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Dietary Terpenoid Lactones are Promiscuous Agonists of Bitter Taste Receptors (TAS2Rs) 1-gen-2026 Salamone, Stefano; Montelatici, Sara; Rinaldi, Maurizio; Appendino, Giovanni; Winnig, Marcel; Morini, Gabriella; Pollastro, Federica
Investigation in the CB1 and CB2 receptor binding profile and intrinsic activity of (−) and (+)-enantiomers of some naturally occurring phytocannabinoids or synthetic derivatives 1-gen-2025 Rodriguez-Carreiro, S.; Gomez-Canas, M.; Lubrini, F.; Gonzalo-Consuegra, C.; Winkler, M.; Caprioglio, D.; Appendino, G.; Garcia, C.; Morales, P.; Jagerovic, N.; Fischer, J. T.; Fiebich, B. L.; Goetz, M. R.; Munoz, E.; Fernandez-Ruiz, J.
Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity 1-gen-2025 Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L.; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo
Analytically Unsupervised Metabolomic Profile of the Premium Malgasy Pepper Voatsipérifery (Piper borbonense): Identification of Marker Components 1-gen-2025 Serino, Elena; Pollastro, Federica; Luciano, Paolo; Touboul, David; Appendino, Giovanni; Chianese, Giuseppina; Taglialatela-Scafati, Orazio
The Impact of a Quinone Scaffold on Thermo-TRPs Modulation by Dimethylheptyl Phytocannabinoids 1-gen-2025 Schiano Moriello, A.; Bossoni, A.; Mattoteia, D.; Caprioglio, D.; Minassi, A.; Appendino, G.; De Petrocellis, L.; Amodeo, P.; Vitale, R. M.
Cannabichromene (CBC) Shows Matrix-Dependent Thermal Configurational Stability 1-gen-2024 Manetto, Simone; Caprioglio, Diego; Grassi, Gianpaolo; Botta, Bruno; Gasparrini, Francesco; Mazzoccanti, Giulia; Appendino, Giovanni
Comparative Evaluation of Anticancer Activity of Natural Methoxylated Flavones Xanthomicrol and Eupatilin in A375 Skin Melanoma Cells 1-gen-2024 Rosa, Antonella; Piras, Franca; Pollastro, Federica; Sogos, Valeria; Appendino, Giovanni; Nieddu, Mariella
Arzanol, a natural phloroglucinol α‐pyrone, protects HaCaT keratinocytes against H2O2‐induced oxidative stress, counteracting cytotoxicity, reactive oxygen species generation, apoptosis, and mitochondrial depolarization 1-gen-2024 Piras, Franca; Sogos, Valeria; Pollastro, Federica; Appendino, Giovanni; Rosa, Antonella
Eukaryotic Initiation Translation Factor 2A activation by cannabidiolic acid alters the protein homeostasis balance in glioblastoma cells 1-gen-2024 Bellone, Maria Laura; Syed, Azmal Ali; Vitale, Rosa Maria; Sigismondo, Gianluca; Mensitieri, Francesca; Pollastro, Federica; Amodeo, Pietro; Appendino, Giovanni; De Tommasi, Nunziatina; Krijgsveld, Jeroen; Dal Piaz, Fabrizio
Synthesis and biological evaluation of hydroxamate isosteres of acidic cannabinoids 1-gen-2023 Amin, Hawraz Ibrahim M.; Ruiz-Pino, Francisco; Collado, Juan A.; Appendino, Giovanni; Tena-Sempere, Manuel; Munoz, Eduardo; Caprioglio, Diego
Cannabidiol acts as molecular switch in innate immune cells to promote the biosynthesis of inflammation-resolving lipid mediators 1-gen-2023 Peltner, Lukas K; Gluthmann, Lars; Börner, Friedemann; Pace, Simona; Hoffstetter, Robert K; Kretzer, Christian; Bilancia, Rosella; Pollastro, Federica; Koeberle, Andreas; Appendino, Giovanni; Rossi, Antonietta; Newcomer, Marcia E; Gilbert, Nathaniel C; Werz, Oliver; Jordan, Paul M
Non-Volatile Terpenoids and Lipophilic Flavonoids from Achillea erba-rotta Subsp. moschata (Wulfen) I. Richardson 1-gen-2023 Salamone, Stefano; Aiello, Nicola; Fusani, Pietro; Rosa, Antonella; Nieddu, Mariella; Appendino, Giovanni; Pollastro, Federica
PPARα/γ-Targeting Amorfrutin Phytocannabinoids from Aerial Parts of Glycyrrhiza foetida 1-gen-2023 Serino, Elena; Iannotti, Fabio Arturo; Al-Hmadi, Hekmat B.; Caprioglio, Diego; Moriello, Claudia; Masi, Francesca; Hammami, Saoussen; Appendino, Giovanni; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio
Novel Skeletal Rearrangements of the Tigliane Diterpenoid Core 1-gen-2023 Maioli, Chiara; Amin, Hawraz Ibrahim M.; Chianese, Giuseppina; Minassi, Alberto; Reddell, Paul W.; Gaeta, Simone; Taglialatela-Scafati, Orazio; Appendino, Giovanni
Rotational constriction of curcuminoids impacts 5-lipoxygenase and mPGES-1 inhibition and evokes a lipid mediator class switch in macrophages 1-gen-2022 Rao, Zhigang; Caprioglio, Diego; Gollowitzer, Andre; Kretzer, Christian; Imperio, Daniela; Collado, Juan A.; Waltl, Lorenz; Lackner, Sandra; Appendino, Giovanni Battista; Munoz, Eduardo; Temml, Veronika; Werz, Oliver; Minassi, Alberto; Koeberle, Andreas
Cryptic Epoxytiglianes from the Kernels of the Blushwood Tree (Fontainea picrosperma) 1-gen-2022 Chianese, Giuseppina; Amin, Hawraz Ibrahim M.; Maioli, Chiara; Reddell, Paul; Parsons, Peter; Cullen, Jason; Johns, Jenny; Handoko, Herlina; Boyle, Glen; Appendino, Giovanni; Taglialatela-Scafati, Orazio; Gaeta, Simone
Minor Phytocannabinoids: A Misleading Name but a Promising Opportunity for Biomedical Research 1-gen-2022 Caprioglio, Diego; Amin, Hawraz Ibrahim M.; Taglialatela-Scafati, Orazio; Muñoz, Eduardo; Appendino, Giovanni
One‐Pot Oxidative Heterofunctionalization of Resorcinolic Cannabinoids to Non‐thiophilic Aminocannabinoquinones 1-gen-2022 Caprioglio, Diego; Mattoteia, Daiana; Muñoz, Eduardo; Taglialatela‐scafati, Orazio; Appendino, Giovanni
Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex 1-gen-2022 Funamoto, M.; Sunagawa, Y.; Gempei, M.; Shimizu, K.; Katanasaka, Y.; Shimizu, S.; Hamabe-Horiike, T.; Appendino, G.; Minassi, A.; Koeberle, A.; Komiyama, M.; Mori, K.; Hasegawa, K.; Morimoto, T.
Agathadiol, a labdane diterpenoid from juniper berries, is a positive allosteric modulator of CB1R 1-gen-2021 Salamone, Stefano; Appendino, Giovanni; Khalili, Adil; Pollastro, Federica; Munoz, Eduardo; Unciti-Broceta, Juan D
Mostrati risultati da 1 a 20 di 339
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