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An adamantane-based ligand as a novel chemical tool for thermosensory TRPM8 channel therapeutic modulation 1-gen-2025 Lamberti, Angela; Aprile, Silvio; Cabañero, David; Travagin, Fabio; Butron, Laura; Fernández-Ballester, Gregorio; Tron, Gian Cesare; Fernández-Carvajal, Asia; Ferrer-Montiel, Antonio; Galli, Ubaldina
Visible Light Promoted Site‐Specific Functionalization of α‐Acyloxy Carboxamides: Unlocking a Forbidden Chemical Space in the Passerini Reaction 1-gen-2024 Brunelli, Francesca; Quartieri, Francesca; Miletto, Ivana; Pulici, Maurizio; Papeo, Gianluca; Tron, Gian Cesare
Exploiting the Different Nucleophilicity of the Isocyano Group: A Strategy for the Isocyanide Functionalization 1-gen-2024 Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare
Discovery of 2,3-Diaminoindole Derivatives as a Novel Class of NOD Antagonists 1-gen-2024 Russo, Camilla; Russomanno, Pasquale; D’Amore, Vincenzo Maria; Alfano, Antonella Ilenia; Santoro, Federica; Guzelj, Samo; Gobec, Martina; Amato, Jussara; Pagano, Bruno; Marinelli, Luciana; Carotenuto, Alfonso; Tron, Gian Cesare; Di Leva, Francesco Saverio; Jakopin, Žiga; Brancaccio, Diego; Giustiniano, Mariateresa
Each Interruption is an Opportunity: Novel Synthetic Strategies Explored Through Interrupted Click Reactions 1-gen-2024 Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare
Identification of novel aza-analogs of TN-16 as disrupters of microtubule dynamics through a multicomponent reaction 1-gen-2023 Foroutan, Arash; Corazzari, Marco; Grolla, Ambra A; Colombo, Giorgia; Travelli, Cristina; Genazzani, Armando A; Theeramunkong, Sewan; Galli, Ubaldina; Tron, Gian Cesare
Visible-Light Photoredox Catalysis in Water 1-gen-2023 Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Isocyanide‐Based Multicomponent Reactions Promoted by Visible Light Photoredox Catalysis 1-gen-2023 Russo, Camilla; Brunelli, Francesca; Cesare Tron, Gian; Giustiniano, Mariateresa
Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization 1-gen-2023 Cannalire, Rolando; Russo, Camilla; Luciano, Paolo; Cerra, Bruno; Gioiello, Antimo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Sulfur‐Centered Radicals in Visible Light Isocyanide Photochemistry 1-gen-2023 Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Isocyanides in med chem: A scaffold hopping approach for the identification of novel 4-isocyanophenylamides as potent antibacterial agents against methicillin-resistant Staphylococcus aureus 1-gen-2023 Brunelli, F.; Ceresa, C.; Aprile, S.; Coppo, L.; Castiglioni, B.; Bosetti, M.; Fracchia, L.; Tron, G. C.
Synthesis of Novel Lipophilic Polyamines via Ugi Reaction and Evaluation of Their Anticancer Activity 1-gen-2022 Nichugovskiy, Artemiy; Maksimova, Varvara; Trapeznikova, Ekaterina; Eshtukova-Shcheglova, Elizaveta; Ivanov, Igor; Yakubovskaya, Marianna; Kirsanov, Kirill; Cheshkov, Dmitry; Tron, Gian Cesare; Maslov, Mikhail
Visible-light photocatalytic metal-free multicomponent Ugi-like chemistry 1-gen-2022 Russo, Camilla; Graziani, Giulia; Cannalire, Rolando; Tron, Gian Cesare; Giustiniano, Mariateresa
Expanding the Chemical Space of Drug-like Passerini Compounds: Can α-Acyloxy Carboxamides Be Considered Hard Drugs? 1-gen-2022 Brunelli, F.; Ceresa, C.; Fracchia, L.; Tron, G. C.; Aprile, S.
Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions 1-gen-2022 Cannalire, Rolando; Santoro, Federica; Russo, Camilla; Graziani, Giulia; Tron, Gian Cesare; Carotenuto, Alfonso; Brancaccio, Diego; Giustiniano, Mariateresa
In-water synthesis of isocyanides under micellar conditions 1-gen-2022 Brunelli, F.; Aprile, S.; Russo, C.; Giustiniano, M.; Tron, G. C.
Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives 1-gen-2021 Russo, C.; Cannalire, R.; Luciano, P.; Brunelli, F.; Tron, G. C.; Giustiniano, M.
Medicinal Chemistry of Isocyanides 1-gen-2021 Massarotti, A.; Brunelli, F.; Aprile, S.; Giustiniano, M.; Tron, G. C.
The 115 Year Old Multicomponent Bargellini Reaction: Perspectives and New Applications 1-gen-2021 Serafini, Marta; Murgia, Ilaria; Giustiniano, Mariateresa; Pirali, Tracey; Tron, Gian Cesare
Visible light photocatalysis in the late-stage functionalization of pharmaceutically relevant compounds 1-gen-2021 Cannalire, R.; Pelliccia, S.; Sancineto, L.; Novellino, E.; Tron, G. C.; Giustiniano, M.
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