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Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors 1-gen-2020 Serafini, M.; Cordero Sanchez, C.; Di Paola, R.; Bhela, I. P.; Aprile, S.; Purghe, B.; Fusco, R.; Cuzzocrea, S.; Genazzani, A.; Riva, B.; Pirali, T.
Soft drugs for dermatological applications: recent trends 1-gen-2019 Aprile, Silvio; Serafini, Marta; Pirali, Tracey
A primer of deuterium in drug design 1-gen-2019 Cargnin, Sarah; Serafini, Marta; Pirali, Tracey
SOCE: EMERGE UN NUOVO TARGET TERAPEUTICO DAL “CALCIUM TOOLKIT” DELLA CELLULA 1-gen-2019 Serafini, Marta; Pirali, Tracey
Applications of deuterium in medicinal chemistry 1-gen-2019 Pirali, Tracey; Serafini, Marta; Cargnin, Sarah; Genazzani, Armando
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 1-gen-2019 Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey
Drug Discovery for Soft Drugs on TRPV1 and TRPM8 Channels Using the Passerini Reaction 1-gen-2019 Pirali, Tracey; Galli, Ubaldina; Serafini, Marta; Griglio, Alessia; Genazzani, Armando; Tron, Gian Cesare
Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis 1-gen-2018 Campa, Carlo C; Silva, Rangel L; Margaria, Jean P; Pirali, Tracey; Mattos, Matheus S; Kraemer, Lucas R; Reis, Diego C; Grosa, Giorgio; Copperi, Francesca; Dalmarco, Eduardo M; Lima-Júnior, Roberto C P; Aprile, Silvio; Sala, Valentina; Dal Bello, Federica; Prado, Douglas Silva; Alves-Filho, Jose Carlos; Medana, Claudio; Cassali, Geovanni D; Tron, Gian Cesare; Teixeira, Mauro M; Ciraolo, Elisa; Russo, Remo C; Hirsch, Emilio
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis 1-gen-2018 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, Celia; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; Biocotino, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders 1-gen-2018 Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies 1-gen-2018 Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia
Arynes and isocyanides: Two close-knit partners in multicomponent reactions 1-gen-2018 Serafini, Marta; Pirali, Tracey
An aryne-based three-component access to α-aroylamino amides 1-gen-2017 Serafini, Marta; Griglio, Alessia; Viarengo, Sara; Aprile, Silvio; Pirali, Tracey
Synthesis, biological evaluation and molecular docking of Ugi and Passerini products as novel indoleamine 2,3-dioxygenase 1 inhibitors 1-gen-2017 Serafini, Marta; Griglio, Alessia; Fallarini, Silvia; Massarotti, Alberto; Pirali, Tracey
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs 1-gen-2017 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
The use of 2-hydroxymethyl benzoic acid as an effective water surrogate in the Passerini reaction: A straightforward access to α-hydroxyamides 1-gen-2017 Serafini, Marta; Griglio, Alessia; Oberto, Elena; Pirali, Tracey; Tron, Gian Cesare
TRPV1 Modulator Compounds 1-gen-2017 Devesa, G. I.; Genazzani, A.; Pirali, T.; Fernandez-Carvajal, A.; Ferrer-Montiel, A. V.
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors 1-gen-2016 Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey
Transition-Metal-Free Synthesis of 2-Arylimidazolones via Cascade Reaction between Arynes and α,α′-Disubstituted α-Isocyanoacetamides 1-gen-2016 Gesu', Alessandro; Pozzoli, Claudio; Torre, Enza; Aprile, Silvio; Pirali, Tracey
Preparation of 1-​(triazolylphenyl)​-​5-​(trifluoromethyl)​pyrazole compounds useful as SOCE modulators 1-gen-2016 Pirali, Tracey; Genazzani, Armando; Riva, Beatrice
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