, Castrese; Massarotti, Alberto; Ferraris, Davide Maria; Valenti, Anna; Perugino, Giuseppe; Miggiano, Riccardo
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors
2017-01-01 Serafini, Marta; Griglio, Alessia; Fallarini, Silvia; Massarotti, Alberto; Pirali, Tracey
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles
2017-01-01 Levré, Doriana; Massarotti, Alberto
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase
2017-01-01 Morrone, Castrese; Miggiano, Riccardo; Serpe, Mario; Massarotti, Alberto; Valenti, Anna; Del Monaco, Giovanni; Rossi, Mosè; Rossi, Franca; Rizzi, Menico; Perugino, Giuseppe; Ciaramella, Maria
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis
2017-01-01 Giustiniano, Mariateresa; Basso, Andrea; Mercalli, Valentina; Massarotti, Alberto; Novellino, Ettore; Tron, Gian Cesare; Zhu, Jieping
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY
2017-01-01 Baldanzi, Gianluca; Velnati, Suresh; Massarotti, Alberto; Ruffo, Elisa; Tron, Gian Cesare; Andrew, Snow; Graziani, Andrea
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis
2017-01-01 Donini, Stefano; Ferraris, DAVIDE MARIA; Miggiano, Riccardo; Massarotti, Alberto; Rizzi, Menico
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS
2016-01-01 Mercalli, Valentina; Massarotti, Alberto; Baldanzi, Gianluca; Graziani, A.; Tron, Gian Cesare
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors
2016-01-01 Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy
2016-01-01 Massarotti, Alberto
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)"
2016-01-01 Bettio, V.; Velnati, S.; Malacarne, V.; Massarotti, Alberto; Graziani, A.; Tron, Gian Cesare; Baldanzi, Gianluca
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis
2016-01-01 Cargnin, Sarah; Massarotti, Alberto; Terrazzino, Salvatore
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring
2016-01-01 Marchetti, Francesco; Massarotti, Alberto; Yauk, Carole L; Pacchierotti, Francesca; Russo, Antonella
The metal face of protein tyrosine phosphatase 1B
2016-01-01 Bellomo, Elisa; Birla Singh, Kshetrimayum; Massarotti, Alberto; Hogstrand, Christer; Maret, Wolfgang
Structural biology in antiviral drug discovery
2016-01-01 Bassetto, M.; Massarotti, Alberto; Coluccia, A.; Brancale, A.
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones
2016-01-01 Massarotti, Alberto; Coluccia, Antonio
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles
2016-01-01 Massarotti, Alberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Natural Product Fragments Preference for Protein Residues | 1-gen-2018 | Levre', Doriana; Massarotti, Alberto | |
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe | 1-gen-2018 | Rossi, Franca; Morrone, Castrese; Massarotti, Alberto; Ferraris, Davide Maria; Valenti, Anna; Perugino, Giuseppe; Miggiano, Riccardo | |
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors | 1-gen-2017 | Serafini, Marta; Griglio, Alessia; Fallarini, Silvia; Massarotti, Alberto; Pirali, Tracey | |
ZINClick 2.0: from a virtual database to smart synthesizable 1,4-disubstituted 1,2,3-triazoles | 1-gen-2017 | Levré, Doriana; Massarotti, Alberto | |
Interdomain interactions rearrangements control the reaction steps of a thermostable DNA alkyltransferase | 1-gen-2017 | Morrone, Castrese; Miggiano, Riccardo; Serpe, Mario; Massarotti, Alberto; Valenti, Anna; Del Monaco, Giovanni; Rossi, Mosè; Rossi, Franca; Rizzi, Menico; Perugino, Giuseppe; Ciaramella, Maria | |
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis | 1-gen-2017 | Giustiniano, Mariateresa; Basso, Andrea; Mercalli, Valentina; Massarotti, Alberto; Novellino, Ettore; Tron, Gian Cesare; Zhu, Jieping | |
NOVEL DIACYLGLYCEROL KINASE ALPHA INHIBITORS FOR X-LINKED LYMPHOPROLIFERATIVE DISEASE 1 THERAPY | 1-gen-2017 | Baldanzi, Gianluca; Velnati, Suresh; Massarotti, Alberto; Ruffo, Elisa; Tron, Gian Cesare; Andrew, Snow; Graziani, Andrea | |
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 1-gen-2017 | Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare | |
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 1-gen-2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare | |
Structural investigations on orotate phosphoribosyltransferase from Mycobacterium tuberculosis, a key enzyme of the de novo pyrimidine biosynthesis | 1-gen-2017 | Donini, Stefano; Ferraris, DAVIDE MARIA; Miggiano, Riccardo; Massarotti, Alberto; Rizzi, Menico | |
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS | 1-gen-2016 | Mercalli, Valentina; Massarotti, Alberto; Baldanzi, Gianluca; Graziani, A.; Tron, Gian Cesare | |
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors | 1-gen-2016 | Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey | |
Discovering the hidden chemical space of chemistry reactions: from 1,2,3-triazoles nucleus to ZINClick galaxy | 1-gen-2016 | Massarotti, Alberto | |
Sviluppo di inibitori di DGKα per la terapia della psoriasi all'interno del progetto "Terapie innovative per la psoriasi (TIPSO)" | 1-gen-2016 | Bettio, V.; Velnati, S.; Malacarne, V.; Massarotti, Alberto; Graziani, A.; Tron, Gian Cesare; Baldanzi, Gianluca | |
BDNF Val66Met and clinical response to antipsychotic drugs: A systematic review and meta-analysis | 1-gen-2016 | Cargnin, Sarah; Massarotti, Alberto; Terrazzino, Salvatore | |
The adverse outcome pathway (AOP) for chemical binding to tubulin in oocytes leading to aneuploid offspring | 1-gen-2016 | Marchetti, Francesco; Massarotti, Alberto; Yauk, Carole L; Pacchierotti, Francesca; Russo, Antonella | |
The metal face of protein tyrosine phosphatase 1B | 1-gen-2016 | Bellomo, Elisa; Birla Singh, Kshetrimayum; Massarotti, Alberto; Hogstrand, Christer; Maret, Wolfgang | |
Structural biology in antiviral drug discovery | 1-gen-2016 | Bassetto, M.; Massarotti, Alberto; Coluccia, A.; Brancale, A. | |
An in-silico approach aimed to clarify the role of Y181C and K103N HIV-1 reverse transcriptase mutations versus Indole Aryl Sulphones | 1-gen-2016 | Massarotti, Alberto; Coluccia, Antonio | |
ZINClick: a virtual database of 16 million novel, patentable and readily synthesizable 1,4-disubstituted 1,2,3-triazoles | 1-gen-2016 | Massarotti, Alberto |
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