Sfoglia per Autore
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents
2013-01-01 Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases
2012-01-01 Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey
PI3K keeps the balance between metabolism and cancer
2012-01-01 Braccini, L; Ciraolo, E; Martini, M; Pirali, Tracey; Germena, G; Rolfo, K; Hirsch, E.
Transition-Metal-Free Direct Arylation of Anilines
2012-01-01 Pirali, Tracey; Zhang, F; Miller, A. H.; Head, J.; Mcausland, D.; Greaney, M. F.
A novel α-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates
2011-01-01 Mossetti, R; Caprioglio, D; Colombano, G; Tron, Gian Cesare; Pirali, Tracey
A novel alpha-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates
2011-01-01 Mossetti, Riccardo; Caprioglio, Diego; Colombano, Giampiero; Tron, Gian Cesare; Pirali, Tracey
Imides: forgotten players in the Ugi reaction. One-pot multicomponent synthesis of quinazolinones
2011-01-01 Mossetti, R; Pirali, Tracey; Saggiorato, D; Tron, Gian Cesare
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues
2011-01-01 Theeramunkong, S; Caldarelli, Antonio; Massarotti, Alberto; Aprile, Silvio; Caprioglio, Diego; Zaninetti, Roberta; Teruggi, A; Pirali, Tracey; Grosa, Giorgio; Tron, Gian Cesare; Genazzani, Armando
Activation of TRPV4 channels reduces migration of immortalized neuroendocrine cells
2011-01-01 Zaninetti, Roberta; Fornarelli, A; Ciarletta, Monica; Lim, Dmitry; Caldarelli, Antonio; Pirali, Tracey; Cariboni, A; Owsianik, G; Nilius, B; Canonico, Pier Luigi; Distasi, Carla; Genazzani, Armando
Stereospecific synthesis of syn-α-oximinoamides by a three-component reaction of isocyanides, syn-chlorooximes, and carboxylic acids
2011-01-01 Pirali, Tracey; Mossetti, R; Galli, S; Tron, Gian Cesare
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors
2011-01-01 Guasconi, M; Lu, X; Massarotti, Alberto; Caldarelli, Antonio; Ciraolo, E; Tron, Gian Cesare; Hirsch, E; Sorba, Giovanni; Pirali, Tracey
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation
2011-01-01 Mesenzani, Ornella; Massarotti, Alberto; Giustiniano, M; Pirali, Tracey; Bevilacqua, V; Caldarelli, Antonio; Canonico, Pier Luigi; Sorba, Giovanni; Novellino, E; Genazzani, Armando; Tron, Gian Cesare
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction
2010-01-01 Massarotti, Alberto; Giustiniano, M.; Pirali, Tracey; Novellino, E.; Sorba, Giovanni; Tron, Gian Cesare
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination
2010-01-01 Giustiniano, M; Pirali, Tracey; Massarotti, Alberto; Biletta, B; Novellino, E; Campiglia, P; Sorba, Giovanni; Tron, Gian Cesare
Efficient Synthesis of α-Ketoamides via 2-Acyl-5-aminooxazoles by Reacting Acyl Chlorides and α-Isocyanoacetamides
2010-01-01 Mossetti, R; Pirali, Tracey; Tron, Gian Cesare; Zhu, J.
Synthesis, molecular docking and biological evalutation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition
2010-01-01 Pirali, T; Faccio, V; Mossetti, R; Grolla, Aa; DI MICCO, S; Bifulco, G; Genazzani, A; Tron, Gc
Synthesis and biological evaluation of combretatriazoles
2009-01-01 Pirali, Tracey; Massarotti, Alberto; DEL GROSSO, Erika; Sorba, Giovanni; Genazzani, Armando; Tron, Gian Cesare
Synthesis of Passerini-Ugi hybrids by a four-component reaction using the glycolaldehyde dimer
2009-01-01 Mossetti, Riccardo; Pirali, Tracey; Tron, Gian Cesare
Synthesis, biological evaluation, and molecular docking of Ugi products containing a zinc-chelating moiety as novel inhibitors of histone deacetylase
2009-01-01 Grolla, Ambra; Podesta, V; Chini, Mg; Di Micco, S; Vallario, A; Genazzani, Armando; Canonico, Pier Luigi; Bifulco, G; Tron, Gian Cesare; Sorba, Giovanni; Pirali, Tracey
A concise entry into nonsymmetrical alkyl polyamines
2008-01-01 Pirali, Tracey; Callipari, G; Ercolano, E; Genazzani, Armando; Giovenzana, Giovanni Battista; Tron, Gian Cesare
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents | 1-gen-2013 | Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey | |
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases | 1-gen-2012 | Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey | |
PI3K keeps the balance between metabolism and cancer | 1-gen-2012 | Braccini, L; Ciraolo, E; Martini, M; Pirali, Tracey; Germena, G; Rolfo, K; Hirsch, E. | |
Transition-Metal-Free Direct Arylation of Anilines | 1-gen-2012 | Pirali, Tracey; Zhang, F; Miller, A. H.; Head, J.; Mcausland, D.; Greaney, M. F. | |
A novel α-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates | 1-gen-2011 | Mossetti, R; Caprioglio, D; Colombano, G; Tron, Gian Cesare; Pirali, Tracey | |
A novel alpha-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates | 1-gen-2011 | Mossetti, Riccardo; Caprioglio, Diego; Colombano, Giampiero; Tron, Gian Cesare; Pirali, Tracey | |
Imides: forgotten players in the Ugi reaction. One-pot multicomponent synthesis of quinazolinones | 1-gen-2011 | Mossetti, R; Pirali, Tracey; Saggiorato, D; Tron, Gian Cesare | |
Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues | 1-gen-2011 | Theeramunkong, S; Caldarelli, Antonio; Massarotti, Alberto; Aprile, Silvio; Caprioglio, Diego; Zaninetti, Roberta; Teruggi, A; Pirali, Tracey; Grosa, Giorgio; Tron, Gian Cesare; Genazzani, Armando | |
Activation of TRPV4 channels reduces migration of immortalized neuroendocrine cells | 1-gen-2011 | Zaninetti, Roberta; Fornarelli, A; Ciarletta, Monica; Lim, Dmitry; Caldarelli, Antonio; Pirali, Tracey; Cariboni, A; Owsianik, G; Nilius, B; Canonico, Pier Luigi; Distasi, Carla; Genazzani, Armando | |
Stereospecific synthesis of syn-α-oximinoamides by a three-component reaction of isocyanides, syn-chlorooximes, and carboxylic acids | 1-gen-2011 | Pirali, Tracey; Mossetti, R; Galli, S; Tron, Gian Cesare | |
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors | 1-gen-2011 | Guasconi, M; Lu, X; Massarotti, Alberto; Caldarelli, Antonio; Ciraolo, E; Tron, Gian Cesare; Hirsch, E; Sorba, Giovanni; Pirali, Tracey | |
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: synthesis and biological evaluation | 1-gen-2011 | Mesenzani, Ornella; Massarotti, Alberto; Giustiniano, M; Pirali, Tracey; Bevilacqua, V; Caldarelli, Antonio; Canonico, Pier Luigi; Sorba, Giovanni; Novellino, E; Genazzani, Armando; Tron, Gian Cesare | |
In search of novel antitubulin agents: synthesis of 1-aryl-5-aroyl tetrazoles by an Ugi 4-CR/hydrogenolysis/transamination reaction | 1-gen-2010 | Massarotti, Alberto; Giustiniano, M.; Pirali, Tracey; Novellino, E.; Sorba, Giovanni; Tron, Gian Cesare | |
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination | 1-gen-2010 | Giustiniano, M; Pirali, Tracey; Massarotti, Alberto; Biletta, B; Novellino, E; Campiglia, P; Sorba, Giovanni; Tron, Gian Cesare | |
Efficient Synthesis of α-Ketoamides via 2-Acyl-5-aminooxazoles by Reacting Acyl Chlorides and α-Isocyanoacetamides | 1-gen-2010 | Mossetti, R; Pirali, Tracey; Tron, Gian Cesare; Zhu, J. | |
Synthesis, molecular docking and biological evalutation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition | 1-gen-2010 | Pirali, T; Faccio, V; Mossetti, R; Grolla, Aa; DI MICCO, S; Bifulco, G; Genazzani, A; Tron, Gc | |
Synthesis and biological evaluation of combretatriazoles | 1-gen-2009 | Pirali, Tracey; Massarotti, Alberto; DEL GROSSO, Erika; Sorba, Giovanni; Genazzani, Armando; Tron, Gian Cesare | |
Synthesis of Passerini-Ugi hybrids by a four-component reaction using the glycolaldehyde dimer | 1-gen-2009 | Mossetti, Riccardo; Pirali, Tracey; Tron, Gian Cesare | |
Synthesis, biological evaluation, and molecular docking of Ugi products containing a zinc-chelating moiety as novel inhibitors of histone deacetylase | 1-gen-2009 | Grolla, Ambra; Podesta, V; Chini, Mg; Di Micco, S; Vallario, A; Genazzani, Armando; Canonico, Pier Luigi; Bifulco, G; Tron, Gian Cesare; Sorba, Giovanni; Pirali, Tracey | |
A concise entry into nonsymmetrical alkyl polyamines | 1-gen-2008 | Pirali, Tracey; Callipari, G; Ercolano, E; Genazzani, Armando; Giovenzana, Giovanni Battista; Tron, Gian Cesare |
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