Sfoglia per Autore
Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors
2020-01-01 Serafini, M.; Cordero Sanchez, C.; Di Paola, R.; Bhela, I. P.; Aprile, S.; Purghe, B.; Fusco, R.; Cuzzocrea, S.; Genazzani, A.; Riva, B.; Pirali, T.
Soft drugs for dermatological applications: recent trends
2019-01-01 Aprile, Silvio; Serafini, Marta; Pirali, Tracey
A primer of deuterium in drug design
2019-01-01 Cargnin, Sarah; Serafini, Marta; Pirali, Tracey
SOCE: EMERGE UN NUOVO TARGET TERAPEUTICO DAL “CALCIUM TOOLKIT” DELLA CELLULA
2019-01-01 Serafini, Marta; Pirali, Tracey
Applications of deuterium in medicinal chemistry
2019-01-01 Pirali, Tracey; Serafini, Marta; Cargnin, Sarah; Genazzani, Armando
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors
2019-01-01 Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction
2019-01-01 Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare
Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis
2018-01-01 Campa, Carlo C; Silva, Rangel L; Margaria, Jean P; Pirali, Tracey; Mattos, Matheus S; Kraemer, Lucas R; Reis, Diego C; Grosa, Giorgio; Copperi, Francesca; Dalmarco, Eduardo M; Lima-Júnior, Roberto C P; Aprile, Silvio; Sala, Valentina; Dal Bello, Federica; Prado, Douglas Silva; Alves-Filho, Jose Carlos; Medana, Claudio; Cassali, Geovanni D; Tron, Gian Cesare; Teixeira, Mauro M; Ciraolo, Elisa; Russo, Remo C; Hirsch, Emilio
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis
2018-01-01 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, Celia; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; Biocotino, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders
2018-01-01 Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
2018-01-01 Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia
Arynes and isocyanides: Two close-knit partners in multicomponent reactions
2018-01-01 Serafini, Marta; Pirali, Tracey
An aryne-based three-component access to α-aroylamino amides
2017-01-01 Serafini, Marta; Griglio, Alessia; Viarengo, Sara; Aprile, Silvio; Pirali, Tracey
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors
2017-01-01 Serafini, Marta; Griglio, Alessia; Fallarini, Silvia; Massarotti, Alberto; Pirali, Tracey
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
The use of 2-hydroxymethyl benzoic acid as an effective water surrogate in the Passerini reaction: A straightforward access to α-hydroxyamides
2017-01-01 Serafini, Marta; Griglio, Alessia; Oberto, Elena; Pirali, Tracey; Tron, Gian Cesare
TRPV1 Modulator Compounds
2017-01-01 Devesa, G. I.; Genazzani, A.; Pirali, T.; Fernandez-Carvajal, A.; Ferrer-Montiel, A. V.
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors
2016-01-01 Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey
Transition-Metal-Free Synthesis of 2-Arylimidazolones via Cascade Reaction between Arynes and α,α′-Disubstituted α-Isocyanoacetamides
2016-01-01 Gesu', Alessandro; Pozzoli, Claudio; Torre, Enza; Aprile, Silvio; Pirali, Tracey
Preparation of 1-(triazolylphenyl)-5-(trifluoromethyl)pyrazole compounds useful as SOCE modulators
2016-01-01 Pirali, Tracey; Genazzani, Armando; Riva, Beatrice
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors | 1-gen-2020 | Serafini, M.; Cordero Sanchez, C.; Di Paola, R.; Bhela, I. P.; Aprile, S.; Purghe, B.; Fusco, R.; Cuzzocrea, S.; Genazzani, A.; Riva, B.; Pirali, T. | |
Soft drugs for dermatological applications: recent trends | 1-gen-2019 | Aprile, Silvio; Serafini, Marta; Pirali, Tracey | |
A primer of deuterium in drug design | 1-gen-2019 | Cargnin, Sarah; Serafini, Marta; Pirali, Tracey | |
SOCE: EMERGE UN NUOVO TARGET TERAPEUTICO DAL “CALCIUM TOOLKIT” DELLA CELLULA | 1-gen-2019 | Serafini, Marta; Pirali, Tracey | |
Applications of deuterium in medicinal chemistry | 1-gen-2019 | Pirali, Tracey; Serafini, Marta; Cargnin, Sarah; Genazzani, Armando | |
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors | 1-gen-2019 | Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey | |
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction | 1-gen-2019 | Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare | |
Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis | 1-gen-2018 | Campa, Carlo C; Silva, Rangel L; Margaria, Jean P; Pirali, Tracey; Mattos, Matheus S; Kraemer, Lucas R; Reis, Diego C; Grosa, Giorgio; Copperi, Francesca; Dalmarco, Eduardo M; Lima-Júnior, Roberto C P; Aprile, Silvio; Sala, Valentina; Dal Bello, Federica; Prado, Douglas Silva; Alves-Filho, Jose Carlos; Medana, Claudio; Cassali, Geovanni D; Tron, Gian Cesare; Teixeira, Mauro M; Ciraolo, Elisa; Russo, Remo C; Hirsch, Emilio | |
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis | 1-gen-2018 | Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, Celia; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; Biocotino, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey | |
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders | 1-gen-2018 | Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio | |
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies | 1-gen-2018 | Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia | |
Arynes and isocyanides: Two close-knit partners in multicomponent reactions | 1-gen-2018 | Serafini, Marta; Pirali, Tracey | |
An aryne-based three-component access to α-aroylamino amides | 1-gen-2017 | Serafini, Marta; Griglio, Alessia; Viarengo, Sara; Aprile, Silvio; Pirali, Tracey | |
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors | 1-gen-2017 | Serafini, Marta; Griglio, Alessia; Fallarini, Silvia; Massarotti, Alberto; Pirali, Tracey | |
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 1-gen-2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare | |
The use of 2-hydroxymethyl benzoic acid as an effective water surrogate in the Passerini reaction: A straightforward access to α-hydroxyamides | 1-gen-2017 | Serafini, Marta; Griglio, Alessia; Oberto, Elena; Pirali, Tracey; Tron, Gian Cesare | |
TRPV1 Modulator Compounds | 1-gen-2017 | Devesa, G. I.; Genazzani, A.; Pirali, T.; Fernandez-Carvajal, A.; Ferrer-Montiel, A. V. | |
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors | 1-gen-2016 | Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey | |
Transition-Metal-Free Synthesis of 2-Arylimidazolones via Cascade Reaction between Arynes and α,α′-Disubstituted α-Isocyanoacetamides | 1-gen-2016 | Gesu', Alessandro; Pozzoli, Claudio; Torre, Enza; Aprile, Silvio; Pirali, Tracey | |
Preparation of 1-(triazolylphenyl)-5-(trifluoromethyl)pyrazole compounds useful as SOCE modulators | 1-gen-2016 | Pirali, Tracey; Genazzani, Armando; Riva, Beatrice |
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