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A Novel Closo-Ortho-Carborane-Based Glucosamine Derivative as a Promising Agent for Boron Neutron Capture Therapy 1-gen-2025 Imperio, Daniela; Postuma, Ian; Villani, Salvatore; Del Grosso, Erika; Cansolino, Laura; Ferrari, Cinzia; Fallarini, Silvia; Bortolussi, Silva; Panza, Luigi
Mucin 1 antigen mimetic functionalized mannosylated peptide nanofibers for antigen uptake and immune modulation 1-gen-2025 Fallarini, S.; Sodini, A.; Susini, F.; Lesca, G.; Scaglione, S.; Palama, M. E. F.; Maestrelli, F.; Salvatici, M. C.; Cefali, F.; Guler, M. O.; Tekinay, A. B.; Nativi, C.
Structural and functional features of Klebsiella pneumoniae capsular degradation by the phage depolymerase KP32gp38: Implications for vaccination against K. pneumoniae 1-gen-2025 Napolitano, V.; Privitera, M.; Drulis-Kawa, Z.; Marasco, D.; Fallarini, S.; Berisio, R.; Squeglia, F.
EZH2 Inhibition in Mesothelioma Cells Increases the Release of Extracellular Vesicles That Skew Neutrophils Toward a Protumor Phenotype 1-gen-2025 Pinton, G.; Bari, E.; Fallarini, S.; Gigliotti, V.; De Giorgis, V.; Chiazza, F.; Torre, M. L.; Manfredi, M.; Moro, L.
Exploring the pharmaceutical potential of ammonium organotrifluoroborate functional group: Comprehensive chemical, metabolic, and plasma stability evaluation 1-gen-2024 Villani, Salvatore; Imperio, Daniela; Panza, Luigi; Confalonieri, Laura; Fallarini, Silvia; Aprile, Silvio; Del Grosso, Erika
Selective inhibition of indoleamine and tryptophan 2,3-dioxygenases: Comparative study on kynurenine pathway in cell lines via LC-MS/MS-based targeted metabolomics 1-gen-2024 Villani, Salvatore; Fallarini, Silvia; Rezzi, Sarah Jane; Di Martino, Rita Maria Concetta; Aprile, Silvio; Del Grosso, Erika
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 1-gen-2024 Panfili, Eleonora; Rezzi, Sarah Jane; Adamo, Annalisa; Mazzoletti, Daniele; Massarotti, Alberto; Miggiano, Riccardo; Fallarini, Silvia; Ambrosino, Sara; Coletti, Alice; Molinaro, Pasquale; Milella, Michele; Paiella, Salvatore; Macchiarulo, Antonio; Ugel, Stefano; Pirali, Tracey; Pallotta, Maria Teresa
Melanoma Cells Inhibit iNKT Cell Functions via PGE2 and IDO1 1-gen-2023 Torre, E.; Pinton, G.; Lombardi, G.; Fallarini, S.
Site-Selective Functionalized PD-1 Mutant for a Modular Immunological Activity against Cancer Cells 1-gen-2023 Fallarini, S.; Cerofolini, L.; Salobehaj, M.; Rizzo, D.; Gheorghita, G. R.; Licciardi, G.; Capialbi, D. E.; Zullo, V.; Sodini, A.; Nativi, C.; Fragai, M.
A Selective ALDH1A3 Inhibitor Impairs Mesothelioma 3-D Multicellular Spheroid Growth and Neutrophil Recruitment 1-gen-2023 Boumya, Sara; Fallarini, Silvia; Siragusa, Sonia; Petrarolo, Giovanni; Aprile, Silvio; Audrito, Valentina; La Motta, Concettina; Garavaglia, Silvia; Moro, Laura; Pinton, Giulia
Niosomes as Biocompatible Scaffolds for the Multivalent Presentation of Tumor-Associated Antigens (TACAs) to the Immune System 1-gen-2023 Fallarini, S.; Papi, F.; Licciardi, F.; Natali, F.; Lombardi, G.; Maestrelli, F.; Nativi, C.
A Pilot Study on Clinical Scores, Immune Cell Modulation, and Microbiota Composition in Allergic Patients with Rhinitis and Asthma Treated with a Probiotic Preparation 1-gen-2022 Torre, Enza; Sola, Daniele; Caramaschi, Alice; Mignone, Flavio; Bona, Elisa; Fallarini, Silvia
Organotrifluoroborate Sugar Conjugates for a Guided Boron Neutron Capture Therapy: From Synthesis to Positron Emission Tomography 1-gen-2022 Confalonieri, Laura; Imperio, Daniela; Erhard, Alvaro; Fallarini, Silvia; Compostella, Federica; Del Grosso, Erika; Balcerzyk, Marcin; Panza, Luigi
Synthesis, equilibrium, and biological study of a C-7 glucose boronic acid derivative as a potential candidate for boron neutron capture therapy 1-gen-2022 Muz, B.; Azab, A. K.; Confalonieri, L.; Del Grosso, E.; Fallarini, S.; Imperio, D.; Panza, L.
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 1-gen-2021 Fallarini, S.; Bhela, I. P.; Aprile, S.; Torre, E.; Ranza, A.; Orecchini, E.; Panfili, E.; Pallotta, M. T.; Massarotti, A.; Serafini, M.; Pirali, T.
Synthesis and characterisation of a boron-rich symmetric triazine bearing a hypoxia-targeting nitroimidazole moiety 1-gen-2021 Bunning, T. H.; Panza, L.; Azab, A. K.; Muz, B.; Fallarini, S.; Imperio, D.
Fucosylated ubiquitin and orthogonally glycosylated mutant A28C: conceptually new ligands for Burkholderia ambifaria lectin (BambL) 1-gen-2020 Kuhaudomlarp, Sakonwan; Cerofolini, Linda; Santarsia, Sabrina; Gillon, Emilie; Fallarini, Silvia; Lombardi, Grazia; Denis, Maxime; Giuntini, Stefano; Valori, Carolina; Fragai, Marco; Imberty, Anne; Dondoni, Alessandro; Nativi, Cristina
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 1-gen-2020 Serafini, M.; Torre, E.; Aprile, S.; Del Grosso, E.; Gesu, A.; Griglio, A.; Colombo, G.; Travelli, C.; Paiella, S.; Adamo, A.; Orecchini, E.; Coletti, A.; Pallotta, M. T.; Ugel, S.; Massarotti, A.; Pirali, T.; Fallarini, S.
Exploring calixarene-based clusters for efficient functional presentation of Streptococcus pneumoniae saccharides 1-gen-2019 Giuliani, M.; Faroldi, F.; Morelli, L.; Torre, E.; Lombardi, G.; Fallarini, S.; Sansone, F.; Compostella, F.
Anomeric sugar boronic acid analogues as potential agents for boron neutron capture therapy 1-gen-2019 Imperio, Daniela; Del Grosso, Erika; Fallarini, Silvia; Lombardi, Grazia; Panza, Luigi
Mostrati risultati da 1 a 20 di 89
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