MERCALLI, VALENTINA
MERCALLI, VALENTINA
Dipartimento di Scienze del Farmaco
An efficient synthesis of 1-arylindazole-3-carboxamides using nitrile imines, isocyanides and 2-hydroxymethylbenzoic acid, followed by a chemoselective Buchwald–Hartwig intramolecular cyclization
2016-01-01 Giustiniano, M.; Mercalli, Valentina; Novellino, E.; Tron, Gian Cesare
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?
2014-01-01 Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare
Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement
2015-01-01 Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare
N-N bond formation in Ugi processes: from nitric acid to libraries of nitramines
2017-01-01 Mercalli, Valentina; Nyadanu, Aude; Cordier, Marie; Tron, Gian Cesare; Grimaud, Laurence; El Kaim, Laurent
Nitrile N-oxides and nitrile imines as electrophilic partners for the discovery of novel isocyanide multicomponent reactions: an innovative strategy for the synthesis of molecular scaffolds useful in medicinal chemistry
2017-01-01 Mercalli, Valentina
Reaction Between (Z)-Arylchlorooximes and alpha-Isocyanoacetamides: a Procedure For The Synthesis of Aryl-alpha-Ketoamide amides
2014-01-01 Giustiniano, Mariateresa; Mercalli, Valentina; Cassese, Hilde; Di Maro, Salvatore; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare
Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols
2014-01-01 Mercalli, Valentina; M., Giustiniano; DEL GROSSO, Erika; Varese, Monica; H., Cassese; Massarotti, Alberto; E., Novellino; Tron, Gian Cesare
SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS
2016-01-01 Mercalli, Valentina; Massarotti, Alberto; Baldanzi, Gianluca; Graziani, A.; Tron, Gian Cesare
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis
2017-01-01 Giustiniano, Mariateresa; Basso, Andrea; Mercalli, Valentina; Massarotti, Alberto; Novellino, Ettore; Tron, Gian Cesare; Zhu, Jieping
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles
2019-01-01 Levré, Doriana; Arcisto, Chiara; Mercalli, Valentina; Massarotti, Alberto
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| An efficient synthesis of 1-arylindazole-3-carboxamides using nitrile imines, isocyanides and 2-hydroxymethylbenzoic acid, followed by a chemoselective Buchwald–Hartwig intramolecular cyclization | 1-gen-2016 | Giustiniano, M.; Mercalli, Valentina; Novellino, E.; Tron, Gian Cesare | |
| Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? | 1-gen-2014 | Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare | |
| Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 1-gen-2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare | |
| Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 1-gen-2017 | Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare | |
| Multicomponent Reaction of Z-Chlorooximes, Isocyanides, and Hydroxylamines as Hypernucleophilic Traps. A One-Pot Route to Aminodioximes and Their Transformation into 5-Amino-1,2,4-oxadiazoles by Mitsunobu-Beckmann Rearrangement | 1-gen-2015 | Mercalli, Valentina; Massarotti, Alberto; Varese, Monica; Giustiniano, Mariateresa; Meneghetti, Fiorella; Novellino, Ettore; Tron, Gian Cesare | |
| N-N bond formation in Ugi processes: from nitric acid to libraries of nitramines | 1-gen-2017 | Mercalli, Valentina; Nyadanu, Aude; Cordier, Marie; Tron, Gian Cesare; Grimaud, Laurence; El Kaim, Laurent | |
| Nitrile N-oxides and nitrile imines as electrophilic partners for the discovery of novel isocyanide multicomponent reactions: an innovative strategy for the synthesis of molecular scaffolds useful in medicinal chemistry | 1-gen-2017 | Mercalli, Valentina | |
| Reaction Between (Z)-Arylchlorooximes and alpha-Isocyanoacetamides: a Procedure For The Synthesis of Aryl-alpha-Ketoamide amides | 1-gen-2014 | Giustiniano, Mariateresa; Mercalli, Valentina; Cassese, Hilde; Di Maro, Salvatore; Galli, Ubaldina; Novellino, Ettore; Tron, Gian Cesare | |
| Solution-Phase Parallel Synthesis of Aryloxyimino Amides via a Novel Multicomponent Reaction among Aromatic (Z)‑Chlorooximes, Isocyanides, and Electron-Deficient Phenols | 1-gen-2014 | Mercalli, Valentina; M., Giustiniano; DEL GROSSO, Erika; Varese, Monica; H., Cassese; Massarotti, Alberto; E., Novellino; Tron, Gian Cesare | |
| SYNTHESIS AND CHARACTERIZATION OF NEW DGKα INHIBITORS | 1-gen-2016 | Mercalli, Valentina; Massarotti, Alberto; Baldanzi, Gianluca; Graziani, A.; Tron, Gian Cesare | |
| To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis | 1-gen-2017 | Giustiniano, Mariateresa; Basso, Andrea; Mercalli, Valentina; Massarotti, Alberto; Novellino, Ettore; Tron, Gian Cesare; Zhu, Jieping | |
| ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles | 1-gen-2019 | Levré, Doriana; Arcisto, Chiara; Mercalli, Valentina; Massarotti, Alberto |