Sfoglia per Autore
Dietary Terpenoid Lactones are Promiscuous Agonists of Bitter Taste Receptors (TAS2Rs)
2026-01-01 Salamone, Stefano; Montelatici, Sara; Rinaldi, Maurizio; Appendino, Giovanni; Winnig, Marcel; Morini, Gabriella; Pollastro, Federica
Investigation in the CB1 and CB2 receptor binding profile and intrinsic activity of (−) and (+)-enantiomers of some naturally occurring phytocannabinoids or synthetic derivatives
2025-01-01 Rodriguez-Carreiro, S.; Gomez-Canas, M.; Lubrini, F.; Gonzalo-Consuegra, C.; Winkler, M.; Caprioglio, D.; Appendino, G.; Garcia, C.; Morales, P.; Jagerovic, N.; Fischer, J. T.; Fiebich, B. L.; Goetz, M. R.; Munoz, E.; Fernandez-Ruiz, J.
Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity
2025-01-01 Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L.; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo
Analytically Unsupervised Metabolomic Profile of the Premium Malgasy Pepper Voatsipérifery (Piper borbonense): Identification of Marker Components
2025-01-01 Serino, Elena; Pollastro, Federica; Luciano, Paolo; Touboul, David; Appendino, Giovanni; Chianese, Giuseppina; Taglialatela-Scafati, Orazio
The Impact of a Quinone Scaffold on Thermo-TRPs Modulation by Dimethylheptyl Phytocannabinoids
2025-01-01 Schiano Moriello, A.; Bossoni, A.; Mattoteia, D.; Caprioglio, D.; Minassi, A.; Appendino, G.; De Petrocellis, L.; Amodeo, P.; Vitale, R. M.
Cannabichromene (CBC) Shows Matrix-Dependent Thermal Configurational Stability
2024-01-01 Manetto, Simone; Caprioglio, Diego; Grassi, Gianpaolo; Botta, Bruno; Gasparrini, Francesco; Mazzoccanti, Giulia; Appendino, Giovanni
Comparative Evaluation of Anticancer Activity of Natural Methoxylated Flavones Xanthomicrol and Eupatilin in A375 Skin Melanoma Cells
2024-01-01 Rosa, Antonella; Piras, Franca; Pollastro, Federica; Sogos, Valeria; Appendino, Giovanni; Nieddu, Mariella
Arzanol, a natural phloroglucinol α‐pyrone, protects HaCaT keratinocytes against H2O2‐induced oxidative stress, counteracting cytotoxicity, reactive oxygen species generation, apoptosis, and mitochondrial depolarization
2024-01-01 Piras, Franca; Sogos, Valeria; Pollastro, Federica; Appendino, Giovanni; Rosa, Antonella
Eukaryotic Initiation Translation Factor 2A activation by cannabidiolic acid alters the protein homeostasis balance in glioblastoma cells
2024-01-01 Bellone, Maria Laura; Syed, Azmal Ali; Vitale, Rosa Maria; Sigismondo, Gianluca; Mensitieri, Francesca; Pollastro, Federica; Amodeo, Pietro; Appendino, Giovanni; De Tommasi, Nunziatina; Krijgsveld, Jeroen; Dal Piaz, Fabrizio
Synthesis and biological evaluation of hydroxamate isosteres of acidic cannabinoids
2023-01-01 Amin, Hawraz Ibrahim M.; Ruiz-Pino, Francisco; Collado, Juan A.; Appendino, Giovanni; Tena-Sempere, Manuel; Munoz, Eduardo; Caprioglio, Diego
Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators
2023-01-01 Peltner, Lukas K; Gluthmann, Lars; Börner, Friedemann; Pace, Simona; Hoffstetter, Robert K; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E; Gilbert, Nathaniel C; Werz, Oliver; Jordan, Paul M
Non-Volatile Terpenoids and Lipophilic Flavonoids from Achillea erba-rotta Subsp. moschata (Wulfen) I. Richardson
2023-01-01 Salamone, Stefano; Aiello, Nicola; Fusani, Pietro; Rosa, Antonella; Nieddu, Mariella; Appendino, Giovanni; Pollastro, Federica
PPARα/γ-Targeting Amorfrutin Phytocannabinoids from Aerial Parts of Glycyrrhiza foetida
2023-01-01 Serino, Elena; Iannotti, Fabio Arturo; Al-Hmadi, Hekmat B.; Caprioglio, Diego; Moriello, Claudia; Masi, Francesca; Hammami, Saoussen; Appendino, Giovanni; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio
Novel Skeletal Rearrangements of the Tigliane Diterpenoid Core
2023-01-01 Maioli, Chiara; Amin, Hawraz Ibrahim M.; Chianese, Giuseppina; Minassi, Alberto; Reddell, Paul W.; Gaeta, Simone; Taglialatela-Scafati, Orazio; Appendino, Giovanni
Rotational constriction of curcuminoids impacts 5-lipoxygenase and mPGES-1 inhibition and evokes a lipid mediator class switch in macrophages
2022-01-01 Rao, Zhigang; Caprioglio, Diego; Gollowitzer, Andre; Kretzer, Christian; Imperio, Daniela; Collado, Juan A.; Waltl, Lorenz; Lackner, Sandra; Appendino, Giovanni Battista; Munoz, Eduardo; Temml, Veronika; Werz, Oliver; Minassi, Alberto; Koeberle, Andreas
Cryptic Epoxytiglianes from the Kernels of the Blushwood Tree (Fontainea picrosperma)
2022-01-01 Chianese, Giuseppina; Amin, Hawraz Ibrahim M.; Maioli, Chiara; Reddell, Paul; Parsons, Peter; Cullen, Jason; Johns, Jenny; Handoko, Herlina; Boyle, Glen; Appendino, Giovanni; Taglialatela-Scafati, Orazio; Gaeta, Simone
Minor Phytocannabinoids: A Misleading Name but a Promising Opportunity for Biomedical Research
2022-01-01 Caprioglio, Diego; Amin, Hawraz Ibrahim M.; Taglialatela-Scafati, Orazio; Muñoz, Eduardo; Appendino, Giovanni
One‐Pot Oxidative Heterofunctionalization of Resorcinolic Cannabinoids to Non‐thiophilic Aminocannabinoquinones
2022-01-01 Caprioglio, Diego; Mattoteia, Daiana; Muñoz, Eduardo; Taglialatela‐scafati, Orazio; Appendino, Giovanni
Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex
2022-01-01 Funamoto, M.; Sunagawa, Y.; Gempei, M.; Shimizu, K.; Katanasaka, Y.; Shimizu, S.; Hamabe-Horiike, T.; Appendino, G.; Minassi, A.; Koeberle, A.; Komiyama, M.; Mori, K.; Hasegawa, K.; Morimoto, T.
Agathadiol, a labdane diterpenoid from juniper berries, is a positive allosteric modulator of CB1R
2021-01-01 Salamone, Stefano; Appendino, Giovanni; Khalili, Adil; Pollastro, Federica; Munoz, Eduardo; Unciti-Broceta, Juan D
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Dietary Terpenoid Lactones are Promiscuous Agonists of Bitter Taste Receptors (TAS2Rs) | 1-gen-2026 | Salamone, Stefano; Montelatici, Sara; Rinaldi, Maurizio; Appendino, Giovanni; Winnig, Marcel; Morini, Gabriella; Pollastro, Federica | |
| Investigation in the CB1 and CB2 receptor binding profile and intrinsic activity of (−) and (+)-enantiomers of some naturally occurring phytocannabinoids or synthetic derivatives | 1-gen-2025 | Rodriguez-Carreiro, S.; Gomez-Canas, M.; Lubrini, F.; Gonzalo-Consuegra, C.; Winkler, M.; Caprioglio, D.; Appendino, G.; Garcia, C.; Morales, P.; Jagerovic, N.; Fischer, J. T.; Fiebich, B. L.; Goetz, M. R.; Munoz, E.; Fernandez-Ruiz, J. | |
| Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity | 1-gen-2025 | Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L.; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo | |
| Analytically Unsupervised Metabolomic Profile of the Premium Malgasy Pepper Voatsipérifery (Piper borbonense): Identification of Marker Components | 1-gen-2025 | Serino, Elena; Pollastro, Federica; Luciano, Paolo; Touboul, David; Appendino, Giovanni; Chianese, Giuseppina; Taglialatela-Scafati, Orazio | |
| The Impact of a Quinone Scaffold on Thermo-TRPs Modulation by Dimethylheptyl Phytocannabinoids | 1-gen-2025 | Schiano Moriello, A.; Bossoni, A.; Mattoteia, D.; Caprioglio, D.; Minassi, A.; Appendino, G.; De Petrocellis, L.; Amodeo, P.; Vitale, R. M. | |
| Cannabichromene (CBC) Shows Matrix-Dependent Thermal Configurational Stability | 1-gen-2024 | Manetto, Simone; Caprioglio, Diego; Grassi, Gianpaolo; Botta, Bruno; Gasparrini, Francesco; Mazzoccanti, Giulia; Appendino, Giovanni | |
| Comparative Evaluation of Anticancer Activity of Natural Methoxylated Flavones Xanthomicrol and Eupatilin in A375 Skin Melanoma Cells | 1-gen-2024 | Rosa, Antonella; Piras, Franca; Pollastro, Federica; Sogos, Valeria; Appendino, Giovanni; Nieddu, Mariella | |
| Arzanol, a natural phloroglucinol α‐pyrone, protects HaCaT keratinocytes against H2O2‐induced oxidative stress, counteracting cytotoxicity, reactive oxygen species generation, apoptosis, and mitochondrial depolarization | 1-gen-2024 | Piras, Franca; Sogos, Valeria; Pollastro, Federica; Appendino, Giovanni; Rosa, Antonella | |
| Eukaryotic Initiation Translation Factor 2A activation by cannabidiolic acid alters the protein homeostasis balance in glioblastoma cells | 1-gen-2024 | Bellone, Maria Laura; Syed, Azmal Ali; Vitale, Rosa Maria; Sigismondo, Gianluca; Mensitieri, Francesca; Pollastro, Federica; Amodeo, Pietro; Appendino, Giovanni; De Tommasi, Nunziatina; Krijgsveld, Jeroen; Dal Piaz, Fabrizio | |
| Synthesis and biological evaluation of hydroxamate isosteres of acidic cannabinoids | 1-gen-2023 | Amin, Hawraz Ibrahim M.; Ruiz-Pino, Francisco; Collado, Juan A.; Appendino, Giovanni; Tena-Sempere, Manuel; Munoz, Eduardo; Caprioglio, Diego | |
| Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators | 1-gen-2023 | Peltner, Lukas K; Gluthmann, Lars; Börner, Friedemann; Pace, Simona; Hoffstetter, Robert K; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E; Gilbert, Nathaniel C; Werz, Oliver; Jordan, Paul M | |
| Non-Volatile Terpenoids and Lipophilic Flavonoids from Achillea erba-rotta Subsp. moschata (Wulfen) I. Richardson | 1-gen-2023 | Salamone, Stefano; Aiello, Nicola; Fusani, Pietro; Rosa, Antonella; Nieddu, Mariella; Appendino, Giovanni; Pollastro, Federica | |
| PPARα/γ-Targeting Amorfrutin Phytocannabinoids from Aerial Parts of Glycyrrhiza foetida | 1-gen-2023 | Serino, Elena; Iannotti, Fabio Arturo; Al-Hmadi, Hekmat B.; Caprioglio, Diego; Moriello, Claudia; Masi, Francesca; Hammami, Saoussen; Appendino, Giovanni; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio | |
| Novel Skeletal Rearrangements of the Tigliane Diterpenoid Core | 1-gen-2023 | Maioli, Chiara; Amin, Hawraz Ibrahim M.; Chianese, Giuseppina; Minassi, Alberto; Reddell, Paul W.; Gaeta, Simone; Taglialatela-Scafati, Orazio; Appendino, Giovanni | |
| Rotational constriction of curcuminoids impacts 5-lipoxygenase and mPGES-1 inhibition and evokes a lipid mediator class switch in macrophages | 1-gen-2022 | Rao, Zhigang; Caprioglio, Diego; Gollowitzer, Andre; Kretzer, Christian; Imperio, Daniela; Collado, Juan A.; Waltl, Lorenz; Lackner, Sandra; Appendino, Giovanni Battista; Munoz, Eduardo; Temml, Veronika; Werz, Oliver; Minassi, Alberto; Koeberle, Andreas | |
| Cryptic Epoxytiglianes from the Kernels of the Blushwood Tree (Fontainea picrosperma) | 1-gen-2022 | Chianese, Giuseppina; Amin, Hawraz Ibrahim M.; Maioli, Chiara; Reddell, Paul; Parsons, Peter; Cullen, Jason; Johns, Jenny; Handoko, Herlina; Boyle, Glen; Appendino, Giovanni; Taglialatela-Scafati, Orazio; Gaeta, Simone | |
| Minor Phytocannabinoids: A Misleading Name but a Promising Opportunity for Biomedical Research | 1-gen-2022 | Caprioglio, Diego; Amin, Hawraz Ibrahim M.; Taglialatela-Scafati, Orazio; Muñoz, Eduardo; Appendino, Giovanni | |
| One‐Pot Oxidative Heterofunctionalization of Resorcinolic Cannabinoids to Non‐thiophilic Aminocannabinoquinones | 1-gen-2022 | Caprioglio, Diego; Mattoteia, Daiana; Muñoz, Eduardo; Taglialatela‐scafati, Orazio; Appendino, Giovanni | |
| Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex | 1-gen-2022 | Funamoto, M.; Sunagawa, Y.; Gempei, M.; Shimizu, K.; Katanasaka, Y.; Shimizu, S.; Hamabe-Horiike, T.; Appendino, G.; Minassi, A.; Koeberle, A.; Komiyama, M.; Mori, K.; Hasegawa, K.; Morimoto, T. | |
| Agathadiol, a labdane diterpenoid from juniper berries, is a positive allosteric modulator of CB1R | 1-gen-2021 | Salamone, Stefano; Appendino, Giovanni; Khalili, Adil; Pollastro, Federica; Munoz, Eduardo; Unciti-Broceta, Juan D |
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