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Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor 1-gen-2023 Alberti, Marta; Sainas, Stefano; Ronchi, Erika; Lolli, Marco L; Boschi, Donatella; Rizzi, Menico; Ferraris, Davide M; Miggiano, Riccardo
The integration of AlphaFold-predicted and crystal structures of human trans-3-hydroxy-l-proline dehydratase reveals a regulatory catalytic mechanism 1-gen-2022 Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M
Curcumin-based-fluorescent probes targeting ALDH1A3 as a promising tool for glioblastoma precision surgery and early diagnosis 1-gen-2022 Gelardi, Edoardo L. M.; Caprioglio, Diego; Colombo, Giorgia; Del Grosso, Erika; Mazzoletti, Daniele; Mattoteia, Daiana; Salamone, Stefano; Ferraris, Davide M.; Aronica, Eleonora; Nato, Giulia; Buffo, Annalisa; Rizzi, Menico; Magrassi, Lorenzo; Minassi, Alberto; Garavaglia, Silvia
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety 1-gen-2022 Sainas, Stefano; Giorgis, Marta; Circosta, Paola; Poli, Giulio; Alberti, Marta; Passoni, Alice; Gaidano, Valentina; Pippione, Agnese C; Vitale, Nicoletta; Bonanni, Davide; Rolando, Barbara; Cignetti, Alessandro; Ramondetti, Cristina; Lanno, Alessia; Ferraris, Davide M; Canepa, Barbara; Buccinnà, Barbara; Piccinini, Marco; Rizzi, Menico; Saglio, Giuseppe; Al-Karadaghi, Salam; Boschi, Donatella; Miggiano, Riccardo; Tuccinardi, Tiziano; Lolli, Marco L
Engineering, Characterization, and Biological Evaluation of an Antibody Targeting the HGF Receptor 1-gen-2021 Desole, C.; Gallo, S.; Vitacolonna, A.; Vigna, E.; Basilico, C.; Montarolo, F.; Zuppini, F.; Casanova, E.; Miggiano, R.; Ferraris, D. M.; Bertolotto, A.; Comoglio, P. M.; Crepaldi, T.
A selective competitive inhibitor of aldehyde dehydrogenase 1A3 hinders cancer cell growth, invasiveness and stemness in vitro 1-gen-2021 Gelardi, E. L. M.; Colombo, G.; Picarazzi, F.; Ferraris, D. M.; Mangione, A.; Petrarolo, G.; Aronica, E.; Rizzi, M.; Mori, M.; La Motta, C.; Garavaglia, S.
Structure of Thermococcus litoralis Δ1-pyrroline-2-carboxylate reductase in complex with NADH and L-proline 1-gen-2020 Ferrario, Eugenio; Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M
Targeting NAD-dependent dehydrogenases in drug discovery against infectious diseases and cancer 1-gen-2020 Ferraris, Davide M; Gelardi, Edoardo L M; Garavaglia, Silvia; Miggiano, Riccardo; Rizzi, Menico
Imidazo[1,2-a]pyridine Derivatives as Aldehyde Dehydrogenase Inhibitors: Novel Chemotypes to Target Glioblastoma Stem Cells 1-gen-2020 Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Coviello, Vito; Sartini, Stefania; Ferraris, Davide Maria; Mori, Mattia; Nakano, Ichiro; Garavaglia, Silvia; La Motta, Concettina
Extracellular NAD+ enhances PARP-dependent DNA repair capacity independently of CD73 activity 1-gen-2020 Wilk, A.; Hayat, F.; Cunningham, R.; Li, J.; Garavaglia, S.; Zamani, L.; Ferraris, D. M.; Sykora, P.; Andrews, J.; Clark, J.; Davis, A.; Chaloin, L.; Rizzi, M.; Migaud, M.; Sobol, R. W.
Mycobacterium tuberculosis Pathogenesis, Infection Prevention and Treatment 1-gen-2020 Miggiano, Riccardo; Rizzi, Menico; Ferraris, Davide M.
A highly selective electrochemical assay based on the Sakaguchi reaction for the detection of protein arginine methylation state 1-gen-2020 Mengyuan, He; Jiarong, Guo; Jiahua, Yang; Yang, Xue; Songyan, Zhao; Qiao, Xu; Tiangxiang, Wei; Ferraris, DAVIDE MARIA; Tao, Gao; Zhigang, Guo
Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2-a]pyridines against the 1A Family 1-gen-2020 Quattrini, Luca; Gelardi, Edoardo Luigi Maria; Petrarolo, Giovanni; Colombo, Giorgia; Ferraris, Davide Maria; Picarazzi, Francesca; Rizzi, Menico; Garavaglia, Silvia; La Motta, Concettina
Structure of Thermococcus litoralis trans-3-hydroxy-L-proline dehydratase in the free and substrate-complexed form 1-gen-2019 Ferraris, D. M.; Miggiano, R.; Watanabe, S.; Rizzi, M.
The synthesis of kynurenic acid in mammals: an updated kynurenine aminotransferase structural KATalogue 1-gen-2019 Rossi, Franca; Miggiano, Riccardo; Ferraris, Davide M.; Rizzi, Menico
Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH 1-gen-2019 Singh, Vinayak; Pacitto, Angela; Donini, Stefano; Ferraris, Davide M.; Boros, Sándor; Illyés, Eszter; Szokol, Bálint; Rizzi, Menico; Blundell, Tom L.; Ascher, David B.; Pato, Janos; Mizrahi, Valerie
Mycobacterium tuberculosis Molecular Determinants of Infection, Survival Strategies, and Vulnerable Targets 1-gen-2018 Ferraris, Davide M; Miggiano, Riccardo; Rossi, Franca; Rizzi, Menico
Hit discovery of Mycobacterium tuberculosis inosine 5′-monophosphate dehydrogenase, GuaB2, inhibitors 1-gen-2018 Sahu, Niteshkumar U.; Singh, Vinayak; Ferraris, Davide M.; Rizzi, Menico; Kharkar, Prashant S.
Development of potent inhibitors of the Mycobacterium tuberculosis virulence factor Zmp1 and evaluation of their effect on mycobacterial survival inside macrophages. 1-gen-2018 Paolino, M.; Brindisi, M.; Vallone, A.; Butini, S.; Campiani, G.; Nannicini, C.; Giuliani, G.; Anzini, M.; Lamponi, S.; Giorgi, G.; Sbardella, D.; Ferraris, D.; Marini, S.; Coletta, M.; Palucci, I.; Minerva, M.; Delogu, G.; Pepponi, I.; Goletti, D.; Cappelli, A.; Gemma, S.; Brogi, ; S. (2018). Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages., Chemmedchem; 13(5), ; 422–430. https://doi. org/10. 1002/cmdc., 201700759
Crystal structure of a thermophilic O6-alkylguanine-DNA alkyltransferase-derived self-labeling protein-tag in covalent complex with a fluorescent probe 1-gen-2018 Rossi, Franca; Morrone, Castrese; Massarotti, Alberto; Ferraris, Davide Maria; Valenti, Anna; Perugino, Giuseppe; Miggiano, Riccardo
Mostrati risultati da 1 a 20 di 34
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