TRON, Gian Cesare

TRON, Gian Cesare  

Dipartimento di Scienze del Farmaco  

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Titolo Data di pubblicazione Autore(i) File
A Concise Entry into Nonsymmetrical Alkyl Polyamines 1-gen-2008 Pirali, Tracey; Callipari, G; Ercolano, E; Genazzani, Aa; Giovenzana, Giovanni Battista; Tron, Gian Cesare
A concise entry into nonsymmetrical alkyl polyamines 1-gen-2008 Pirali, Tracey; Callipari, G; Ercolano, E; Genazzani, Armando; Giovenzana, Giovanni Battista; Tron, Gian Cesare
A fast route for the synthesis of tetrazolyl oximes by a novel multicomponent reaction between Z-chlorooximes, isocyanides and trimethylsilyl azide 1-gen-2017 Mariateresa, Giustiniano; Sveva, Pelliccia; Ana Belen, Muñoz garcia; Michele, Pavone; Bruno, Pagano; Galli, Ubaldina; Ettore, Novellino; Tron, Gian Cesare
A Mimicry of Primary Amines by Bis-Secondary Diamines as Components in the Ugi Four-Component Reaction 1-gen-2006 Giovenzana, Giovanni Battista; Tron, Gian Cesare; DI PAOLA, Stefano; Menegotto, Ivan Guglielmo; Pirali, Tracey
A novel alpha-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates 1-gen-2011 Mossetti, Riccardo; Caprioglio, Diego; Colombano, Giampiero; Tron, Gian Cesare; Pirali, Tracey
A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry 1-gen-2010 Colombano, Giampiero; Travelli, Cristina; Galli, Ubaldina; Caldarelli, Antonio; Chini, Mg; Canonico, Pier Luigi; Sorba, Giovanni; Bifulco, G; Tron, Gian Cesare; Genazzani, Armando
A novel α-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates 1-gen-2011 Mossetti, R; Caprioglio, D; Colombano, G; Tron, Gian Cesare; Pirali, Tracey
A practical synthesis of 5-aroyl-1-aryltetrazoles using an Ugi-like 4-component reaction followed by a biomimetic transamination 1-gen-2010 Giustiniano, M; Pirali, Tracey; Massarotti, Alberto; Biletta, B; Novellino, E; Campiglia, P; Sorba, Giovanni; Tron, Gian Cesare
A Successful Replacement of Phenols with Isocyanides in the Bargellini Reaction: Synthesis of 3-Carboxamido-Isobutyric Acids 1-gen-2016 Giustiniano, Mariateresa; Pelliccia, Sveva; Galli, Ubaldina; Amato, Jussara; Travagin, Fabio; Novellino, Ettore; Tron, Gian Cesare
A three-component synthesis of (1,3-oxazol-2-yl)-1,2-dihydro(iso)quinoline and its further structural diversifications 1-gen-2005 Tron, Gian Cesare; Jieping, Zhu
Ammonium Chloride Promoted Three-Component Synthesis of 5-Iminooxazoline and its Subsequent Transformation to Macrocyclodepsipeptide 1-gen-2007 Pirali, Tracey; Tron, Gian Cesare; Masson, G; Zhu, J.
Amphoteric 2-(sulfonylamino)benzaldehydes, secondary amines and isocyanides in the multicomponent synthesis of elusive N-alkyl-2,3-diaminoindoles 1-gen-2017 Mariateresa, Giustiniano; Sveva, Pelliccia; Luca, Sangaletti; Fiorella, Meneghetti; Jussara, Amato; Ettore, Novellino; Tron, Gian Cesare
An efficient synthesis of 1-arylindazole-3-carboxamides using nitrile imines, isocyanides and 2-hydroxymethylbenzoic acid, followed by a chemoselective Buchwald–Hartwig intramolecular cyclization 1-gen-2016 Giustiniano, M.; Mercalli, Valentina; Novellino, E.; Tron, Gian Cesare
An efficient synthesis of symmetric and unsymmetric bis-(ß-aminoamides) via Ugi multicomponent reaction. 1-gen-2012 La Spisa, F; Feo, A; Mossetti, R; Tron, Gian Cesare
An expeditious procedure for the isolation of ingenol from the seeds of Euphorbia lathyris 1-gen-1999 Appendino, Giovanni Battista; Tron, Gian Cesare; Cravotto, ; Palmisano, G.; Jakupovic, J.
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? 1-gen-2014 Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare
Are the 1,4 and 1,5-disubstituted-1,2,3-triazoles good pharmacophoric groups? 1-gen-2012 Massarotti, Alberto; Genazzani, A. A.; Tron, Gian Cesare
Aryl Azides as Forgotten Electrophiles in the Van Leusen Reaction: A Multicomponent Transformation Affording 4-Tosyl-1-arylimidazoles 1-gen-2019 Necardo, Cristiana; Alfano, Antonella Ilenia; Del Grosso, Erika; Pelliccia, Sveva; Galli, Ubaldina; Novellino, Ettore; Meneghetti, Fiorella; Giustiniano, Mariateresa; Tron, Gian Cesare
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 1-gen-2020 Pelliccia, Sveva; Amato, Jussara; Capasso, Domenica; Di Gaetano, Sonia; Massarotti, Alberto; Piccolo, Marialuisa; Irace, Carlo; Tron, Gian Cesare; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Giustiniano, Mariateresa
Bisnorsesquiterpenoids from Euphorbia resinifera berg. and an expeditious procedure to obtain resiniferatoxin from its fresh latex 1-gen-2002 Fattorusso, E.; Lanzotti, V.; TAGLIALATELA SCAFATA, O.; Tron, Gian Cesare; Appendino, Giovanni Battista