Sfoglia per Autore
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1
2024-01-01 Panfili, Eleonora; Rezzi, Sarah Jane; Adamo, Annalisa; Mazzoletti, Daniele; Massarotti, Alberto; Miggiano, Riccardo; Fallarini, Silvia; Ambrosino, Sara; Coletti, Alice; Molinaro, Pasquale; Milella, Michele; Paiella, Salvatore; Macchiarulo, Antonio; Ugel, Stefano; Pirali, Tracey; Pallotta, Maria Teresa
Exploring the pharmaceutical potential of ammonium organotrifluoroborate functional group: Comprehensive chemical, metabolic, and plasma stability evaluation
2024-01-01 Villani, Salvatore; Imperio, Daniela; Panza, Luigi; Confalonieri, Laura; Fallarini, Silvia; Aprile, Silvio; Del Grosso, Erika
Selective inhibition of indoleamine and tryptophan 2,3-dioxygenases: Comparative study on kynurenine pathway in cell lines via LC-MS/MS-based targeted metabolomics
2024-01-01 Villani, Salvatore; Fallarini, Silvia; Rezzi, Sarah Jane; Di Martino, Rita Maria Concetta; Aprile, Silvio; Del Grosso, Erika
A Selective ALDH1A3 Inhibitor Impairs Mesothelioma 3-D Multicellular Spheroid Growth and Neutrophil Recruitment
2023-01-01 Boumya, Sara; Fallarini, Silvia; Siragusa, Sonia; Petrarolo, Giovanni; Aprile, Silvio; Audrito, Valentina; La Motta, Concettina; Garavaglia, Silvia; Moro, Laura; Pinton, Giulia
Niosomes as Biocompatible Scaffolds for the Multivalent Presentation of Tumor-Associated Antigens (TACAs) to the Immune System
2023-01-01 Fallarini, S.; Papi, F.; Licciardi, F.; Natali, F.; Lombardi, G.; Maestrelli, F.; Nativi, C.
Melanoma Cells Inhibit iNKT Cell Functions via PGE2 and IDO1
2023-01-01 Torre, E.; Pinton, G.; Lombardi, G.; Fallarini, S.
Synthesis, equilibrium, and biological study of a C-7 glucose boronic acid derivative as a potential candidate for boron neutron capture therapy
2022-01-01 Muz, B.; Azab, A. K.; Confalonieri, L.; Del Grosso, E.; Fallarini, S.; Imperio, D.; Panza, L.
Organotrifluoroborate Sugar Conjugates for a Guided Boron Neutron Capture Therapy: From Synthesis to Positron Emission Tomography
2022-01-01 Confalonieri, Laura; Imperio, Daniela; Erhard, Alvaro; Fallarini, Silvia; Compostella, Federica; Del Grosso, Erika; Balcerzyk, Marcin; Panza, Luigi
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors
2021-01-01 Fallarini, S.; Bhela, I. P.; Aprile, S.; Torre, E.; Ranza, A.; Orecchini, E.; Panfili, E.; Pallotta, M. T.; Massarotti, A.; Serafini, M.; Pirali, T.
A Pilot Study on Clinical Scores, Immune Cell Modulation, and Microbiota Composition in Allergic Patients with Rhinitis and Asthma Treated with a Probiotic Preparation
2021-01-01 Torre, Enza; Sola, Daniele; Caramaschi, Alice; Mignone, Flavio; Bona, Elisa; Fallarini, Silvia
Synthesis and characterisation of a boron-rich symmetric triazine bearing a hypoxia-targeting nitroimidazole moiety
2021-01-01 Bunning, T. H.; Panza, L.; Azab, A. K.; Muz, B.; Fallarini, S.; Imperio, D.
Fucosylated ubiquitin and orthogonally glycosylated mutant A28C: conceptually new ligands for Burkholderia ambifaria lectin (BambL)
2020-01-01 Kuhaudomlarp, Sakonwan; Cerofolini, Linda; Santarsia, Sabrina; Gillon, Emilie; Fallarini, Silvia; Lombardi, Grazia; Denis, Maxime; Giuntini, Stefano; Valori, Carolina; Fragai, Marco; Imberty, Anne; Dondoni, Alessandro; Nativi, Cristina
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity
2020-01-01 Serafini, M.; Torre, E.; Aprile, S.; Del Grosso, E.; Gesu, A.; Griglio, A.; Colombo, G.; Travelli, C.; Paiella, S.; Adamo, A.; Orecchini, E.; Coletti, A.; Pallotta, M. T.; Ugel, S.; Massarotti, A.; Pirali, T.; Fallarini, S.
Selectively charged and zwitterionic analogues of the smallest immunogenic structure of Streptococcus pneumoniae type 14
2019-01-01 Gragnani, T.; Cuffaro, D.; Fallarini, S.; Lombardi, G.; D'Andrea, F.; Guazzelli, L.
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors
2019-01-01 Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey
Anomeric sugar boronic acid analogues as potential agents for boron neutron capture therapy
2019-01-01 Imperio, Daniela; Del Grosso, Erika; Fallarini, Silvia; Lombardi, Grazia; Panza, Luigi
A Short and Convenient Synthesis of closo -Dodecaborate Sugar Conjugates
2019-01-01 Imperio, Daniela; Muz, Barbara; Azab, Abdel Kareem; Fallarini, Silvia; Lombardi, Grazia; Panza, Luigi
Exploring calixarene-based clusters for efficient functional presentation of Streptococcus pneumoniae saccharides
2019-01-01 Giuliani, M.; Faroldi, F.; Morelli, L.; Torre, E.; Lombardi, G.; Fallarini, S.; Sansone, F.; Compostella, F.
“In vitro” studies on galectin-3 in human natural killer cells
2018-01-01 Brittoli, Alvaro; Fallarini, Silvia; Zhang, Hao; Pieters, Roland J.; Lombardi, Grazia
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
2018-01-01 Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 | 1-gen-2024 | Panfili, Eleonora; Rezzi, Sarah Jane; Adamo, Annalisa; Mazzoletti, Daniele; Massarotti, Alberto; Miggiano, Riccardo; Fallarini, Silvia; Ambrosino, Sara; Coletti, Alice; Molinaro, Pasquale; Milella, Michele; Paiella, Salvatore; Macchiarulo, Antonio; Ugel, Stefano; Pirali, Tracey; Pallotta, Maria Teresa | |
Exploring the pharmaceutical potential of ammonium organotrifluoroborate functional group: Comprehensive chemical, metabolic, and plasma stability evaluation | 1-gen-2024 | Villani, Salvatore; Imperio, Daniela; Panza, Luigi; Confalonieri, Laura; Fallarini, Silvia; Aprile, Silvio; Del Grosso, Erika | |
Selective inhibition of indoleamine and tryptophan 2,3-dioxygenases: Comparative study on kynurenine pathway in cell lines via LC-MS/MS-based targeted metabolomics | 1-gen-2024 | Villani, Salvatore; Fallarini, Silvia; Rezzi, Sarah Jane; Di Martino, Rita Maria Concetta; Aprile, Silvio; Del Grosso, Erika | |
A Selective ALDH1A3 Inhibitor Impairs Mesothelioma 3-D Multicellular Spheroid Growth and Neutrophil Recruitment | 1-gen-2023 | Boumya, Sara; Fallarini, Silvia; Siragusa, Sonia; Petrarolo, Giovanni; Aprile, Silvio; Audrito, Valentina; La Motta, Concettina; Garavaglia, Silvia; Moro, Laura; Pinton, Giulia | |
Niosomes as Biocompatible Scaffolds for the Multivalent Presentation of Tumor-Associated Antigens (TACAs) to the Immune System | 1-gen-2023 | Fallarini, S.; Papi, F.; Licciardi, F.; Natali, F.; Lombardi, G.; Maestrelli, F.; Nativi, C. | |
Melanoma Cells Inhibit iNKT Cell Functions via PGE2 and IDO1 | 1-gen-2023 | Torre, E.; Pinton, G.; Lombardi, G.; Fallarini, S. | |
Synthesis, equilibrium, and biological study of a C-7 glucose boronic acid derivative as a potential candidate for boron neutron capture therapy | 1-gen-2022 | Muz, B.; Azab, A. K.; Confalonieri, L.; Del Grosso, E.; Fallarini, S.; Imperio, D.; Panza, L. | |
Organotrifluoroborate Sugar Conjugates for a Guided Boron Neutron Capture Therapy: From Synthesis to Positron Emission Tomography | 1-gen-2022 | Confalonieri, Laura; Imperio, Daniela; Erhard, Alvaro; Fallarini, Silvia; Compostella, Federica; Del Grosso, Erika; Balcerzyk, Marcin; Panza, Luigi | |
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors | 1-gen-2021 | Fallarini, S.; Bhela, I. P.; Aprile, S.; Torre, E.; Ranza, A.; Orecchini, E.; Panfili, E.; Pallotta, M. T.; Massarotti, A.; Serafini, M.; Pirali, T. | |
A Pilot Study on Clinical Scores, Immune Cell Modulation, and Microbiota Composition in Allergic Patients with Rhinitis and Asthma Treated with a Probiotic Preparation | 1-gen-2021 | Torre, Enza; Sola, Daniele; Caramaschi, Alice; Mignone, Flavio; Bona, Elisa; Fallarini, Silvia | |
Synthesis and characterisation of a boron-rich symmetric triazine bearing a hypoxia-targeting nitroimidazole moiety | 1-gen-2021 | Bunning, T. H.; Panza, L.; Azab, A. K.; Muz, B.; Fallarini, S.; Imperio, D. | |
Fucosylated ubiquitin and orthogonally glycosylated mutant A28C: conceptually new ligands for Burkholderia ambifaria lectin (BambL) | 1-gen-2020 | Kuhaudomlarp, Sakonwan; Cerofolini, Linda; Santarsia, Sabrina; Gillon, Emilie; Fallarini, Silvia; Lombardi, Grazia; Denis, Maxime; Giuntini, Stefano; Valori, Carolina; Fragai, Marco; Imberty, Anne; Dondoni, Alessandro; Nativi, Cristina | |
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity | 1-gen-2020 | Serafini, M.; Torre, E.; Aprile, S.; Del Grosso, E.; Gesu, A.; Griglio, A.; Colombo, G.; Travelli, C.; Paiella, S.; Adamo, A.; Orecchini, E.; Coletti, A.; Pallotta, M. T.; Ugel, S.; Massarotti, A.; Pirali, T.; Fallarini, S. | |
Selectively charged and zwitterionic analogues of the smallest immunogenic structure of Streptococcus pneumoniae type 14 | 1-gen-2019 | Gragnani, T.; Cuffaro, D.; Fallarini, S.; Lombardi, G.; D'Andrea, F.; Guazzelli, L. | |
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors | 1-gen-2019 | Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey | |
Anomeric sugar boronic acid analogues as potential agents for boron neutron capture therapy | 1-gen-2019 | Imperio, Daniela; Del Grosso, Erika; Fallarini, Silvia; Lombardi, Grazia; Panza, Luigi | |
A Short and Convenient Synthesis of closo -Dodecaborate Sugar Conjugates | 1-gen-2019 | Imperio, Daniela; Muz, Barbara; Azab, Abdel Kareem; Fallarini, Silvia; Lombardi, Grazia; Panza, Luigi | |
Exploring calixarene-based clusters for efficient functional presentation of Streptococcus pneumoniae saccharides | 1-gen-2019 | Giuliani, M.; Faroldi, F.; Morelli, L.; Torre, E.; Lombardi, G.; Fallarini, S.; Sansone, F.; Compostella, F. | |
“In vitro” studies on galectin-3 in human natural killer cells | 1-gen-2018 | Brittoli, Alvaro; Fallarini, Silvia; Zhang, Hao; Pieters, Roland J.; Lombardi, Grazia | |
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies | 1-gen-2018 | Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia |
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