ALBERTI, MARTA
ALBERTI, MARTA
Dipartimento di Scienze del Farmaco
An alternative conformation of the N-terminal loop of human dihydroorotate dehydrogenase drives binding to a potent antiproliferative agent
2024-01-01 Alberti, Marta; Poli, Giulio; Broggini, Luca; Sainas, Stefano; Rizzi, Menico; Boschi, Donatella; Ferraris, Davide M; Martino, Elena; Ricagno, Stefano; Tuccinardi, Tiziano; Lolli, Marco L; Miggiano, Riccardo
Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity
2025-01-01 Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L.; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo
Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor
2023-01-01 Alberti, Marta; Sainas, Stefano; Ronchi, Erika; Lolli, Marco L; Boschi, Donatella; Rizzi, Menico; Ferraris, Davide M; Miggiano, Riccardo
Fluorescent Isostere (Fluostere) of the Carboxylate: Design of hDHODH Fluorescent Inhibitors as Proof of Concept
2025-01-01 Sainas, S.; Martino, E.; Garino, C.; Circosta, P.; Luganini, A.; Giorgis, M.; Bavo, F.; Piccinini, M.; Ramondetti, C.; Alberti, M.; Miggiano, R.; Gribaudo, G.; Boschi, D.; Frolund, B.; Lolli, M. L.
Rationally-driven targeting of dihydroorotate dehydrogenase: key enzyme of pyrimidine biosynthesis pathway
2024-01-01 Alberti, Marta
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety
2022-01-01 Sainas, Stefano; Giorgis, Marta; Circosta, Paola; Poli, Giulio; Alberti, Marta; Passoni, Alice; Gaidano, Valentina; Pippione, Agnese C; Vitale, Nicoletta; Bonanni, Davide; Rolando, Barbara; Cignetti, Alessandro; Ramondetti, Cristina; Lanno, Alessia; Ferraris, Davide M; Canepa, Barbara; Buccinnà, Barbara; Piccinini, Marco; Rizzi, Menico; Saglio, Giuseppe; Al-Karadaghi, Salam; Boschi, Donatella; Miggiano, Riccardo; Tuccinardi, Tiziano; Lolli, Marco L
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| An alternative conformation of the N-terminal loop of human dihydroorotate dehydrogenase drives binding to a potent antiproliferative agent | 1-gen-2024 | Alberti, Marta; Poli, Giulio; Broggini, Luca; Sainas, Stefano; Rizzi, Menico; Boschi, Donatella; Ferraris, Davide M; Martino, Elena; Ricagno, Stefano; Tuccinardi, Tiziano; Lolli, Marco L; Miggiano, Riccardo | |
| Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity | 1-gen-2025 | Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L.; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo | |
| Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor | 1-gen-2023 | Alberti, Marta; Sainas, Stefano; Ronchi, Erika; Lolli, Marco L; Boschi, Donatella; Rizzi, Menico; Ferraris, Davide M; Miggiano, Riccardo | |
| Fluorescent Isostere (Fluostere) of the Carboxylate: Design of hDHODH Fluorescent Inhibitors as Proof of Concept | 1-gen-2025 | Sainas, S.; Martino, E.; Garino, C.; Circosta, P.; Luganini, A.; Giorgis, M.; Bavo, F.; Piccinini, M.; Ramondetti, C.; Alberti, M.; Miggiano, R.; Gribaudo, G.; Boschi, D.; Frolund, B.; Lolli, M. L. | |
| Rationally-driven targeting of dihydroorotate dehydrogenase: key enzyme of pyrimidine biosynthesis pathway | 1-gen-2024 | Alberti, Marta | |
| Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety | 1-gen-2022 | Sainas, Stefano; Giorgis, Marta; Circosta, Paola; Poli, Giulio; Alberti, Marta; Passoni, Alice; Gaidano, Valentina; Pippione, Agnese C; Vitale, Nicoletta; Bonanni, Davide; Rolando, Barbara; Cignetti, Alessandro; Ramondetti, Cristina; Lanno, Alessia; Ferraris, Davide M; Canepa, Barbara; Buccinnà, Barbara; Piccinini, Marco; Rizzi, Menico; Saglio, Giuseppe; Al-Karadaghi, Salam; Boschi, Donatella; Miggiano, Riccardo; Tuccinardi, Tiziano; Lolli, Marco L |