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Mostrati risultati da 1 a 20 di 89
Titolo Data di pubblicazione Autore(i) File
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT2 1-gen-2024 Kaya, Selen Gozde; Eren, Gokcen; Massarotti, Alberto; Gunindi, Habibe Beyza; Bakar‐ates, Filiz; Ozkan, Erva
A nonnatural peptide targeting the A-kinase anchoring function of PI3Kγ for therapeutic cAMP modulation in pulmonary cells 1-gen-2024 Della Sala, Angela; Tasca, Laura; Butnarasu, Cosmin; Sala, Valentina; Prono, Giulia; Murabito, Alessandra; Garbero, Olga Valentina; Millo, Enrico; Terranova, Leonardo; Blasi, Francesco; Gramegna, Andrea; Aliberti, Stefano; Massarotti, Alberto; Visentin, Sonja; Hirsch, Emilio; Ghigo, Alessandra
Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1 1-gen-2024 Panfili, Eleonora; Rezzi, Sarah Jane; Adamo, Annalisa; Mazzoletti, Daniele; Massarotti, Alberto; Miggiano, Riccardo; Fallarini, Silvia; Ambrosino, Sara; Coletti, Alice; Molinaro, Pasquale; Milella, Michele; Paiella, Salvatore; Macchiarulo, Antonio; Ugel, Stefano; Pirali, Tracey; Pallotta, Maria Teresa
2‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition 1-gen-2024 Kaya, Selen Gozde; Eren, Gokcen; Massarotti, Alberto; Bakar‐ates, Filiz; Ozkan, Erva; Gozelle, Mahmut; Ozkan, Yesim
In silico approach reveals N-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits 1-gen-2023 Gozelle, Mahmut; Bakar-Ates, Filiz; Massarotti, Alberto; Ozkan, Erva; Gunindi, Habibe Beyza; Ozkan, Yesim; Eren, Gokcen
Therapeutic peptides for the treatment of cystic fibrosis: Challenges and perspectives 1-gen-2021 Sala, V.; Cnudde, S. J.; Murabito, A.; Massarotti, A.; Hirsch, E.; Ghigo, A.
PI(3,4)P2-mediated cytokinetic abscission prevents early senescence and cataract formation 1-gen-2021 Gulluni, Federico; Prever, Lorenzo; Li, Huayi; Krafcikova, Petra; Corrado, Ilaria; Lo, Wen-Ting; Margaria, Jean Piero; Chen, Anlu; De Santis, Maria Chiara; Cnudde, Sophie J.; Fogerty, Joseph; Yuan, Alex; Massarotti, Alberto; Sarijalo, Nasrin Torabi; Vadas, Oscar; Williams, Roger L.; Thelen, Marcus; Powell, David R.; Schueler, Markus; Wiesener, Michael S.; Balla, Tamas; Baris, Hagit N.; Tiosano, Dov; Mcdermott, Brian M.; Perkins, Brian D.; Ghigo, Alessandra; Martini, Miriam; Haucke, Volker; Boura, Evzen; Merlo, Giorgio Roberto; Buchner, David A.; Hirsch, Emilio
Medicinal Chemistry of Isocyanides 1-gen-2021 Massarotti, A.; Brunelli, F.; Aprile, S.; Giustiniano, M.; Tron, G. C.
What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications 1-gen-2021 Serafini, M.; Cargnin, S.; Massarotti, A.; Tron, G. C.; Pirali, T.; Genazzani, A.
The [1,2,4]Triazolo[4,3-a]pyridine as a New Player in the Field of IDO1 Catalytic Holo-Inhibitors 1-gen-2021 Fallarini, S.; Bhela, I. P.; Aprile, S.; Torre, E.; Ranza, A.; Orecchini, E.; Panfili, E.; Pallotta, M. T.; Massarotti, A.; Serafini, M.; Pirali, T.
The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate 1-gen-2021 Merlo, R.; Caprioglio, D.; Cillo, M.; Valenti, A.; Mattossovich, R.; Morrone, C.; Massarotti, A.; Rossi, F.; Miggiano, R.; Leonardi, A.; Minassi, A.; Perugino, G.
Investigation of the Click-Chemical Space for Drug Design Using ZINClick 1-gen-2021 Massarotti, A.
Photocatalytic Isocyanide-based Multicomponent Domino Cascade Towards the Stereoselective Formation of Iminofurans 1-gen-2020 Pelliccia, Sveva; Alfano, Antonella Ilenia; Luciano, Paolo; Novellino, Ettore; Massarotti, Alberto; Tron, Gian Cesare; Ravelli, Davide; Giustiniano, Mariateresa
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity 1-gen-2020 Serafini, M.; Torre, E.; Aprile, S.; Del Grosso, E.; Gesu, A.; Griglio, A.; Colombo, G.; Travelli, C.; Paiella, S.; Adamo, A.; Orecchini, E.; Coletti, A.; Pallotta, M. T.; Ugel, S.; Massarotti, A.; Pirali, T.; Fallarini, S.
Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors 1-gen-2020 Velnati, Suresh; Massarotti, Alberto; Antona, Annamaria; Talmon, Maria; Fresu, Luigia Grazia; Galetto, Alessandra Silvia; Capello, Daniela; Bertoni, Alessandra; Mercalli, Valentina; Graziani, Andrea; Tron, Gian Cesare; Baldanzi, Gianluca
Psychotropic Drugs Show Anticancer Activity by Disrupting Mitochondrial and Lysosomal Function 1-gen-2020 Varalda, Marco; Antona, Annamaria; Bettio, Valentina; Roy, Konkonika; Vachamaram, Ajay; Yellenki, Vaibhav; Massarotti, Alberto; Baldanzi, Gianluca; Capello, Daniela
Bio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine Derivatives 1-gen-2020 Pelliccia, Sveva; Amato, Jussara; Capasso, Domenica; Di Gaetano, Sonia; Massarotti, Alberto; Piccolo, Marialuisa; Irace, Carlo; Tron, Gian Cesare; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Giustiniano, Mariateresa
The Essential Medicinal Chemistry of Essential Medicines 1-gen-2020 Serafini, Marta; Cargnin, Sarah; Massarotti, Alberto; Pirali, Tracey; Genazzani, Armando
Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors 1-gen-2019 Serafini, Marta; Torre, Enza; Aprile, Silvio; Massarotti, Alberto; Fallarini, Silvia; Pirali, Tracey
ZINClick v.18: Expanding Chemical Space of 1,2,3-Triazoles 1-gen-2019 Levré, Doriana; Arcisto, Chiara; Mercalli, Valentina; Massarotti, Alberto
Mostrati risultati da 1 a 20 di 89
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