Sfoglia per Autore
Pt(iv) antitumor prodrugs: dogmas, paradigms, and realities
2022-01-01 Ravera, Mauro; Gabano, Elisabetta; Mcglinchey, Michael J.; Osella, Domenico
The Strange Case: The Unsymmetric Cisplatin-Based Pt(IV) Prodrug [Pt(CH3COO)Cl2(NH3)2(OH)] Exhibits Higher Cytotoxic Activity with respect to Its Symmetric Congeners due to Carrier-Mediated Cellular Uptake
2022-01-01 Gabano, E.; Zanellato, I.; Pinton, G.; Moro, L.; Ravera, M.; Osella, D.
Formulations of highly antiproliferative hydrophobic Pt(IV) complexes into lipidic nanoemulsions as delivery vehicles
2022-01-01 Gabano, E.; Ferraris, C.; Osella, D.; Battaglia, L. S.; Ravera, M.
Hyperspectral characterization of the MSTO-211H cell spheroid model: A FPA–FTIR imaging approach
2021-01-01 Notarstefano, Valentina; Sabbatini, Simona; Sabbatini, Maurizio; Arrais, Aldo; Belloni, Alessia; Pro, Chiara; Vaccari, Lisa; Osella, Domenico; Giorgini, Elisabetta
The effects of sulphur dioxide on wine metabolites: New insights from 1H NMR spectroscopy based in-situ screening, detection, identification and quantification
2021-01-01 Cassino, C.; Tsolakis, C.; Gulino, F.; Vaudano, E.; Osella, D.
Can the Self-Assembling of Dicarboxylate Pt(IV) Prodrugs Influence Their Cell Uptake?
2021-01-01 Ravera, Mauro; Gabano, Elisabetta; Perin, Elena; Rangone, Beatrice; Bonzani, Diego; Osella, Domenico
Unsymmetric cisplatin-based pt(Iv) conjugates containing a parp-1 inhibitor pharmacophore tested on malignant pleural mesothelioma cell lines
2021-01-01 Gabano, E.; Pinton, G.; Balzano, C.; Boumya, S.; Osella, D.; Moro, L.; Ravera, M.
Cis,cis,trans-[PtIVCl2(NH3)2(perillato)2], a dual-action prodrug with excellent cytotoxic and antimetastatic activity
2021-01-01 Ravera, Mauro; Gabano, Elisabetta; Zanellato, Ilaria; Rangone, Beatrice; Perin, Elena; Ferrari, Beatrice; Bottone, Maria Grazia; Osella, Domenico
A multi-methodological inquiry of the behavior of cisplatin-based Pt(IV) derivatives in the presence of bioreductants with a focus on the isolated encounter complexes
2020-01-01 Corinti, D.; Crestoni, M. E.; Fornarini, S.; Dabbish, E.; Sicilia, E.; Gabano, E.; Perin, E.; Osella, D.
Can an Elusive Platinum(III) Oxidation State be Exposed in an Isolated Complex?
2020-01-01 Corinti, D.; Frison, G.; Chiavarino, B.; Gabano, E.; Osella, D.; Crestoni, M. E.; Fornarini, S.
New Platinum-Based Prodrug Pt(IV)Ac-POA: Antitumour Effects in Rat C6 Glioblastoma Cells
2020-01-01 Ferrari, B.; Urselli, F.; Gilodi, M.; Camuso, S.; Priori, E. C.; Rangone, B.; Ravera, M.; Veneroni, P.; Zanellato, I.; Roda, E.; Osella, D.; Bottone, M. G.
Dual- and multi-action Pt(IV) antitumor prodrugs or how to kill two birds with one stone
2020-01-01 Ravera, Mauro; Gabano, Elisabetta; Osella, Domenico
Wine evolution during bottle aging, studied by 1H NMR spectroscopy and multivariate statistical analysis
2019-01-01 Cassino, Claudio; Tsolakis, Christos; Bonello, Federica; Gianotti, Valentina; Osella, Domenico
Antiproliferative Activity of Pt(IV) Conjugates Containing the Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) Ketoprofen and Naproxen
2019-01-01 Ravera, M.; Zanellato, I.; Gabano, E.; Perin, E.; Rangone, B.; Coppola, M.; Osella, D.
Synthesis and characterization of cyclohexane-1R,2R-diamine-based Pt(iv) dicarboxylato anticancer prodrugs: their selective activity against human colon cancer cell lines
2019-01-01 Gabano, E.; Ravera, M.; Perin, E.; Zanellato, I.; Rangone, B.; Mcglinchey, M. J.; Osella, D.
Elusive Intermediates in the Breakdown Reactivity Patterns of Prodrug Platinum(IV) Complexes
2019-01-01 Corinti, D.; Crestoni, M. E.; Fornarini, S.; Ponte, F.; Russo, N.; Sicilia, E.; Gabano, E.; Osella, D.
A view on multi-action Pt(IV) antitumor prodrugs
2019-01-01 Ravera, Mauro; Gabano, Elisabetta; Mcglinchey, Michael J.; Osella, Domenico
Pt(IV) Bifunctional Prodrug Containing 2-(2-Propynyl)octanoato Axial Ligand: Induction of Immunogenic Cell Death on Colon Cancer
2019-01-01 Sabbatini, Maurizio; Zanellato, Ilaria; Ravera, Mauro; Gabano, Elisabetta; Perin, Elena; Rangone, Beatrice; Osella, Domenico
Wine Traceability with Rare Earth Elements
2018-01-01 Aceto, Maurizio; Bonello, Federica; Musso, Davide; Tsolakis, Christos; Cassino, Claudio; Osella, Domenico
JQ1, a BET Inhibitor, Synergizes with Cisplatin and Induces Apoptosis in Highly Chemoresistant Malignant Pleural Mesothelioma Cells
2018-01-01 Zanellato, Ilaria; Colangelo, Donato; Osella, Domenico
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