Sfoglia per Autore
Icilio Guareschi and his amazing “1897 reaction”
2021-01-01 Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G.
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders
2018-01-01 Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
2018-01-01 Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis
2018-01-01 Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, Celia; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; Biocotino, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs
2017-01-01 Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity
2017-01-01 Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors
2016-01-01 Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents
2015-01-01 Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors
2015-01-01 Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?
2014-01-01 Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles
2014-01-01 Massarotti, Alberto; A., Brunco; Sorba, Giovanni; Tron, Gian Cesare
Inhibitors of Nicotinamide Phosphoribosyltransferase, compositions, products and uses thereof.
2014-01-01 Genazzani Armando, A.; Tron, Gian Cesare; Galli, Ubaldina; Travelli, Cristina; Cuzzocrea, Salvatore; Grosa, Giorgio; Sorba, Giovanni; Canonico Pier, Luigi
Capitolo 23. Istamina e agenti antistaminici
2014-01-01 Sorba, Giovanni; Massarotti, Alberto
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus
2013-01-01 Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A.
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents
2013-01-01 Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey
“Synthesis and in vitro evaluation of tetrasubstituted pyridines as potential PI3Ks inhibitors”
2013-01-01 Galli, Ubaldina; E., Ciraolo; E., Hirsch; Sorba, Giovanni; Tron, Gian Cesare
The tubulin colchicine domain: a molecular modelling perspective
2012-01-01 Massarotti, A; Coluccia, A; Silvestri, R; Sorba, G; Brancale, A
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2
2012-01-01 Galli, Ubaldina; Mesenzani, Ornella; Coppo, C; Sorba, Giovanni; Canonico, Pier Luigi; Tron, Gian Cesare; Genazzani, Armando
De novo computer-aided design of novel antiviral agents
2012-01-01 Massarotti, Alberto; Coluccia, A; Sorba, Giovanni; Silvestri, R; Brancale, A.
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases
2012-01-01 Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Icilio Guareschi and his amazing “1897 reaction” | 1-gen-2021 | Tron, G. C.; Minassi, A.; Sorba, G.; Fausone, M.; Appendino, G. | |
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders | 1-gen-2018 | Serafini, Marta; Griglio, Alessia; Aprile, Silvio; Seiti, Fabio; Travelli, Cristina; Pattarino, Franco; Grosa, Giorgio; Sorba, Giovanni; Genazzani, Armando; Gonzalez-Rodriguez, Sara; Butron, Laura; Devesa, Isabel; Fernandez-Carvajal, Asia; Pirali, Tracey; Ferrer-Montiel, Antonio | |
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies | 1-gen-2018 | Griglio, Alessia; Torre, Enza; Serafini, Marta; Bianchi, Alice; Schmid, Roberta; CODA ZABETTA, Giulia; Massarotti, Alberto; Sorba, Giovanni; Pirali, Tracey; Fallarini, Silvia | |
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis | 1-gen-2018 | Riva, Beatrice; Griglio, Alessia; Serafini, Marta; CORDERO SANCHEZ, Celia; Aprile, Silvio; Di Paola, Rosanna; Gugliandolo, Enrico; Alansary, Dalia; Biocotino, Isabella; Lim, Dmitry; Grosa, Giorgio; Galli, Ubaldina; Niemeyer, Barbara; Sorba, Giovanni; Canonico, Pier Luigi; Cuzzocrea, Salvatore; Genazzani, Armando; Pirali, Tracey | |
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs | 1-gen-2017 | Pirali, Tracey; Ciraolo, Elisa; Aprile, Silvio; Massarotti, Alberto; Berndt, Alex; Griglio, Alessia; Serafini, Marta; Mercalli, Valentina; Landoni, Clarissa; Campa, Carlo Cosimo; Margaria, Jean Piero; Silva, Rangel L.; Grosa, Giorgio; Sorba, Giovanni; Williams, Roger; Hirsch, Emilio; Tron, Gian Cesare | |
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity | 1-gen-2017 | Travelli, Cristina; Aprile, Silvio; Rahimian, Reza; Grolla, Ambra A.; Rogati, Federica; Bertolotti, Mattia; Malagnino, Floriana; Di Paola, Rosanna; Impellizzeri, Daniela; Fusco, Roberta; Mercalli, Valentina; Massarotti, Alberto; Stortini, Giorgio; Terrazzino, Salvatore; DEL GROSSO, Erika; Fakhfouri, Gohar; Troiani, Maria Pia; Alisi, Maria Alessandra; Grosa, Giorgio; Sorba, Giovanni; Canonico, Pier Luigi; Orsomando, Giuseppe; Cuzzocrea, Salvatore; Genazzani, Armando; Galli, Ubaldina; Tron, Gian Cesare | |
In silico-driven multicomponent synthesis of 4,5- and 1,5-disubstituted imidazoles as indoleamine 2,3-dioxygenase inhibitors | 1-gen-2016 | Fallarini, Silvia; Massarotti, Alberto; Gesù, A.; Giovarruscio, Sara; Coda Zabetta, G.; Bergo, R.; Giannelli, B.; Brunco, A.; Lombardi, Grazia; Sorba, Giovanni; Pirali, Tracey | |
Design, synthesis, and biological evaluation of combretabenzodiazepines: a novel class of anti-tubulin agents | 1-gen-2015 | Galli, Ubaldina; Travelli, Cristina; Aprile, Silvio; Arrigoni, Elena; Torretta, Simone; Grosa, Giorgio; Massarotti, Alberto; Sorba, Giovanni; Canonico, Pier Luigi; Genazzani, Armando; Tron, Gian Cesare | |
The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors | 1-gen-2015 | Galli, Ubaldina; Ciraolo, Elisa; Massarotti, Alberto; Margaria, Jean Piero; Sorba, Giovanni; Hirsch, Emilio; Tron, Gian Cesare | |
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups? | 1-gen-2014 | Massarotti, Alberto; Aprile, Silvio; Mercalli, Valentina; DEL GROSSO, Erika; Grosa, Giorgio; Sorba, Giovanni; Tron, Gian Cesare | |
ZINClick: A Database of 16 Million Novel, Patentable, and Readily Synthesizable 1,4-Disubstituted Triazoles | 1-gen-2014 | Massarotti, Alberto; A., Brunco; Sorba, Giovanni; Tron, Gian Cesare | |
Inhibitors of Nicotinamide Phosphoribosyltransferase, compositions, products and uses thereof. | 1-gen-2014 | Genazzani Armando, A.; Tron, Gian Cesare; Galli, Ubaldina; Travelli, Cristina; Cuzzocrea, Salvatore; Grosa, Giorgio; Sorba, Giovanni; Canonico Pier, Luigi | |
Capitolo 23. Istamina e agenti antistaminici | 1-gen-2014 | Sorba, Giovanni; Massarotti, Alberto | |
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus | 1-gen-2013 | Bassetto, M; De Burghgraeve, T; Delang, L; Massarotti, Alberto; Coluccia, A; Zonta, N; Gatti, V; Colombano, Giampiero; Sorba, Giovanni; Silvestri, R; Tron, Gian Cesare; Neyts, J; Leyssen, P; Brancale, A. | |
A Concise Synthesis of Pyrazole Analogues of Combretastatin A1 as Potent Antitubulin Agents | 1-gen-2013 | Zaninetti, Roberta; Cortese, Sv; Aprile, Silvio; Massarotti, Alberto; Canonico, Pier Luigi; Sorba, Giovanni; Grosa, Giorgio; Genazzani, Armando; Pirali, Tracey | |
“Synthesis and in vitro evaluation of tetrasubstituted pyridines as potential PI3Ks inhibitors” | 1-gen-2013 | Galli, Ubaldina; E., Ciraolo; E., Hirsch; Sorba, Giovanni; Tron, Gian Cesare | |
The tubulin colchicine domain: a molecular modelling perspective | 1-gen-2012 | Massarotti, A; Coluccia, A; Silvestri, R; Sorba, G; Brancale, A | |
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2 | 1-gen-2012 | Galli, Ubaldina; Mesenzani, Ornella; Coppo, C; Sorba, Giovanni; Canonico, Pier Luigi; Tron, Gian Cesare; Genazzani, Armando | |
De novo computer-aided design of novel antiviral agents | 1-gen-2012 | Massarotti, Alberto; Coluccia, A; Sorba, Giovanni; Silvestri, R; Brancale, A. | |
Quinolin-4 (1h) -one derivatives as inhibitors of phosphatidylinositol 3-kinases | 1-gen-2012 | Sorba, Giovanni; Tron, Gian Cesare; Galli, Ubaldina; Massarotti, Alberto; Hirsch, E; Ciraolo, E; Pirali, Tracey |
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