Sfoglia per Autore
Arzanol, a natural phloroglucinol α‐pyrone, protects HaCaT keratinocytes against H2O2‐induced oxidative stress, counteracting cytotoxicity, reactive oxygen species generation, apoptosis, and mitochondrial depolarization
2024-01-01 Piras, Franca; Sogos, Valeria; Pollastro, Federica; Appendino, Giovanni; Rosa, Antonella
Comparative Evaluation of Anticancer Activity of Natural Methoxylated Flavones Xanthomicrol and Eupatilin in A375 Skin Melanoma Cells
2024-01-01 Rosa, Antonella; Piras, Franca; Pollastro, Federica; Sogos, Valeria; Appendino, Giovanni; Nieddu, Mariella
Novel Skeletal Rearrangements of the Tigliane Diterpenoid Core
2023-01-01 Maioli, Chiara; Amin, Hawraz Ibrahim M.; Chianese, Giuseppina; Minassi, Alberto; Reddell, Paul W.; Gaeta, Simone; Taglialatela-Scafati, Orazio; Appendino, Giovanni
PPARα/γ-Targeting Amorfrutin Phytocannabinoids from Aerial Parts of Glycyrrhiza foetida
2023-01-01 Serino, Elena; Iannotti, Fabio Arturo; Al-Hmadi, Hekmat B.; Caprioglio, Diego; Moriello, Claudia; Masi, Francesca; Hammami, Saoussen; Appendino, Giovanni; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio
Synthesis and biological evaluation of hydroxamate isosteres of acidic cannabinoids
2023-01-01 Amin, Hawraz Ibrahim M.; Ruiz-Pino, Francisco; Collado, Juan A.; Appendino, Giovanni; Tena-Sempere, Manuel; Munoz, Eduardo; Caprioglio, Diego
Non-Volatile Terpenoids and Lipophilic Flavonoids from Achillea erba-rotta Subsp. moschata (Wulfen) I. Richardson
2023-01-01 Salamone, Stefano; Aiello, Nicola; Fusani, Pietro; Rosa, Antonella; Nieddu, Mariella; Appendino, Giovanni; Pollastro, Federica
Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators
2023-01-01 Peltner, Lukas K; Gluthmann, Lars; Börner, Friedemann; Pace, Simona; Hoffstetter, Robert K; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E; Gilbert, Nathaniel C; Werz, Oliver; Jordan, Paul M
Rotational constriction of curcuminoids impacts 5-lipoxygenase and mPGES-1 inhibition and evokes a lipid mediator class switch in macrophages
2022-01-01 Rao, Zhigang; Caprioglio, Diego; Gollowitzer, Andre; Kretzer, Christian; Imperio, Daniela; Collado, Juan A.; Waltl, Lorenz; Lackner, Sandra; Appendino, Giovanni Battista; Munoz, Eduardo; Temml, Veronika; Werz, Oliver; Minassi, Alberto; Koeberle, Andreas
Minor Phytocannabinoids: A Misleading Name but a Promising Opportunity for Biomedical Research
2022-01-01 Caprioglio, Diego; Amin, Hawraz Ibrahim M.; Taglialatela-Scafati, Orazio; Muñoz, Eduardo; Appendino, Giovanni
One‐Pot Oxidative Heterofunctionalization of Resorcinolic Cannabinoids to Non‐thiophilic Aminocannabinoquinones
2022-01-01 Caprioglio, Diego; Mattoteia, Daiana; Muñoz, Eduardo; Taglialatela‐scafati, Orazio; Appendino, Giovanni
Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex
2022-01-01 Funamoto, M.; Sunagawa, Y.; Gempei, M.; Shimizu, K.; Katanasaka, Y.; Shimizu, S.; Hamabe-Horiike, T.; Appendino, G.; Minassi, A.; Koeberle, A.; Komiyama, M.; Mori, K.; Hasegawa, K.; Morimoto, T.
Δ9-cis-Tetrahydrocannabinol: Natural Occurrence, Chirality, and Pharmacology
2021-01-01 Schafroth, Michael A; Mazzoccanti, Giulia; Reynoso-Moreno, Ines; Erni, Reto; Pollastro, Federica; Caprioglio, Diego; Botta, Bruno; Allegrone, Gianna; Grassi, Giulio; Chicca, Andrea; Gasparrini, Francesco; Gertsch, Jürg; Carreira, Erick M; Appendino, Giovanni
Agathadiol, a labdane diterpenoid from juniper berries, is a positive allosteric modulator of CB1R
2021-01-01 Salamone, Stefano; Appendino, Giovanni; Khalili, Adil; Pollastro, Federica; Munoz, Eduardo; Unciti-Broceta, Juan D
EHP-101 alleviates angiotensin II-induced fibrosis and inflammation in mice
2021-01-01 Garcia-Martin, A.; Navarrete, C.; Garrido-Rodriguez, M.; Prados, M. E.; Caprioglio, D.; Appendino, G.; Munoz, E.
Betulinic acid hydroxamate prevents colonic inflammation and fibrosis in murine models of inflammatory bowel disease
2021-01-01 Prados, M. E.; Garcia-Martin, A.; Unciti-Broceta, J. D.; Palomares, B.; Collado, J. A.; Minassi, A.; Calzado, M. A.; Appendino, G.; Munoz, E.
Betulinic Acid Hydroxamate is Neuroprotective and Induces Protein Phosphatase 2A-Dependent HIF-1α Stabilization and Post-transcriptional Dephosphorylation of Prolyl Hydrolase 2
2021-01-01 Prados, M. E.; Correa-Saez, A.; Unciti-Broceta, J. D.; Garrido-Rodriguez, M.; Jimenez-Jimenez, C.; Mazzone, M.; Minassi, A.; Appendino, G.; Calzado, M. A.; Munoz, E.
The combined effect of branching and elongation on the bioactivity profile of phytocannabinoids. Part i: Thermo-trps
2021-01-01 Mattoteia, D.; Moriello, A. S.; Taglialatela-Scafati, O.; Amodeo, P.; De Petrocellis, L.; Appendino, G.; Vitale, R. M.; Caprioglio, D.
Cannabinoquinones: Synthesis and biological profile
2021-01-01 Caprioglio, D.; Mattoteia, D.; Taglialatela-Scafati, O.; Munoz, E.; Appendino, G.
Icilio Guareschi and his amazing “1897 reaction”
2021-01-01 Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G.
Best practice in research – Overcoming common challenges in phytopharmacological research
2020-01-01 Heinrich, M.; Appendino, G.; Efferth, T.; Furst, R.; Izzo, A. A.; Kayser, O.; Pezzuto, J. M.; Viljoen, A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Arzanol, a natural phloroglucinol α‐pyrone, protects HaCaT keratinocytes against H2O2‐induced oxidative stress, counteracting cytotoxicity, reactive oxygen species generation, apoptosis, and mitochondrial depolarization | 1-gen-2024 | Piras, Franca; Sogos, Valeria; Pollastro, Federica; Appendino, Giovanni; Rosa, Antonella | |
Comparative Evaluation of Anticancer Activity of Natural Methoxylated Flavones Xanthomicrol and Eupatilin in A375 Skin Melanoma Cells | 1-gen-2024 | Rosa, Antonella; Piras, Franca; Pollastro, Federica; Sogos, Valeria; Appendino, Giovanni; Nieddu, Mariella | |
Novel Skeletal Rearrangements of the Tigliane Diterpenoid Core | 1-gen-2023 | Maioli, Chiara; Amin, Hawraz Ibrahim M.; Chianese, Giuseppina; Minassi, Alberto; Reddell, Paul W.; Gaeta, Simone; Taglialatela-Scafati, Orazio; Appendino, Giovanni | |
PPARα/γ-Targeting Amorfrutin Phytocannabinoids from Aerial Parts of Glycyrrhiza foetida | 1-gen-2023 | Serino, Elena; Iannotti, Fabio Arturo; Al-Hmadi, Hekmat B.; Caprioglio, Diego; Moriello, Claudia; Masi, Francesca; Hammami, Saoussen; Appendino, Giovanni; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio | |
Synthesis and biological evaluation of hydroxamate isosteres of acidic cannabinoids | 1-gen-2023 | Amin, Hawraz Ibrahim M.; Ruiz-Pino, Francisco; Collado, Juan A.; Appendino, Giovanni; Tena-Sempere, Manuel; Munoz, Eduardo; Caprioglio, Diego | |
Non-Volatile Terpenoids and Lipophilic Flavonoids from Achillea erba-rotta Subsp. moschata (Wulfen) I. Richardson | 1-gen-2023 | Salamone, Stefano; Aiello, Nicola; Fusani, Pietro; Rosa, Antonella; Nieddu, Mariella; Appendino, Giovanni; Pollastro, Federica | |
Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators | 1-gen-2023 | Peltner, Lukas K; Gluthmann, Lars; Börner, Friedemann; Pace, Simona; Hoffstetter, Robert K; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E; Gilbert, Nathaniel C; Werz, Oliver; Jordan, Paul M | |
Rotational constriction of curcuminoids impacts 5-lipoxygenase and mPGES-1 inhibition and evokes a lipid mediator class switch in macrophages | 1-gen-2022 | Rao, Zhigang; Caprioglio, Diego; Gollowitzer, Andre; Kretzer, Christian; Imperio, Daniela; Collado, Juan A.; Waltl, Lorenz; Lackner, Sandra; Appendino, Giovanni Battista; Munoz, Eduardo; Temml, Veronika; Werz, Oliver; Minassi, Alberto; Koeberle, Andreas | |
Minor Phytocannabinoids: A Misleading Name but a Promising Opportunity for Biomedical Research | 1-gen-2022 | Caprioglio, Diego; Amin, Hawraz Ibrahim M.; Taglialatela-Scafati, Orazio; Muñoz, Eduardo; Appendino, Giovanni | |
One‐Pot Oxidative Heterofunctionalization of Resorcinolic Cannabinoids to Non‐thiophilic Aminocannabinoquinones | 1-gen-2022 | Caprioglio, Diego; Mattoteia, Daiana; Muñoz, Eduardo; Taglialatela‐scafati, Orazio; Appendino, Giovanni | |
Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex | 1-gen-2022 | Funamoto, M.; Sunagawa, Y.; Gempei, M.; Shimizu, K.; Katanasaka, Y.; Shimizu, S.; Hamabe-Horiike, T.; Appendino, G.; Minassi, A.; Koeberle, A.; Komiyama, M.; Mori, K.; Hasegawa, K.; Morimoto, T. | |
Δ9-cis-Tetrahydrocannabinol: Natural Occurrence, Chirality, and Pharmacology | 1-gen-2021 | Schafroth, Michael A; Mazzoccanti, Giulia; Reynoso-Moreno, Ines; Erni, Reto; Pollastro, Federica; Caprioglio, Diego; Botta, Bruno; Allegrone, Gianna; Grassi, Giulio; Chicca, Andrea; Gasparrini, Francesco; Gertsch, Jürg; Carreira, Erick M; Appendino, Giovanni | |
Agathadiol, a labdane diterpenoid from juniper berries, is a positive allosteric modulator of CB1R | 1-gen-2021 | Salamone, Stefano; Appendino, Giovanni; Khalili, Adil; Pollastro, Federica; Munoz, Eduardo; Unciti-Broceta, Juan D | |
EHP-101 alleviates angiotensin II-induced fibrosis and inflammation in mice | 1-gen-2021 | Garcia-Martin, A.; Navarrete, C.; Garrido-Rodriguez, M.; Prados, M. E.; Caprioglio, D.; Appendino, G.; Munoz, E. | |
Betulinic acid hydroxamate prevents colonic inflammation and fibrosis in murine models of inflammatory bowel disease | 1-gen-2021 | Prados, M. E.; Garcia-Martin, A.; Unciti-Broceta, J. D.; Palomares, B.; Collado, J. A.; Minassi, A.; Calzado, M. A.; Appendino, G.; Munoz, E. | |
Betulinic Acid Hydroxamate is Neuroprotective and Induces Protein Phosphatase 2A-Dependent HIF-1α Stabilization and Post-transcriptional Dephosphorylation of Prolyl Hydrolase 2 | 1-gen-2021 | Prados, M. E.; Correa-Saez, A.; Unciti-Broceta, J. D.; Garrido-Rodriguez, M.; Jimenez-Jimenez, C.; Mazzone, M.; Minassi, A.; Appendino, G.; Calzado, M. A.; Munoz, E. | |
The combined effect of branching and elongation on the bioactivity profile of phytocannabinoids. Part i: Thermo-trps | 1-gen-2021 | Mattoteia, D.; Moriello, A. S.; Taglialatela-Scafati, O.; Amodeo, P.; De Petrocellis, L.; Appendino, G.; Vitale, R. M.; Caprioglio, D. | |
Cannabinoquinones: Synthesis and biological profile | 1-gen-2021 | Caprioglio, D.; Mattoteia, D.; Taglialatela-Scafati, O.; Munoz, E.; Appendino, G. | |
Icilio Guareschi and his amazing “1897 reaction” | 1-gen-2021 | Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G. | |
Best practice in research – Overcoming common challenges in phytopharmacological research | 1-gen-2020 | Heinrich, M.; Appendino, G.; Efferth, T.; Furst, R.; Izzo, A. A.; Kayser, O.; Pezzuto, J. M.; Viljoen, A. |
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