Sfoglia per Autore
An adamantane-based ligand as a novel chemical tool for thermosensory TRPM8 channel therapeutic modulation
2025-01-01 Lamberti, Angela; Aprile, Silvio; Cabañero, David; Travagin, Fabio; Butron, Laura; Fernández-Ballester, Gregorio; Tron, Gian Cesare; Fernández-Carvajal, Asia; Ferrer-Montiel, Antonio; Galli, Ubaldina
Visible Light Promoted Site‐Specific Functionalization of α‐Acyloxy Carboxamides: Unlocking a Forbidden Chemical Space in the Passerini Reaction
2024-01-01 Brunelli, Francesca; Quartieri, Francesca; Miletto, Ivana; Pulici, Maurizio; Papeo, Gianluca; Tron, Gian Cesare
Exploiting the Different Nucleophilicity of the Isocyano Group: A Strategy for the Isocyanide Functionalization
2024-01-01 Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare
Discovery of 2,3-Diaminoindole Derivatives as a Novel Class of NOD Antagonists
2024-01-01 Russo, Camilla; Russomanno, Pasquale; D’Amore, Vincenzo Maria; Alfano, Antonella Ilenia; Santoro, Federica; Guzelj, Samo; Gobec, Martina; Amato, Jussara; Pagano, Bruno; Marinelli, Luciana; Carotenuto, Alfonso; Tron, Gian Cesare; Di Leva, Francesco Saverio; Jakopin, Žiga; Brancaccio, Diego; Giustiniano, Mariateresa
Each Interruption is an Opportunity: Novel Synthetic Strategies Explored Through Interrupted Click Reactions
2024-01-01 Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare
Identification of novel aza-analogs of TN-16 as disrupters of microtubule dynamics through a multicomponent reaction
2023-01-01 Foroutan, Arash; Corazzari, Marco; Grolla, Ambra A; Colombo, Giorgia; Travelli, Cristina; Genazzani, Armando A; Theeramunkong, Sewan; Galli, Ubaldina; Tron, Gian Cesare
Visible-Light Photoredox Catalysis in Water
2023-01-01 Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Isocyanide‐Based Multicomponent Reactions Promoted by Visible Light Photoredox Catalysis
2023-01-01 Russo, Camilla; Brunelli, Francesca; Cesare Tron, Gian; Giustiniano, Mariateresa
Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization
2023-01-01 Cannalire, Rolando; Russo, Camilla; Luciano, Paolo; Cerra, Bruno; Gioiello, Antimo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Sulfur‐Centered Radicals in Visible Light Isocyanide Photochemistry
2023-01-01 Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa
Isocyanides in med chem: A scaffold hopping approach for the identification of novel 4-isocyanophenylamides as potent antibacterial agents against methicillin-resistant Staphylococcus aureus
2023-01-01 Brunelli, F.; Ceresa, C.; Aprile, S.; Coppo, L.; Castiglioni, B.; Bosetti, M.; Fracchia, L.; Tron, G. C.
Visible-light photocatalytic metal-free multicomponent Ugi-like chemistry
2022-01-01 Russo, Camilla; Graziani, Giulia; Cannalire, Rolando; Tron, Gian Cesare; Giustiniano, Mariateresa
Expanding the Chemical Space of Drug-like Passerini Compounds: Can α-Acyloxy Carboxamides Be Considered Hard Drugs?
2022-01-01 Brunelli, F.; Ceresa, C.; Fracchia, L.; Tron, G. C.; Aprile, S.
Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions
2022-01-01 Cannalire, Rolando; Santoro, Federica; Russo, Camilla; Graziani, Giulia; Tron, Gian Cesare; Carotenuto, Alfonso; Brancaccio, Diego; Giustiniano, Mariateresa
In-water synthesis of isocyanides under micellar conditions
2022-01-01 Brunelli, F.; Aprile, S.; Russo, C.; Giustiniano, M.; Tron, G. C.
Synthesis of Novel Lipophilic Polyamines via Ugi Reaction and Evaluation of Their Anticancer Activity
2022-01-01 Nichugovskiy, Artemiy; Maksimova, Varvara; Trapeznikova, Ekaterina; Eshtukova-Shcheglova, Elizaveta; Ivanov, Igor; Yakubovskaya, Marianna; Kirsanov, Kirill; Cheshkov, Dmitry; Tron, Gian Cesare; Maslov, Mikhail
Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives
2021-01-01 Russo, C.; Cannalire, R.; Luciano, P.; Brunelli, F.; Tron, G. C.; Giustiniano, M.
Medicinal Chemistry of Isocyanides
2021-01-01 Massarotti, A.; Brunelli, F.; Aprile, S.; Giustiniano, M.; Tron, G. C.
The 115 Year Old Multicomponent Bargellini Reaction: Perspectives and New Applications
2021-01-01 Serafini, Marta; Murgia, Ilaria; Giustiniano, Mariateresa; Pirali, Tracey; Tron, Gian Cesare
Tritylamine as an ammonia surrogate in the ugi reaction provides access to unprecedented 5-sulfamido oxazoles using burgess-type reagents
2021-01-01 Bhela, I. P.; Serafini, M.; Del Grosso, E.; Tron, G. C.; Pirali, T.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| An adamantane-based ligand as a novel chemical tool for thermosensory TRPM8 channel therapeutic modulation | 1-gen-2025 | Lamberti, Angela; Aprile, Silvio; Cabañero, David; Travagin, Fabio; Butron, Laura; Fernández-Ballester, Gregorio; Tron, Gian Cesare; Fernández-Carvajal, Asia; Ferrer-Montiel, Antonio; Galli, Ubaldina | |
| Visible Light Promoted Site‐Specific Functionalization of α‐Acyloxy Carboxamides: Unlocking a Forbidden Chemical Space in the Passerini Reaction | 1-gen-2024 | Brunelli, Francesca; Quartieri, Francesca; Miletto, Ivana; Pulici, Maurizio; Papeo, Gianluca; Tron, Gian Cesare | |
| Exploiting the Different Nucleophilicity of the Isocyano Group: A Strategy for the Isocyanide Functionalization | 1-gen-2024 | Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare | |
| Discovery of 2,3-Diaminoindole Derivatives as a Novel Class of NOD Antagonists | 1-gen-2024 | Russo, Camilla; Russomanno, Pasquale; D’Amore, Vincenzo Maria; Alfano, Antonella Ilenia; Santoro, Federica; Guzelj, Samo; Gobec, Martina; Amato, Jussara; Pagano, Bruno; Marinelli, Luciana; Carotenuto, Alfonso; Tron, Gian Cesare; Di Leva, Francesco Saverio; Jakopin, Žiga; Brancaccio, Diego; Giustiniano, Mariateresa | |
| Each Interruption is an Opportunity: Novel Synthetic Strategies Explored Through Interrupted Click Reactions | 1-gen-2024 | Brunelli, Francesca; Russo, Camilla; Giustiniano, Mariateresa; Tron, Gian Cesare | |
| Identification of novel aza-analogs of TN-16 as disrupters of microtubule dynamics through a multicomponent reaction | 1-gen-2023 | Foroutan, Arash; Corazzari, Marco; Grolla, Ambra A; Colombo, Giorgia; Travelli, Cristina; Genazzani, Armando A; Theeramunkong, Sewan; Galli, Ubaldina; Tron, Gian Cesare | |
| Visible-Light Photoredox Catalysis in Water | 1-gen-2023 | Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa | |
| Isocyanide‐Based Multicomponent Reactions Promoted by Visible Light Photoredox Catalysis | 1-gen-2023 | Russo, Camilla; Brunelli, Francesca; Cesare Tron, Gian; Giustiniano, Mariateresa | |
| Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization | 1-gen-2023 | Cannalire, Rolando; Russo, Camilla; Luciano, Paolo; Cerra, Bruno; Gioiello, Antimo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa | |
| Sulfur‐Centered Radicals in Visible Light Isocyanide Photochemistry | 1-gen-2023 | Russo, Camilla; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa | |
| Isocyanides in med chem: A scaffold hopping approach for the identification of novel 4-isocyanophenylamides as potent antibacterial agents against methicillin-resistant Staphylococcus aureus | 1-gen-2023 | Brunelli, F.; Ceresa, C.; Aprile, S.; Coppo, L.; Castiglioni, B.; Bosetti, M.; Fracchia, L.; Tron, G. C. | |
| Visible-light photocatalytic metal-free multicomponent Ugi-like chemistry | 1-gen-2022 | Russo, Camilla; Graziani, Giulia; Cannalire, Rolando; Tron, Gian Cesare; Giustiniano, Mariateresa | |
| Expanding the Chemical Space of Drug-like Passerini Compounds: Can α-Acyloxy Carboxamides Be Considered Hard Drugs? | 1-gen-2022 | Brunelli, F.; Ceresa, C.; Fracchia, L.; Tron, G. C.; Aprile, S. | |
| Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions | 1-gen-2022 | Cannalire, Rolando; Santoro, Federica; Russo, Camilla; Graziani, Giulia; Tron, Gian Cesare; Carotenuto, Alfonso; Brancaccio, Diego; Giustiniano, Mariateresa | |
| In-water synthesis of isocyanides under micellar conditions | 1-gen-2022 | Brunelli, F.; Aprile, S.; Russo, C.; Giustiniano, M.; Tron, G. C. | |
| Synthesis of Novel Lipophilic Polyamines via Ugi Reaction and Evaluation of Their Anticancer Activity | 1-gen-2022 | Nichugovskiy, Artemiy; Maksimova, Varvara; Trapeznikova, Ekaterina; Eshtukova-Shcheglova, Elizaveta; Ivanov, Igor; Yakubovskaya, Marianna; Kirsanov, Kirill; Cheshkov, Dmitry; Tron, Gian Cesare; Maslov, Mikhail | |
| Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives | 1-gen-2021 | Russo, C.; Cannalire, R.; Luciano, P.; Brunelli, F.; Tron, G. C.; Giustiniano, M. | |
| Medicinal Chemistry of Isocyanides | 1-gen-2021 | Massarotti, A.; Brunelli, F.; Aprile, S.; Giustiniano, M.; Tron, G. C. | |
| The 115 Year Old Multicomponent Bargellini Reaction: Perspectives and New Applications | 1-gen-2021 | Serafini, Marta; Murgia, Ilaria; Giustiniano, Mariateresa; Pirali, Tracey; Tron, Gian Cesare | |
| Tritylamine as an ammonia surrogate in the ugi reaction provides access to unprecedented 5-sulfamido oxazoles using burgess-type reagents | 1-gen-2021 | Bhela, I. P.; Serafini, M.; Del Grosso, E.; Tron, G. C.; Pirali, T. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile