Sfoglia per Autore
Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor
2023-01-01 Alberti, Marta; Sainas, Stefano; Ronchi, Erika; Lolli, Marco L; Boschi, Donatella; Rizzi, Menico; Ferraris, Davide M; Miggiano, Riccardo
The integration of AlphaFold-predicted and crystal structures of human trans-3-hydroxy-l-proline dehydratase reveals a regulatory catalytic mechanism
2022-01-01 Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M
Curcumin-based-fluorescent probes targeting ALDH1A3 as a promising tool for glioblastoma precision surgery and early diagnosis
2022-01-01 Gelardi, Edoardo L. M.; Caprioglio, Diego; Colombo, Giorgia; Del Grosso, Erika; Mazzoletti, Daniele; Mattoteia, Daiana; Salamone, Stefano; Ferraris, Davide M.; Aronica, Eleonora; Nato, Giulia; Buffo, Annalisa; Rizzi, Menico; Magrassi, Lorenzo; Minassi, Alberto; Garavaglia, Silvia
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety
2022-01-01 Sainas, Stefano; Giorgis, Marta; Circosta, Paola; Poli, Giulio; Alberti, Marta; Passoni, Alice; Gaidano, Valentina; Pippione, Agnese C; Vitale, Nicoletta; Bonanni, Davide; Rolando, Barbara; Cignetti, Alessandro; Ramondetti, Cristina; Lanno, Alessia; Ferraris, Davide M; Canepa, Barbara; Buccinnà, Barbara; Piccinini, Marco; Rizzi, Menico; Saglio, Giuseppe; Al-Karadaghi, Salam; Boschi, Donatella; Miggiano, Riccardo; Tuccinardi, Tiziano; Lolli, Marco L
Engineering, Characterization, and Biological Evaluation of an Antibody Targeting the HGF Receptor
2021-01-01 Desole, C.; Gallo, S.; Vitacolonna, A.; Vigna, E.; Basilico, C.; Montarolo, F.; Zuppini, F.; Casanova, E.; Miggiano, R.; Ferraris, D. M.; Bertolotto, A.; Comoglio, P. M.; Crepaldi, T.
A selective competitive inhibitor of aldehyde dehydrogenase 1A3 hinders cancer cell growth, invasiveness and stemness in vitro
2021-01-01 Gelardi, E. L. M.; Colombo, G.; Picarazzi, F.; Ferraris, D. M.; Mangione, A.; Petrarolo, G.; Aronica, E.; Rizzi, M.; Mori, M.; La Motta, C.; Garavaglia, S.
Structure of Thermococcus litoralis Δ1-pyrroline-2-carboxylate reductase in complex with NADH and L-proline
2020-01-01 Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M
Targeting NAD-dependent dehydrogenases in drug discovery against infectious diseases and cancer
2020-01-01 Ferraris, Davide M; Gelardi, Edoardo L M; Garavaglia, Silvia; Miggiano, Riccardo; Rizzi, Menico
Imidazo[1,2-a]pyridine Derivatives as Aldehyde Dehydrogenase Inhibitors: Novel Chemotypes to Target Glioblastoma Stem Cells
2020-01-01 Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Coviello, Vito; Sartini, Stefania; Ferraris, Davide Maria; Mori, Mattia; Nakano, Ichiro; Garavaglia, Silvia; La Motta, Concettina
Extracellular NAD+ enhances PARP-dependent DNA repair capacity independently of CD73 activity
2020-01-01 Wilk, A.; Hayat, F.; Cunningham, R.; Li, J.; Garavaglia, S.; Zamani, L.; Ferraris, D. M.; Sykora, P.; Andrews, J.; Clark, J.; Davis, A.; Chaloin, L.; Rizzi, M.; Migaud, M.; Sobol, R. W.
Mycobacterium tuberculosis Pathogenesis, Infection Prevention and Treatment
2020-01-01 Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M.
A highly selective electrochemical assay based on the Sakaguchi reaction for the detection of protein arginine methylation state
2020-01-01 Mengyuan, He; Jiarong, Guo; Jiahua, Yang; Yang, Xue; Songyan, Zhao; Qiao, Xu; Tiangxiang, Wei; Ferraris, DAVIDE MARIA; Tao, Gao; Zhigang, Guo
Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2-a]pyridines against the 1A Family
2020-01-01 Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Petrarolo, Giovanni; Colombo, Giorgia; Ferraris, Davide Maria; Picarazzi, Francesca; Rizzi, Menico; Garavaglia, Silvia; La Motta, Concettina
Structure of Thermococcus litoralis trans-3-hydroxy-L-proline dehydratase in the free and substrate-complexed form
2019-01-01 Ferraris, D. M.; Miggiano, R.; Watanabe, S.; Rizzi, M.
The synthesis of kynurenic acid in mammals: an updated kynurenine aminotransferase structural KATalogue
2019-01-01 Rossi, Franca; Miggiano, Riccardo; Ferraris, Davide M.; Rizzi, Menico
Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH
2019-01-01 Singh, Vinayak; Pacitto, Angela; Donini, Stefano; Ferraris, Davide M.; Boros, Sándor; Illyés, Eszter; Szokol, Bálint; Rizzi, Menico; Blundell, Tom L.; Ascher, David B.; Pato, Janos; Mizrahi, Valerie
Mycobacterium tuberculosis Molecular Determinants of Infection, Survival Strategies, and Vulnerable Targets
2018-01-01 Ferraris, Davide M; Miggiano, Riccardo; Rossi, Franca; Rizzi, Menico
Hit discovery of Mycobacterium tuberculosis inosine 5′-monophosphate dehydrogenase, GuaB2, inhibitors
2018-01-01 Sahu, Niteshkumar U.; Singh, Vinayak; Ferraris, Davide M.; Rizzi, Menico; Kharkar, Prashant S.
Development of potent inhibitors of the Mycobacterium tuberculosis virulence factor Zmp1 and evaluation of their effect on mycobacterial survival inside macrophages.
2018-01-01 Paolino, M.; Brindisi, M.; Vallone, A.; Butini, S.; Campiani, G.; Nannicini, C.; Giuliani, G.; Anzini, M.; Lamponi, S.; Giorgi, G.; Sbardella, D.; Ferraris, D.; Marini, S.; Coletta, M.; Palucci, I.; Minerva, M.; Delogu, G.; Pepponi, I.; Goletti, D.; Cappelli, A.; Gemma, S.; Brogi, ; S. (2018). Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages., Chemmedchem; 13(5), ; 422–430. https://doi. org/10. 1002/cmdc., 201700759
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe
2018-01-01 Rossi, Franca; Morrone, Castrese; Massarotti, Alberto; Ferraris, Davide Maria; Valenti, Anna; Perugino, Giuseppe; Miggiano, Riccardo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor | 1-gen-2023 | Alberti, Marta; Sainas, Stefano; Ronchi, Erika; Lolli, Marco L; Boschi, Donatella; Rizzi, Menico; Ferraris, Davide M; Miggiano, Riccardo | |
The integration of AlphaFold-predicted and crystal structures of human trans-3-hydroxy-l-proline dehydratase reveals a regulatory catalytic mechanism | 1-gen-2022 | Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M | |
Curcumin-based-fluorescent probes targeting ALDH1A3 as a promising tool for glioblastoma precision surgery and early diagnosis | 1-gen-2022 | Gelardi, Edoardo L. M.; Caprioglio, Diego; Colombo, Giorgia; Del Grosso, Erika; Mazzoletti, Daniele; Mattoteia, Daiana; Salamone, Stefano; Ferraris, Davide M.; Aronica, Eleonora; Nato, Giulia; Buffo, Annalisa; Rizzi, Menico; Magrassi, Lorenzo; Minassi, Alberto; Garavaglia, Silvia | |
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety | 1-gen-2022 | Sainas, Stefano; Giorgis, Marta; Circosta, Paola; Poli, Giulio; Alberti, Marta; Passoni, Alice; Gaidano, Valentina; Pippione, Agnese C; Vitale, Nicoletta; Bonanni, Davide; Rolando, Barbara; Cignetti, Alessandro; Ramondetti, Cristina; Lanno, Alessia; Ferraris, Davide M; Canepa, Barbara; Buccinnà, Barbara; Piccinini, Marco; Rizzi, Menico; Saglio, Giuseppe; Al-Karadaghi, Salam; Boschi, Donatella; Miggiano, Riccardo; Tuccinardi, Tiziano; Lolli, Marco L | |
Engineering, Characterization, and Biological Evaluation of an Antibody Targeting the HGF Receptor | 1-gen-2021 | Desole, C.; Gallo, S.; Vitacolonna, A.; Vigna, E.; Basilico, C.; Montarolo, F.; Zuppini, F.; Casanova, E.; Miggiano, R.; Ferraris, D. M.; Bertolotto, A.; Comoglio, P. M.; Crepaldi, T. | |
A selective competitive inhibitor of aldehyde dehydrogenase 1A3 hinders cancer cell growth, invasiveness and stemness in vitro | 1-gen-2021 | Gelardi, E. L. M.; Colombo, G.; Picarazzi, F.; Ferraris, D. M.; Mangione, A.; Petrarolo, G.; Aronica, E.; Rizzi, M.; Mori, M.; La Motta, C.; Garavaglia, S. | |
Structure of Thermococcus litoralis Δ1-pyrroline-2-carboxylate reductase in complex with NADH and L-proline | 1-gen-2020 | Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M | |
Targeting NAD-dependent dehydrogenases in drug discovery against infectious diseases and cancer | 1-gen-2020 | Ferraris, Davide M; Gelardi, Edoardo L M; Garavaglia, Silvia; Miggiano, Riccardo; Rizzi, Menico | |
Imidazo[1,2-a]pyridine Derivatives as Aldehyde Dehydrogenase Inhibitors: Novel Chemotypes to Target Glioblastoma Stem Cells | 1-gen-2020 | Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Coviello, Vito; Sartini, Stefania; Ferraris, Davide Maria; Mori, Mattia; Nakano, Ichiro; Garavaglia, Silvia; La Motta, Concettina | |
Extracellular NAD+ enhances PARP-dependent DNA repair capacity independently of CD73 activity | 1-gen-2020 | Wilk, A.; Hayat, F.; Cunningham, R.; Li, J.; Garavaglia, S.; Zamani, L.; Ferraris, D. M.; Sykora, P.; Andrews, J.; Clark, J.; Davis, A.; Chaloin, L.; Rizzi, M.; Migaud, M.; Sobol, R. W. | |
Mycobacterium tuberculosis Pathogenesis, Infection Prevention and Treatment | 1-gen-2020 | Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M. | |
A highly selective electrochemical assay based on the Sakaguchi reaction for the detection of protein arginine methylation state | 1-gen-2020 | Mengyuan, He; Jiarong, Guo; Jiahua, Yang; Yang, Xue; Songyan, Zhao; Qiao, Xu; Tiangxiang, Wei; Ferraris, DAVIDE MARIA; Tao, Gao; Zhigang, Guo | |
Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2-a]pyridines against the 1A Family | 1-gen-2020 | Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Petrarolo, Giovanni; Colombo, Giorgia; Ferraris, Davide Maria; Picarazzi, Francesca; Rizzi, Menico; Garavaglia, Silvia; La Motta, Concettina | |
Structure of Thermococcus litoralis trans-3-hydroxy-L-proline dehydratase in the free and substrate-complexed form | 1-gen-2019 | Ferraris, D. M.; Miggiano, R.; Watanabe, S.; Rizzi, M. | |
The synthesis of kynurenic acid in mammals: an updated kynurenine aminotransferase structural KATalogue | 1-gen-2019 | Rossi, Franca; Miggiano, Riccardo; Ferraris, Davide M.; Rizzi, Menico | |
Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH | 1-gen-2019 | Singh, Vinayak; Pacitto, Angela; Donini, Stefano; Ferraris, Davide M.; Boros, Sándor; Illyés, Eszter; Szokol, Bálint; Rizzi, Menico; Blundell, Tom L.; Ascher, David B.; Pato, Janos; Mizrahi, Valerie | |
Mycobacterium tuberculosis Molecular Determinants of Infection, Survival Strategies, and Vulnerable Targets | 1-gen-2018 | Ferraris, Davide M; Miggiano, Riccardo; Rossi, Franca; Rizzi, Menico | |
Hit discovery of Mycobacterium tuberculosis inosine 5′-monophosphate dehydrogenase, GuaB2, inhibitors | 1-gen-2018 | Sahu, Niteshkumar U.; Singh, Vinayak; Ferraris, Davide M.; Rizzi, Menico; Kharkar, Prashant S. | |
Development of potent inhibitors of the Mycobacterium tuberculosis virulence factor Zmp1 and evaluation of their effect on mycobacterial survival inside macrophages. | 1-gen-2018 | Paolino, M.; Brindisi, M.; Vallone, A.; Butini, S.; Campiani, G.; Nannicini, C.; Giuliani, G.; Anzini, M.; Lamponi, S.; Giorgi, G.; Sbardella, D.; Ferraris, D.; Marini, S.; Coletta, M.; Palucci, I.; Minerva, M.; Delogu, G.; Pepponi, I.; Goletti, D.; Cappelli, A.; Gemma, S.; Brogi, ; S. (2018). Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages., Chemmedchem; 13(5), ; 422–430. https://doi. org/10. 1002/cmdc., 201700759 | |
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe | 1-gen-2018 | Rossi, Franca; Morrone, Castrese; Massarotti, Alberto; Ferraris, Davide Maria; Valenti, Anna; Perugino, Giuseppe; Miggiano, Riccardo |
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