Sfoglia per Autore
Dual- and multi-action Pt(IV) antitumor prodrugs or how to kill two birds with one stone
2020-01-01 Ravera, Mauro; Gabano, Elisabetta; Osella, Domenico
New Platinum-Based Prodrug Pt(IV)Ac-POA: Antitumour Effects in Rat C6 Glioblastoma Cells
2020-01-01 Ferrari, B.; Urselli, F.; Gilodi, M.; Camuso, S.; Priori, E. C.; Rangone, B.; Ravera, M.; Veneroni, P.; Zanellato, I.; Roda, E.; Osella, D.; Bottone, M. G.
A step towards development of promising trypanocidal agents: Synthesis, characterization and in vitro biological evaluation of ferrocenyl Mannich base-type derivatives
2019-01-01 Paucar, Rocío; Martín-Escolano, Rubén; Moreno-Viguri, Elsa; Cirauqui, Nuria; Rodrigues, Carlos Rangel; Marín, Clotilde; Sánchez-Moreno, Manuel; Pérez-Silanes, Silvia; Ravera, Mauro; Gabano, Elisabetta
Synthesis and characterization of cyclohexane-1R,2R-diamine-based Pt(iv) dicarboxylato anticancer prodrugs: their selective activity against human colon cancer cell lines
2019-01-01 Gabano, E.; Ravera, M.; Perin, E.; Zanellato, I.; Rangone, B.; Mcglinchey, M. J.; Osella, D.
A view on multi-action Pt(IV) antitumor prodrugs
2019-01-01 Ravera, Mauro; Gabano, Elisabetta; Mcglinchey, Michael J.; Osella, Domenico
Antiproliferative Activity of Pt(IV) Conjugates Containing the Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) Ketoprofen and Naproxen
2019-01-01 Ravera, M.; Zanellato, I.; Gabano, E.; Perin, E.; Rangone, B.; Coppola, M.; Osella, D.
Pt(IV) Bifunctional Prodrug Containing 2-(2-Propynyl)octanoato Axial Ligand: Induction of Immunogenic Cell Death on Colon Cancer
2019-01-01 Sabbatini, Maurizio; Zanellato, Ilaria; Ravera, Mauro; Gabano, Elisabetta; Perin, Elena; Rangone, Beatrice; Osella, Domenico
Conjugation between maleimide-containing Pt(IV) prodrugs and furan or furan-containing drug delivery vectors via Diels-Alder cycloaddition
2019-01-01 Gabano, Elisabetta; Perin, Elena; Bonzani, Diego; Ravera, Mauro
Hybrid inorganic (nonporous silica)/organic (alginate) core-shell platform for targeting a cisplatin-based Pt(IV) anticancer prodrug
2018-01-01 Ravera, Mauro; Gabano, Elisabetta; Bonzani, Diego; Zanellato, Ilaria; Arrais, Aldo; Cantamessa, Simone; Biggiogera, Marco; Osella, Domenico
Pt(IV)/Re(I) Chitosan Conjugates as a Flexible Platform for the Transport of Therapeutic and/or Diagnostic Anticancer Agents
2018-01-01 Gabano, Elisabetta; do Quental, Letícia; Perin, Elena; Silva, Francisco; Raposinho, Paula; Paulo, António; Ravera, Mauro
Organometallic compounds in the discovery of new agents against kinetoplastid-caused diseases
2018-01-01 Ravera, M.; Moreno-Viguri, E.; Paucar, R.; Perez-Silanes, S.; Gabano, E.
The cisplatin-based Pt(IV)-diclorofibrato multi-action anticancer prodrug exhibits excellent performances also under hypoxic conditions
2018-01-01 Gabano, Elisabetta; Ravera, Mauro; Trivero, Francesca; Tinello, Stefano; Gallina, Andrea; Zanellato, Ilaria; Gariboldi, Marzia B; Monti, Elena; Osella, Domenico
Transition metal carbonyl clusters in biology: A futile or niche research area?
2018-01-01 Arrais, Aldo; Gabano, Elisabetta; Ravera, Mauro; Osella, Domenico
May glutamine addiction drive the delivery of antitumor cisplatin-based Pt(IV) prodrugs?
2017-01-01 Ravera, Mauro; Gabano, Elisabetta; Tinello, Stefano; Zanellato, Ilaria; Osella, Domenico
Cisplatin and valproate released from the bifunctional [Pt(IV)Cl2(NH3)2(valproato)2] antitumor prodrug or from liposome formulations: who does what?
2017-01-01 Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Gallina, A.; Perin, Elena; Arrais, Aldo; Cantamessa, Simone; Osella, Domenico
How to obtain Pt(IV) complexes suitable for conjugation to nanovectors from the oxidation of [PtCl(terpyridine)]+
2017-01-01 Gabano, Elisabetta; Perin, Elena; Fielden, C.; Platts, J. A.; Gallina, Andrea; Rangone, Beatrice; Ravera, Mauro
An unsymmetric cisplatin-based Pt(IV) derivative containing 2-(2-propynyl)octanoate: A very efficient multi-action antitumor prodrug candidate
2017-01-01 Gabano, Elisabetta; Ravera, Mauro; Zanellato, Ilaria; Tinello, Stefano; Gallina, Andrea; Rangone, Beatrice; Gandin, Valentina; Marzano, Cristina; Bottone, Maria Grazia; Osella, Domenico
Anthracene-terpyridine metal complexes as new G-quadruplex DNA binders
2016-01-01 Gama, Sofia; Rodrigues, Inês; Mendes, Filipa; Santos, Isabel C.; Gabano, Elisabetta; Klejevskaja, Beata; Gonzalez Garcia, Jorge; Ravera, Mauro; Vilar, Ramon; Paulo, António
Functionalized nonporous silica nanoparticles as carriers for Pt(IV) anticancer prodrugs
2016-01-01 Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Perin, Elena; Arrais, Aldo; Osella, Domenico
Antiproliferative activity of a series of cisplatin-based Pt(IV)-acetylamido/carboxylato prodrugs
2016-01-01 Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Fregonese, Federico; Pelosi, Giorgio; Platts, James A.; Osella, Domenico
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Dual- and multi-action Pt(IV) antitumor prodrugs or how to kill two birds with one stone | 1-gen-2020 | Ravera, Mauro; Gabano, Elisabetta; Osella, Domenico | |
New Platinum-Based Prodrug Pt(IV)Ac-POA: Antitumour Effects in Rat C6 Glioblastoma Cells | 1-gen-2020 | Ferrari, B.; Urselli, F.; Gilodi, M.; Camuso, S.; Priori, E. C.; Rangone, B.; Ravera, M.; Veneroni, P.; Zanellato, I.; Roda, E.; Osella, D.; Bottone, M. G. | |
A step towards development of promising trypanocidal agents: Synthesis, characterization and in vitro biological evaluation of ferrocenyl Mannich base-type derivatives | 1-gen-2019 | Paucar, Rocío; Martín-Escolano, Rubén; Moreno-Viguri, Elsa; Cirauqui, Nuria; Rodrigues, Carlos Rangel; Marín, Clotilde; Sánchez-Moreno, Manuel; Pérez-Silanes, Silvia; Ravera, Mauro; Gabano, Elisabetta | |
Synthesis and characterization of cyclohexane-1R,2R-diamine-based Pt(iv) dicarboxylato anticancer prodrugs: their selective activity against human colon cancer cell lines | 1-gen-2019 | Gabano, E.; Ravera, M.; Perin, E.; Zanellato, I.; Rangone, B.; Mcglinchey, M. J.; Osella, D. | |
A view on multi-action Pt(IV) antitumor prodrugs | 1-gen-2019 | Ravera, Mauro; Gabano, Elisabetta; Mcglinchey, Michael J.; Osella, Domenico | |
Antiproliferative Activity of Pt(IV) Conjugates Containing the Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) Ketoprofen and Naproxen | 1-gen-2019 | Ravera, M.; Zanellato, I.; Gabano, E.; Perin, E.; Rangone, B.; Coppola, M.; Osella, D. | |
Pt(IV) Bifunctional Prodrug Containing 2-(2-Propynyl)octanoato Axial Ligand: Induction of Immunogenic Cell Death on Colon Cancer | 1-gen-2019 | Sabbatini, Maurizio; Zanellato, Ilaria; Ravera, Mauro; Gabano, Elisabetta; Perin, Elena; Rangone, Beatrice; Osella, Domenico | |
Conjugation between maleimide-containing Pt(IV) prodrugs and furan or furan-containing drug delivery vectors via Diels-Alder cycloaddition | 1-gen-2019 | Gabano, Elisabetta; Perin, Elena; Bonzani, Diego; Ravera, Mauro | |
Hybrid inorganic (nonporous silica)/organic (alginate) core-shell platform for targeting a cisplatin-based Pt(IV) anticancer prodrug | 1-gen-2018 | Ravera, Mauro; Gabano, Elisabetta; Bonzani, Diego; Zanellato, Ilaria; Arrais, Aldo; Cantamessa, Simone; Biggiogera, Marco; Osella, Domenico | |
Pt(IV)/Re(I) Chitosan Conjugates as a Flexible Platform for the Transport of Therapeutic and/or Diagnostic Anticancer Agents | 1-gen-2018 | Gabano, Elisabetta; do Quental, Letícia; Perin, Elena; Silva, Francisco; Raposinho, Paula; Paulo, António; Ravera, Mauro | |
Organometallic compounds in the discovery of new agents against kinetoplastid-caused diseases | 1-gen-2018 | Ravera, M.; Moreno-Viguri, E.; Paucar, R.; Perez-Silanes, S.; Gabano, E. | |
The cisplatin-based Pt(IV)-diclorofibrato multi-action anticancer prodrug exhibits excellent performances also under hypoxic conditions | 1-gen-2018 | Gabano, Elisabetta; Ravera, Mauro; Trivero, Francesca; Tinello, Stefano; Gallina, Andrea; Zanellato, Ilaria; Gariboldi, Marzia B; Monti, Elena; Osella, Domenico | |
Transition metal carbonyl clusters in biology: A futile or niche research area? | 1-gen-2018 | Arrais, Aldo; Gabano, Elisabetta; Ravera, Mauro; Osella, Domenico | |
May glutamine addiction drive the delivery of antitumor cisplatin-based Pt(IV) prodrugs? | 1-gen-2017 | Ravera, Mauro; Gabano, Elisabetta; Tinello, Stefano; Zanellato, Ilaria; Osella, Domenico | |
Cisplatin and valproate released from the bifunctional [Pt(IV)Cl2(NH3)2(valproato)2] antitumor prodrug or from liposome formulations: who does what? | 1-gen-2017 | Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Gallina, A.; Perin, Elena; Arrais, Aldo; Cantamessa, Simone; Osella, Domenico | |
How to obtain Pt(IV) complexes suitable for conjugation to nanovectors from the oxidation of [PtCl(terpyridine)]+ | 1-gen-2017 | Gabano, Elisabetta; Perin, Elena; Fielden, C.; Platts, J. A.; Gallina, Andrea; Rangone, Beatrice; Ravera, Mauro | |
An unsymmetric cisplatin-based Pt(IV) derivative containing 2-(2-propynyl)octanoate: A very efficient multi-action antitumor prodrug candidate | 1-gen-2017 | Gabano, Elisabetta; Ravera, Mauro; Zanellato, Ilaria; Tinello, Stefano; Gallina, Andrea; Rangone, Beatrice; Gandin, Valentina; Marzano, Cristina; Bottone, Maria Grazia; Osella, Domenico | |
Anthracene-terpyridine metal complexes as new G-quadruplex DNA binders | 1-gen-2016 | Gama, Sofia; Rodrigues, Inês; Mendes, Filipa; Santos, Isabel C.; Gabano, Elisabetta; Klejevskaja, Beata; Gonzalez Garcia, Jorge; Ravera, Mauro; Vilar, Ramon; Paulo, António | |
Functionalized nonporous silica nanoparticles as carriers for Pt(IV) anticancer prodrugs | 1-gen-2016 | Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Perin, Elena; Arrais, Aldo; Osella, Domenico | |
Antiproliferative activity of a series of cisplatin-based Pt(IV)-acetylamido/carboxylato prodrugs | 1-gen-2016 | Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Fregonese, Federico; Pelosi, Giorgio; Platts, James A.; Osella, Domenico |
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